FI883838A - ESTRAR OCH AMIDER AV CARBOCYCLISKA SYROR OCH CYCLISKA ALCOHOL SAMT AMINER. - Google Patents
ESTRAR OCH AMIDER AV CARBOCYCLISKA SYROR OCH CYCLISKA ALCOHOL SAMT AMINER. Download PDFInfo
- Publication number
- FI883838A FI883838A FI883838A FI883838A FI883838A FI 883838 A FI883838 A FI 883838A FI 883838 A FI883838 A FI 883838A FI 883838 A FI883838 A FI 883838A FI 883838 A FI883838 A FI 883838A
- Authority
- FI
- Finland
- Prior art keywords
- och
- cycliska
- carbocycliska
- amider
- syror
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C61/00—Compounds having carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- C07D451/06—Oxygen atoms
- C07D451/12—Oxygen atoms acylated by aromatic or heteroaromatic carboxylic acids, e.g. cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/08—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions not involving the formation of amino groups, hydroxy groups or etherified or esterified hydroxy groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nutrition Science (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE3727733 | 1987-08-20 |
Publications (2)
Publication Number | Publication Date |
---|---|
FI883838A0 FI883838A0 (en) | 1988-08-18 |
FI883838A true FI883838A (en) | 1989-02-21 |
Family
ID=6334102
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI883838A FI883838A (en) | 1987-08-20 | 1988-08-18 | ESTRAR OCH AMIDER AV CARBOCYCLISKA SYROR OCH CYCLISKA ALCOHOL SAMT AMINER. |
Country Status (17)
Country | Link |
---|---|
JP (1) | JPS6471874A (en) |
KR (1) | KR950000509B1 (en) |
AU (1) | AU2110588A (en) |
DE (1) | DE3827253A1 (en) |
DK (1) | DK465188A (en) |
FI (1) | FI883838A (en) |
FR (1) | FR2619565A1 (en) |
GB (1) | GB2208862A (en) |
GR (1) | GR880100538A (en) |
IL (1) | IL87489A0 (en) |
IT (1) | IT1226742B (en) |
LU (1) | LU87314A1 (en) |
NL (1) | NL8802059A (en) |
PL (1) | PL274318A1 (en) |
PT (1) | PT88296B (en) |
SE (1) | SE8802926L (en) |
ZA (1) | ZA886180B (en) |
Families Citing this family (32)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1990012569A1 (en) | 1989-04-21 | 1990-11-01 | Sandoz Ag | Therapeutic use of 5-ht3 receptor antagonists |
US5225419A (en) * | 1989-10-14 | 1993-07-06 | John Wyeth & Brother, Limited | Certain 1,8-ethano or propano-1,4-dihydro-4-oxo-quinoline-3-carboxamides and derivatives thereof |
GB2236751B (en) * | 1989-10-14 | 1993-04-28 | Wyeth John & Brother Ltd | Heterocyclic compounds |
US5187166A (en) * | 1990-07-31 | 1993-02-16 | Nisshin Flour Milling Co., Ltd. | Azabicyclo derivatives and their use as antiemetics |
US5143923B1 (en) * | 1991-04-29 | 1993-11-02 | Hoechst-Roussel Pharmaceuticals Incorporated | Benzoisothiazole-and benzisoxazole-3-carboxamides |
US5225412A (en) * | 1991-04-29 | 1993-07-06 | Hoechst-Roussel Pharmaceuticals Incorporated | Benzoisothiazole-and benzisoxazole-3-carboxamides |
DE4126999A1 (en) * | 1991-08-16 | 1993-02-18 | Basf Ag | HERBICIDE AGENT, CONTAINING 3-AMINOBENZO (B) THIOPHENE AS ANTIDOTS |
US20100074949A1 (en) | 2008-08-13 | 2010-03-25 | William Rowe | Pharmaceutical composition and administration thereof |
DE10164139A1 (en) | 2001-12-27 | 2003-07-10 | Bayer Ag | 2-heteroaryl carboxamides |
CN101006076B (en) | 2004-06-24 | 2010-09-29 | 沃泰克斯药物股份有限公司 | Modulators of ATP-binding cassette transporters |
US8354427B2 (en) | 2004-06-24 | 2013-01-15 | Vertex Pharmaceutical Incorporated | Modulators of ATP-binding cassette transporters |
US7592461B2 (en) | 2005-12-21 | 2009-09-22 | Bristol-Myers Squibb Company | Indane modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
DK3219705T3 (en) | 2005-12-28 | 2020-04-14 | Vertex Pharma | PHARMACEUTICAL COMPOSITIONS OF THE AMORPHIC FORM OF N- [2,4-BIS (1,1-DIMETHYLETHYL) -5-HYDROXYPHENYL] -1,4-DIHYDRO-4-OXOQUINOLIN-3-CARBOXAMIDE |
EP2046753A2 (en) | 2006-07-06 | 2009-04-15 | Brystol-Myers Squibb Company | Pyridone/hydroxypyridine 11-beta hydroxysteroid dehydrogenase type i inhibitors |
NZ578744A (en) | 2007-01-31 | 2012-02-24 | Vertex Pharma | 2-aminopyridine derivatives useful as kinase inhibitors |
US8569337B2 (en) | 2008-07-23 | 2013-10-29 | Vertex Pharmaceuticals Incorporated | Tri-cyclic pyrazolopyridine kinase inhibitors |
NZ590784A (en) | 2008-07-23 | 2012-12-21 | Vertex Pharma | Pyrazolopyridine kinase inhibitors |
EP2328896B1 (en) | 2008-07-23 | 2013-10-23 | Vertex Pharmaceuticals Incorporated | Tri-cyclic pyrazolopyridine kinase inhibitors |
WO2010017350A1 (en) | 2008-08-06 | 2010-02-11 | Vertex Pharmaceuticals Incorporated | Aminopyridine kinase inhibitors |
KR20180011888A (en) | 2008-11-19 | 2018-02-02 | 포럼 파마슈티칼즈 인크. | Treatment of cognitive disorders with (r)-7-chloro-n-(quinuclidin-3-yl)benzo[b]thiophene-2-carboxamide and pharmaceutically acceptable salts thereof |
PT2408750E (en) | 2009-03-20 | 2015-10-15 | Vertex Pharma | Process for making modulators of cystic fibrosis transmembrane conductance regulator |
EP2427464A1 (en) | 2009-05-06 | 2012-03-14 | Vertex Pharmaceuticals Incorporated | Pyrazolopyridines |
AU2011209649A1 (en) | 2010-01-27 | 2012-08-09 | Vertex Pharmaceuticals Incorporated | Pyrazolopyrazine kinase inhibitors |
JP2013518114A (en) | 2010-01-27 | 2013-05-20 | バーテックス ファーマシューティカルズ インコーポレイテッド | Pyrazolopyrimidine kinase inhibitor |
JP5769733B2 (en) | 2010-01-27 | 2015-08-26 | バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated | Pyrazolopyridine kinase inhibitor |
RS54742B1 (en) | 2010-05-17 | 2016-10-31 | Forum Pharmaceuticals Inc | A crystalline form of (r)-7-chloro-n-(quinuclidin-3-yl)benzo[b]thiophene-2-carboxamide hydrochloride monohydrate |
US8802700B2 (en) | 2010-12-10 | 2014-08-12 | Vertex Pharmaceuticals Incorporated | Modulators of ATP-Binding Cassette transporters |
EP2819670A1 (en) | 2012-02-27 | 2015-01-07 | Vertex Pharmaceuticals Incorporated | Pharmaceutical composition and administration thereof |
WO2013169646A1 (en) | 2012-05-08 | 2013-11-14 | Envivo Pharmaceuticals, Inc. | Methods of maintaining, treating or improving cognitive function |
RU2749213C2 (en) | 2014-10-07 | 2021-06-07 | Вертекс Фармасьютикалз Инкорпорейтед | Co-crystals of transmembrane conduction regulator modulators in cystic fibrosis |
GB201511382D0 (en) | 2015-06-29 | 2015-08-12 | Imp Innovations Ltd | Novel compounds and their use in therapy |
CA3158150A1 (en) | 2019-10-18 | 2021-04-22 | The Regents Of The University Of California | 3-phenylsulphonyl-quinoline derivatives as agents for treating pathogenic blood vessels disorders |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3368061D1 (en) * | 1982-05-11 | 1987-01-15 | Beecham Group Plc | Azabicycloalkane derivatives, their preparation and medicaments containing them |
FI74707C (en) * | 1982-06-29 | 1988-03-10 | Sandoz Ag | FOERFARANDE FOER FRAMSTAELLNING AV TERAPEUTISKT ANVAENDBARA ALKYLENOEVERBRYGGADE PIPERIDYLESTRAR ELLER -AMIDER AV BICYKLISKA KARBOXYLSYROR. |
DE3429830A1 (en) * | 1983-08-26 | 1985-03-07 | Sandoz-Patent-GmbH, 7850 Lörrach | AUTOMATIC CARBONIC ACID AND SULPHONIC ACID ESTERS OR AMIDES |
-
1988
- 1988-08-11 DE DE3827253A patent/DE3827253A1/en not_active Withdrawn
- 1988-08-16 GB GB8819438A patent/GB2208862A/en not_active Withdrawn
- 1988-08-16 FR FR8810975A patent/FR2619565A1/en not_active Withdrawn
- 1988-08-16 LU LU87314A patent/LU87314A1/en unknown
- 1988-08-18 FI FI883838A patent/FI883838A/en not_active IP Right Cessation
- 1988-08-18 AU AU21105/88A patent/AU2110588A/en not_active Abandoned
- 1988-08-18 DK DK465188A patent/DK465188A/en not_active Application Discontinuation
- 1988-08-18 PT PT88296A patent/PT88296B/en not_active IP Right Cessation
- 1988-08-18 SE SE8802926A patent/SE8802926L/en unknown
- 1988-08-18 IL IL87489A patent/IL87489A0/en unknown
- 1988-08-19 PL PL27431888A patent/PL274318A1/en unknown
- 1988-08-19 JP JP63207189A patent/JPS6471874A/en active Pending
- 1988-08-19 NL NL8802059A patent/NL8802059A/en not_active Application Discontinuation
- 1988-08-19 ZA ZA886180A patent/ZA886180B/en unknown
- 1988-08-19 IT IT8821719A patent/IT1226742B/en active
- 1988-08-19 KR KR1019880010957A patent/KR950000509B1/en not_active Application Discontinuation
- 1988-08-22 GR GR880100538A patent/GR880100538A/en unknown
Also Published As
Publication number | Publication date |
---|---|
DK465188A (en) | 1989-02-21 |
GB8819438D0 (en) | 1988-09-21 |
JPS6471874A (en) | 1989-03-16 |
FR2619565A1 (en) | 1989-02-24 |
SE8802926D0 (en) | 1988-08-18 |
IL87489A0 (en) | 1989-01-31 |
GR880100538A (en) | 1989-05-25 |
PT88296B (en) | 1995-03-31 |
KR950000509B1 (en) | 1995-01-24 |
DK465188D0 (en) | 1988-08-18 |
KR890003679A (en) | 1989-04-17 |
IT1226742B (en) | 1991-02-05 |
IT8821719A0 (en) | 1988-08-19 |
SE8802926L (en) | 1989-02-21 |
ZA886180B (en) | 1990-07-25 |
LU87314A1 (en) | 1989-03-08 |
AU2110588A (en) | 1989-03-23 |
NL8802059A (en) | 1989-03-16 |
GB2208862A (en) | 1989-04-19 |
PL274318A1 (en) | 1989-04-17 |
PT88296A (en) | 1989-06-30 |
FI883838A0 (en) | 1988-08-18 |
DE3827253A1 (en) | 1989-03-02 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM | Patent lapsed |
Owner name: SANDOZ AG |