FI932446A7 - 2b,19-metyleeniaminosillan sisältäviä steroideja aromataasi-inhibiitto reina - Google Patents

2b,19-metyleeniaminosillan sisältäviä steroideja aromataasi-inhibiitto reina Download PDF

Info

Publication number
FI932446A7
FI932446A7 FI932446A FI932446A FI932446A7 FI 932446 A7 FI932446 A7 FI 932446A7 FI 932446 A FI932446 A FI 932446A FI 932446 A FI932446 A FI 932446A FI 932446 A7 FI932446 A7 FI 932446A7
Authority
FI
Finland
Prior art keywords
aromatase inhibition
methylene amino
steroids containing
amino bridge
bridge
Prior art date
Application number
FI932446A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI932446A0 (fi
FI932446L (fi
Inventor
John O'neal Johnston
Joseph Paul Burkhart
Norton P Peet
Original Assignee
Merrell Dow Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma
Publication of FI932446A0 publication Critical patent/FI932446A0/fi
Publication of FI932446L publication Critical patent/FI932446L/fi
Publication of FI932446A7 publication Critical patent/FI932446A7/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036—Nitrogen-containing hetero ring
    • C07J71/0042—Nitrogen only
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
FI932446A 1990-11-30 1991-10-17 2b,19-metyleeniaminosillan sisältäviä steroideja aromataasi-inhibiitto reina FI932446A7 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/621,183 US5126488A (en) 1990-11-30 1990-11-30 2β,19-methyleneamino bridged steroids as aromatase inhibitors
PCT/US1991/007810 WO1992009619A1 (en) 1990-11-30 1991-11-17 2β,19-METHYLENEAMINO BRIDGED STEROIDS AS AROMATASE INHIBITORS

Publications (3)

Publication Number Publication Date
FI932446A0 FI932446A0 (fi) 1993-05-28
FI932446L FI932446L (fi) 1993-05-28
FI932446A7 true FI932446A7 (fi) 1993-05-28

Family

ID=24489088

Family Applications (1)

Application Number Title Priority Date Filing Date
FI932446A FI932446A7 (fi) 1990-11-30 1991-10-17 2b,19-metyleeniaminosillan sisältäviä steroideja aromataasi-inhibiitto reina

Country Status (15)

Country Link
US (1) US5126488A (enExample)
EP (1) EP0559706B1 (enExample)
JP (1) JP3021651B2 (enExample)
KR (1) KR100200462B1 (enExample)
AT (1) ATE154606T1 (enExample)
AU (1) AU647226B2 (enExample)
CA (1) CA2096020C (enExample)
DE (1) DE69126622T2 (enExample)
DK (1) DK0559706T3 (enExample)
ES (1) ES2104736T3 (enExample)
FI (1) FI932446A7 (enExample)
GR (1) GR3024298T3 (enExample)
HU (1) HU213608B (enExample)
NO (1) NO302123B1 (enExample)
WO (1) WO1992009619A1 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5510340A (en) * 1992-06-12 1996-04-23 Sri International Antihypercholesterolemic compounds and related pharmaceutical compositions and methods of use
ATE473759T1 (de) 1998-05-22 2010-07-15 Univ Leland Stanford Junior Bifunktionelle moleküle sowie darauf basierende therapien.
EP3827747A1 (en) 2005-04-28 2021-06-02 Otsuka Pharmaceutical Co., Ltd. Pharma-informatics system
US9062126B2 (en) 2005-09-16 2015-06-23 Raptor Pharmaceuticals Inc. Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
DK3395372T3 (da) 2009-02-20 2022-04-19 Enhanx Biopharm Inc System til afgivelse af glutathion-baseret medikament
CN110075069A (zh) 2009-05-06 2019-08-02 实验室护肤股份有限公司 包含活性剂-磷酸钙颗粒复合物的皮肤递送组合物及其应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4322416A (en) * 1980-06-27 1982-03-30 Merrell Dow Pharmaceuticals Inc. 10-Alkynyl steroids
ZA9010082B (en) * 1989-12-20 1991-10-30 Merrell Dow Pharma 2,19-methyleneoxy and 2,19-methylenethio bridged steriods as aromatase and 19-hydroxylase inhibitors

Also Published As

Publication number Publication date
FI932446A0 (fi) 1993-05-28
CA2096020A1 (en) 1992-05-31
ATE154606T1 (de) 1997-07-15
AU647226B2 (en) 1994-03-17
KR100200462B1 (ko) 1999-06-15
DK0559706T3 (da) 1997-09-08
WO1992009619A1 (en) 1992-06-11
JP3021651B2 (ja) 2000-03-15
ES2104736T3 (es) 1997-10-16
EP0559706B1 (en) 1997-06-18
CA2096020C (en) 2003-06-17
EP0559706A4 (enExample) 1994-02-09
FI932446L (fi) 1993-05-28
US5126488A (en) 1992-06-30
NO931951L (no) 1993-05-28
EP0559706A1 (en) 1993-09-15
NO931951D0 (no) 1993-05-28
HUT64365A (en) 1993-12-28
GR3024298T3 (en) 1997-10-31
AU9027991A (en) 1992-06-25
DE69126622T2 (de) 1997-10-23
DE69126622D1 (de) 1997-07-24
JPH06509543A (ja) 1994-10-27
HU213608B (en) 1997-08-28
NO302123B1 (no) 1998-01-26

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