FI831617A0 - Nya aziridin- och fenyletanolaminderivat - Google Patents
Nya aziridin- och fenyletanolaminderivatInfo
- Publication number
- FI831617A0 FI831617A0 FI831617A FI831617A FI831617A0 FI 831617 A0 FI831617 A0 FI 831617A0 FI 831617 A FI831617 A FI 831617A FI 831617 A FI831617 A FI 831617A FI 831617 A0 FI831617 A0 FI 831617A0
- Authority
- FI
- Finland
- Prior art keywords
- ananamin
- nya
- aziridin
- derivatives
- och
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
- C07D295/26—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D203/00—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom
- C07D203/04—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D203/06—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D203/08—Heterocyclic compounds containing three-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
- C07D295/135—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH301382 | 1982-05-14 | ||
| CH143483 | 1983-03-16 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FI831617A0 true FI831617A0 (fi) | 1983-05-10 |
| FI831617L FI831617L (fi) | 1983-11-15 |
Family
ID=25687635
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI831617A FI831617L (fi) | 1982-05-14 | 1983-05-10 | Nya aziridin- och fenyletanolaminderivat |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US4652679A (fi) |
| EP (1) | EP0094595B1 (fi) |
| AU (1) | AU1442483A (fi) |
| CA (1) | CA1219865A (fi) |
| DE (1) | DE3369130D1 (fi) |
| DK (1) | DK209383A (fi) |
| ES (1) | ES522403A0 (fi) |
| FI (1) | FI831617L (fi) |
| HU (1) | HU191523B (fi) |
| IL (1) | IL68635A (fi) |
| MC (1) | MC1516A1 (fi) |
| NO (1) | NO831727L (fi) |
| NZ (1) | NZ204177A (fi) |
| PT (1) | PT76688B (fi) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1258454A (en) * | 1982-08-10 | 1989-08-15 | Leo Alig | Phenethanolamines |
| CA1292747C (en) * | 1983-11-21 | 1991-12-03 | John Robert Carson | Aralykyl (arylethynyl) aralkyl amines and their use as vasodilators and antihypertensives |
| EP0305543B1 (en) * | 1987-03-12 | 1994-11-09 | Nippon Shokubai Kagaku Kogyo Co., Ltd | Process for producing aziridines |
| SI9111433B (sl) * | 1991-08-22 | 1999-02-28 | Pliva | Novi N-sulfonil-tetrahidro-/1,3/-dioksepino/5,6-b/azirini, postopek priprave, intermediati za njihovo pripravo in uporaba |
| US5321036A (en) * | 1993-02-10 | 1994-06-14 | Bristol-Myers Squibb Company | Thiazole and oxazole-based β3 adrenergic receptor agonists |
| DE4335718A1 (de) * | 1993-10-20 | 1995-04-27 | Merck Patent Gmbh | Cyclische Aminderivate |
| US5578638A (en) * | 1993-11-05 | 1996-11-26 | American Cyanamid Company | Treatment of glaucoma and ocular hypertension with β3 -adrenergic agonists |
| US5563171A (en) * | 1993-11-05 | 1996-10-08 | American Cyanamid Company | Treatment of glaucoma and ocular hypertension with β3-adrenergic agonists |
| EP0669335A1 (en) * | 1994-02-21 | 1995-08-30 | PLIVA, farmaceutska, kemijska, prehrambena i kozmeticka industrija, dionicko drustvo | N-sulfonyl-tetrahydro-[1,3]-dioxepino [5,6] azirines with hypoglycemic activity |
| ZA967892B (en) * | 1995-09-21 | 1998-03-18 | Lilly Co Eli | Selective β3 adrenergic agonists. |
| US6075040A (en) | 1996-09-05 | 2000-06-13 | Eli Lilly And Company | Selective β3 adrenergic agonists |
| ES2171839T3 (es) | 1996-09-05 | 2002-09-16 | Lilly Co Eli | Analogos de carbazol como agonistas adrenergicos selectivos de beta3. |
| CO5011072A1 (es) | 1997-12-05 | 2001-02-28 | Lilly Co Eli | Etanolaminas pirazinil substituidas como agfonistas de los receptores |
| US7812035B2 (en) | 2001-12-11 | 2010-10-12 | Sepracor Inc. | 4-substituted piperidines, and methods of use thereof |
Family Cites Families (36)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DD45721A (fi) * | ||||
| DE108532C (fi) * | ||||
| US3092636A (en) * | 1959-10-21 | 1963-06-04 | Upjohn Co | Alpha-[2-(1-alkyleneimino) ethylamino]-alkanophenones and the corresponding alcohols |
| US3732300A (en) * | 1966-09-23 | 1973-05-08 | Allen & Hanburys Ltd | Phenylaminoethanol derivatives |
| GB1200886A (en) * | 1966-09-23 | 1970-08-05 | Allen & Hanburys Ltd | Phenylaminoethanol derivatives |
| US3514465A (en) * | 1966-12-30 | 1970-05-26 | Degussa | Certain thiazolyl- and pyridinylaminoketones |
| DE1593836A1 (de) * | 1967-06-29 | 1971-08-19 | Degussa | Verfahren zur Herstellung von neuen Aminoketonen |
| DE1593837A1 (de) * | 1967-06-29 | 1970-10-29 | Degussa | Verfahren zur Herstellung von neuen Aminoketonen |
| US3867455A (en) * | 1970-06-02 | 1975-02-18 | Allen & Hanburys Ltd | Preparation of phenylaminoethanols |
| US3709913A (en) * | 1970-09-14 | 1973-01-09 | Smith Kline French Lab | N-thienylalkyl-beta-alkoxy-trifluoro-methylphenalkylamines |
| US3803173A (en) * | 1971-04-26 | 1974-04-09 | Degussa | 3-(3-(1-(4-hydroxyphenyl)-1-hydroxypropyl-(2)-amino)-propionyl)-thiophene |
| DD108532A1 (fi) * | 1973-02-15 | 1974-09-20 | ||
| CA1030146A (en) * | 1974-04-18 | 1978-04-25 | American Home Products Corporation | Thiophene ethanolamines |
| GB1540463A (en) * | 1976-10-07 | 1979-02-14 | Ici Ltd | Alkanolamine derivatives |
| GB1593651A (en) * | 1977-02-03 | 1981-07-22 | Allen & Hanburys Ltd | Amides |
| US4374149A (en) * | 1977-06-03 | 1983-02-15 | Sterling Drug Inc. | α-{[(Arylalkyl)amino]alkyl}-4-hydroxy-3-(lower-alkylsulfinyl)benzenemethanols |
| CA1147342A (en) * | 1977-10-12 | 1983-05-31 | Kazuo Imai | Process of producing novel phenylethanolamine derivatives |
| DE2965655D1 (en) * | 1978-06-28 | 1983-07-21 | Beecham Group Plc | Secondary amines, their preparation, pharmaceutical compositions containing them and their use |
| CA1142954A (en) * | 1978-07-03 | 1983-03-15 | Jack Mills | Phenethanolamines, compositions containing the same, and method for effecting weight control |
| IL57670A (en) * | 1978-07-03 | 1982-11-30 | Lilly Co Eli | Phenethanolamines,their preparation and pharmaceutical formulations comprising them |
| CA1145766A (en) * | 1978-07-03 | 1983-05-03 | Jack Mills | Optically active phenethanolamines and method for increasing cardiac contractility |
| EP0023385B1 (en) * | 1979-06-16 | 1982-12-15 | Beecham Group Plc | Ethanamine derivatives, their preparation and use in pharmaceutical compositions |
| ATE1899T1 (de) * | 1979-06-16 | 1982-12-15 | Beecham Group Plc | Sekundaere amine, ihre herstellung und verwendung in pharmazeutischen zusammensetzungen. |
| EP0025331B1 (en) * | 1979-09-06 | 1983-03-02 | Beecham Group Plc | Cinnamic acid derivatives, their preparation, and pharmaceutical compositions containing them |
| ATE2265T1 (de) * | 1979-10-25 | 1983-02-15 | Beecham Group Plc | Sekundaere amine, ihre herstellung und verwendung in pharmazeutischen zusammensetzungen. |
| EP0029320B1 (en) * | 1979-11-15 | 1985-07-10 | Beecham Group Plc | Secondary ethanol amines, their preparation and their use in pharmaceutical compositions |
| EP0040000B1 (en) * | 1980-05-08 | 1983-10-12 | Beecham Group Plc | Arylethanolamine derivatives, their preparation and use in pharmaceutical compositions |
| DE3162756D1 (en) * | 1980-05-22 | 1984-04-26 | Beecham Group Plc | Arylethanolamine derivatives, their preparation and use in pharmaceutical compositions |
| GB2084577B (en) * | 1980-09-26 | 1984-05-02 | Beecham Group Ltd | Secondary amines |
| IT1149846B (it) * | 1980-10-16 | 1986-12-10 | Blasinachim Spa | Processo per la sintesi di 1-ammino-3-p(b-metossi-etil)-fenosi-2-propanolo |
| GB2096988B (en) * | 1980-11-20 | 1984-08-01 | Beecham Group Ltd | Aromatic hydroxyamines |
| EP0068699A1 (en) * | 1981-06-22 | 1983-01-05 | Beecham Group Plc | Decahydroquinolyl benzamides, process for their preparation and pharmaceutical compositions containing them |
| US4379166A (en) * | 1981-08-03 | 1983-04-05 | Schering Corporation | Arylmethoxy-, arylmethylthio-, heteroarylmethoxy-, and heteroarylmethylthio-alkylaminoalcohols |
| DE3360426D1 (en) * | 1982-04-08 | 1985-08-29 | Beecham Group Plc | N-substituted derivatives of ethanol amine |
| EP0091749A3 (en) * | 1982-04-08 | 1984-12-05 | Beecham Group Plc | Ethanolamine derivatives, process for their preparation and pharmaceutical compositions containing them |
| CA1258454A (en) * | 1982-08-10 | 1989-08-15 | Leo Alig | Phenethanolamines |
-
1983
- 1983-05-04 CA CA000427392A patent/CA1219865A/en not_active Expired
- 1983-05-09 US US06/492,981 patent/US4652679A/en not_active Expired - Fee Related
- 1983-05-09 NZ NZ204177A patent/NZ204177A/en unknown
- 1983-05-09 IL IL68635A patent/IL68635A/xx unknown
- 1983-05-10 MC MC821634A patent/MC1516A1/xx unknown
- 1983-05-10 DK DK209383A patent/DK209383A/da not_active Application Discontinuation
- 1983-05-10 DE DE8383104589T patent/DE3369130D1/de not_active Expired
- 1983-05-10 FI FI831617A patent/FI831617L/fi not_active Application Discontinuation
- 1983-05-10 AU AU14424/83A patent/AU1442483A/en not_active Abandoned
- 1983-05-10 EP EP83104589A patent/EP0094595B1/de not_active Expired
- 1983-05-11 HU HU831627A patent/HU191523B/hu unknown
- 1983-05-13 ES ES522403A patent/ES522403A0/es active Granted
- 1983-05-13 NO NO831727A patent/NO831727L/no unknown
- 1983-05-13 PT PT76688A patent/PT76688B/pt unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL68635A0 (en) | 1983-09-30 |
| IL68635A (en) | 1986-10-31 |
| CA1219865A (en) | 1987-03-31 |
| EP0094595B1 (de) | 1987-01-14 |
| HU191523B (en) | 1987-03-30 |
| DE3369130D1 (en) | 1987-02-19 |
| ES8407004A1 (es) | 1984-08-16 |
| FI831617L (fi) | 1983-11-15 |
| MC1516A1 (fr) | 1984-02-10 |
| NO831727L (no) | 1983-11-15 |
| EP0094595A1 (de) | 1983-11-23 |
| NZ204177A (en) | 1986-04-11 |
| DK209383D0 (da) | 1983-05-10 |
| PT76688B (en) | 1986-03-27 |
| AU1442483A (en) | 1983-11-17 |
| ES522403A0 (es) | 1984-08-16 |
| US4652679A (en) | 1987-03-24 |
| DK209383A (da) | 1983-11-15 |
| PT76688A (en) | 1983-06-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD | Application lapsed |
Owner name: F. HOFFMANN-LA ROCHE & CO. |