FI763613A - PROCEDURE FOR THE FRAMSTATION OF 6,7-DIMETOXY-4-AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) QUINAZOLINE WITH BLODTRYCKSSAENKANDE VERKAN - Google Patents
PROCEDURE FOR THE FRAMSTATION OF 6,7-DIMETOXY-4-AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) QUINAZOLINE WITH BLODTRYCKSSAENKANDE VERKANInfo
- Publication number
- FI763613A FI763613A FI763613A FI763613A FI763613A FI 763613 A FI763613 A FI 763613A FI 763613 A FI763613 A FI 763613A FI 763613 A FI763613 A FI 763613A FI 763613 A FI763613 A FI 763613A
- Authority
- FI
- Finland
- Prior art keywords
- blodtryckssaenkande
- verkan
- framstation
- dimetoxy
- furoyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C331/00—Derivatives of thiocyanic acid or of isothiocyanic acid
- C07C331/16—Isothiocyanates
- C07C331/28—Isothiocyanates having isothiocyanate groups bound to carbon atoms of six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Furan Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Priority Applications (17)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FI763613A FI58125C (en) | 1976-12-15 | 1976-12-15 | PROCEDURE FOR FRAMSTATING AV 6,7-DIMETOXY-4-AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) QUINAZOLINE WITH BLODTRYCKSSAENKANDE VEKAN |
CH1438177A CH630625A5 (en) | 1976-12-15 | 1977-11-24 | Process for the preparation of antihypertensive 6,7-dimethoxy-4-amino-2-[4-(2-furoyl)-1-piperazinyl]quinazoline |
SE7713376A SE435284B (en) | 1976-12-15 | 1977-11-25 | PROCEDURE FOR PREPARING 6,7-DIMETOXY-4-AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) QUINOAZOLINE |
AT867277A AT358048B (en) | 1976-12-15 | 1977-12-05 | METHOD FOR PRODUCING 6,7-DIMETHOXY-4- -AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) CHINAZOLINE |
ZA00777223A ZA777223B (en) | 1976-12-15 | 1977-12-05 | Method for the production of 6,7-dimethoxy-4-amino-2-(4-(2-furoyl)-1-piperazinyl)quinazoline having an antihypertensive effect |
NL7713702A NL7713702A (en) | 1976-12-15 | 1977-12-11 | PROCESS FOR THE PREPARATION OF 6,7-DIMETHOXY- -4-AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) CHINAZOLINE THAT HAS ANTI-HYPERTENSIVE ACTION. |
NO774262A NO147244C (en) | 1976-12-15 | 1977-12-12 | PROCEDURE FOR PREPARING 6,7-DIMETOXY-4-AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) CHINAZOLINE |
HU77OA538A HU174047B (en) | 1976-12-15 | 1977-12-13 | Process for producing 6,7-dimethoxy-4-amino-2square bracket-4-bracket-2-furoyl-bracket closed-piperazinyl-square bracket closed-quinasoline of anti-hypertensive activity |
PL1977202899A PL106031B1 (en) | 1976-12-15 | 1977-12-13 | METHOD OF MANUFACTURING 6.7-DIMETOXY-4-AMINO-2- / 4- / 2-FUROYLO / -1-PIPERAZINE / CHINAZOLINE WITH AN PRESSURE ACTION |
DK558277A DK144972C (en) | 1976-12-15 | 1977-12-14 | METHOD FOR PREPARING 6,7-DIMETHOXY-4-AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) QUINAZOLINE |
DE19772755637 DE2755637A1 (en) | 1976-12-15 | 1977-12-14 | METHOD FOR PRODUCING BLOOD PRESSURE-REDUCING 6,7-DIMETHOXY-4-AMINO-2 CORNER CLAMP ON 4- (2-FUROYL) -1-PIPERAZINYL CORNER CLAMP TO CHINAZOLINE |
BE183424A BE861821A (en) | 1976-12-15 | 1977-12-14 | PROCESS FOR PREPARING 6,7-DIMETHOXY-4-AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) -QUINAZOLINE EXERCISING AN ANTIHYPERTENSIFY EFFECT |
SU772555247A SU753360A3 (en) | 1976-12-15 | 1977-12-14 | Method of preparing 6,7-dimethoxy-4-amino-2/4-(2-furoyl)-1-piperazinyl/-quinazoline |
CA293,065A CA1092117A (en) | 1976-12-15 | 1977-12-14 | Method for the production of 6,7-dimethoxy-4-amino-2- ¬4-(2-furoyl)-1-piperazinyl| quinazoline having an antihypertensive effect |
DD7700202666A DD133671A1 (en) | 1976-12-15 | 1977-12-15 | METHOD OF GENERATING 6,7-DIMETHOXY-4-AMINO-2-CORNER CLAUSE ON 4- (2-FUROYL) -1-PIPERAZINYL SQUARE BRACKET TO CHINAZOLIN |
JP15157077A JPS5387377A (en) | 1976-12-15 | 1977-12-15 | Method of producing 6*77dimethoxyy44aminoo22 *44*22furoyl**11piperazinyl*quinazoline |
CS778432A CS195347B2 (en) | 1976-12-15 | 1977-12-15 | Process for preparing antihypertensive 6,7-dimethoxy4-4-amino-2-/4-/2-furoyl/-1-piperazinyl/quinazoline |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FI763613A FI58125C (en) | 1976-12-15 | 1976-12-15 | PROCEDURE FOR FRAMSTATING AV 6,7-DIMETOXY-4-AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) QUINAZOLINE WITH BLODTRYCKSSAENKANDE VEKAN |
FI763613 | 1976-12-15 |
Publications (3)
Publication Number | Publication Date |
---|---|
FI763613A true FI763613A (en) | 1978-06-16 |
FI58125B FI58125B (en) | 1980-08-29 |
FI58125C FI58125C (en) | 1985-01-02 |
Family
ID=8510503
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI763613A FI58125C (en) | 1976-12-15 | 1976-12-15 | PROCEDURE FOR FRAMSTATING AV 6,7-DIMETOXY-4-AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) QUINAZOLINE WITH BLODTRYCKSSAENKANDE VEKAN |
Country Status (17)
Country | Link |
---|---|
JP (1) | JPS5387377A (en) |
AT (1) | AT358048B (en) |
BE (1) | BE861821A (en) |
CA (1) | CA1092117A (en) |
CH (1) | CH630625A5 (en) |
CS (1) | CS195347B2 (en) |
DD (1) | DD133671A1 (en) |
DE (1) | DE2755637A1 (en) |
DK (1) | DK144972C (en) |
FI (1) | FI58125C (en) |
HU (1) | HU174047B (en) |
NL (1) | NL7713702A (en) |
NO (1) | NO147244C (en) |
PL (1) | PL106031B1 (en) |
SE (1) | SE435284B (en) |
SU (1) | SU753360A3 (en) |
ZA (1) | ZA777223B (en) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FI67699C (en) * | 1979-01-31 | 1985-05-10 | Orion Yhtymae Oy | PROCEDURE FOR THE FRAMSTATION OF AV 6,7-DIMETOXY-4-AMINO-2- (4- (2-FUROYL) -1-PIPERAZINYL) QUINAZOLINE HYDROCHLORIDE WITH BLODTRYCKSSAENKANDE VERKAN |
EP3333166B1 (en) * | 2012-05-23 | 2019-11-06 | Nerviano Medical Sciences S.R.L. | Process for the preparation of n-[5-(3,5-difluoro-benzyl)-1h-indazol-3-yl]-4-(4-methyl-piperazin-1-yl)-2-(tetrahydro-pyran-4-ylamino)-benzamide |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3935213A (en) * | 1973-12-05 | 1976-01-27 | Pfizer Inc. | Process for hypotensive 4-amino-2-(piperazin-1-yl) quinazoline derivatives |
-
1976
- 1976-12-15 FI FI763613A patent/FI58125C/en not_active IP Right Cessation
-
1977
- 1977-11-24 CH CH1438177A patent/CH630625A5/en not_active IP Right Cessation
- 1977-11-25 SE SE7713376A patent/SE435284B/en not_active IP Right Cessation
- 1977-12-05 ZA ZA00777223A patent/ZA777223B/en unknown
- 1977-12-05 AT AT867277A patent/AT358048B/en not_active IP Right Cessation
- 1977-12-11 NL NL7713702A patent/NL7713702A/en not_active Application Discontinuation
- 1977-12-12 NO NO774262A patent/NO147244C/en unknown
- 1977-12-13 PL PL1977202899A patent/PL106031B1/en unknown
- 1977-12-13 HU HU77OA538A patent/HU174047B/en not_active IP Right Cessation
- 1977-12-14 DK DK558277A patent/DK144972C/en not_active IP Right Cessation
- 1977-12-14 SU SU772555247A patent/SU753360A3/en active
- 1977-12-14 BE BE183424A patent/BE861821A/en not_active IP Right Cessation
- 1977-12-14 DE DE19772755637 patent/DE2755637A1/en active Granted
- 1977-12-14 CA CA293,065A patent/CA1092117A/en not_active Expired
- 1977-12-15 CS CS778432A patent/CS195347B2/en unknown
- 1977-12-15 JP JP15157077A patent/JPS5387377A/en active Granted
- 1977-12-15 DD DD7700202666A patent/DD133671A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
NO774262L (en) | 1978-06-16 |
SE435284B (en) | 1984-09-17 |
DK144972B (en) | 1982-07-19 |
PL202899A1 (en) | 1978-08-28 |
JPS5387377A (en) | 1978-08-01 |
DE2755637A1 (en) | 1978-06-22 |
SU753360A3 (en) | 1980-07-30 |
ATA867277A (en) | 1980-01-15 |
JPS6225147B2 (en) | 1987-06-01 |
NL7713702A (en) | 1978-06-19 |
CH630625A5 (en) | 1982-06-30 |
CA1092117A (en) | 1980-12-23 |
NO147244C (en) | 1984-10-09 |
CS195347B2 (en) | 1980-01-31 |
FI58125B (en) | 1980-08-29 |
NO147244B (en) | 1982-11-22 |
ZA777223B (en) | 1978-09-27 |
DE2755637C2 (en) | 1987-09-24 |
DK558277A (en) | 1978-06-16 |
AT358048B (en) | 1980-08-11 |
DD133671A1 (en) | 1979-01-17 |
PL106031B1 (en) | 1979-11-30 |
FI58125C (en) | 1985-01-02 |
DK144972C (en) | 1988-08-29 |
SE7713376L (en) | 1978-06-16 |
HU174047B (en) | 1979-10-28 |
BE861821A (en) | 1978-03-31 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM | Patent lapsed |
Owner name: ORION-YHTYMAE OY |