FI56011C - Foerfarande foer framstaellning av 2-(1-piperazinyl)- eller 2-(4-alkyl-1-piperazinyl)-8-etyl-5,8-dihydro-5-oxopyrido (2,3-d)-pyrimidin-6-karboxylsyror - Google Patents

Foerfarande foer framstaellning av 2-(1-piperazinyl)- eller 2-(4-alkyl-1-piperazinyl)-8-etyl-5,8-dihydro-5-oxopyrido (2,3-d)-pyrimidin-6-karboxylsyror

Info

Publication number
FI56011C
FI56011C FI298/74A FI29874A FI56011C FI 56011 C FI56011 C FI 56011C FI 298/74 A FI298/74 A FI 298/74A FI 29874 A FI29874 A FI 29874A FI 56011 C FI56011 C FI 56011C
Authority
FI
Finland
Prior art keywords
piperazinyl
carboxylsyror
oxopyrido
eller
framstaellning
Prior art date
Application number
FI298/74A
Other languages
English (en)
Finnish (fi)
Other versions
FI56011B (fi
Inventor
Shinsaku Minami
Jun-Ichi Matsumoto
Kazuyo Kawaguchi
Shinsaku Mishio
Masanao Shimizu
Yoshiyuki Takase
Shinichi Nakamura
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP3845373A external-priority patent/JPS5546400B2/ja
Priority claimed from JP5654473A external-priority patent/JPS565753B2/ja
Priority claimed from JP6446473A external-priority patent/JPS565755B2/ja
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Publication of FI56011B publication Critical patent/FI56011B/fi
Application granted granted Critical
Publication of FI56011C publication Critical patent/FI56011C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI298/74A 1973-04-03 1974-02-04 Foerfarande foer framstaellning av 2-(1-piperazinyl)- eller 2-(4-alkyl-1-piperazinyl)-8-etyl-5,8-dihydro-5-oxopyrido (2,3-d)-pyrimidin-6-karboxylsyror FI56011C (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP3845373A JPS5546400B2 (de) 1973-04-03 1973-04-03
JP5654473A JPS565753B2 (de) 1973-05-21 1973-05-21
JP6446473A JPS565755B2 (de) 1973-06-07 1973-06-07

Publications (2)

Publication Number Publication Date
FI56011B FI56011B (fi) 1979-07-31
FI56011C true FI56011C (fi) 1979-11-12

Family

ID=27289838

Family Applications (1)

Application Number Title Priority Date Filing Date
FI298/74A FI56011C (fi) 1973-04-03 1974-02-04 Foerfarande foer framstaellning av 2-(1-piperazinyl)- eller 2-(4-alkyl-1-piperazinyl)-8-etyl-5,8-dihydro-5-oxopyrido (2,3-d)-pyrimidin-6-karboxylsyror

Country Status (11)

Country Link
AR (2) AR204003A1 (de)
AT (1) AT340931B (de)
CA (1) CA1066701A (de)
CH (1) CH593281A5 (de)
ES (1) ES424851A1 (de)
FI (1) FI56011C (de)
IE (1) IE39102B1 (de)
NL (1) NL186087C (de)
NO (1) NO142221C (de)
PH (2) PH10529A (de)
SE (1) SE416051B (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1209163B (it) * 1979-12-21 1989-07-10 Unibios S P A Trecate Novara Procedimento per la fabbricazione di: 6-alcossicarbonil-8-etil-5-oxo-5,8diidro-aperta par. quadrata 2,3-dchiusa par. quadrata-primidine 2-sostituite ed acidi libri corrispondenti.
CN104945420A (zh) 2009-06-29 2015-09-30 因塞特公司 作为pi3k抑制剂的嘧啶酮类
US8759359B2 (en) 2009-12-18 2014-06-24 Incyte Corporation Substituted heteroaryl fused derivatives as PI3K inhibitors
TW201130842A (en) 2009-12-18 2011-09-16 Incyte Corp Substituted fused aryl and heteroaryl derivatives as PI3K inhibitors
AR084366A1 (es) 2010-12-20 2013-05-08 Incyte Corp N-(1-(fenil sustituido)etil)-9h-purin-6-aminas como inhibidores de pi3k
HUE043703T2 (hu) 2011-09-02 2019-09-30 Incyte Holdings Corp Heterociklusos aminok PI3K inhibitorokként
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
US10077277B2 (en) 2014-06-11 2018-09-18 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
TWI764392B (zh) 2015-02-27 2022-05-11 美商英塞特公司 Pi3k抑制劑之鹽及製備方法
US9732097B2 (en) 2015-05-11 2017-08-15 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor
WO2016183063A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Crystalline forms of a pi3k inhibitor

Also Published As

Publication number Publication date
NL186087C (nl) 1990-09-17
FI56011B (fi) 1979-07-31
CH593281A5 (en) 1977-11-30
NO740349L (no) 1974-10-04
NL7401509A (de) 1974-10-07
IE39102B1 (en) 1978-08-02
PH10529A (en) 1977-05-30
PH10984A (en) 1977-10-18
AR204660A1 (es) 1976-02-20
NL186087B (nl) 1990-04-17
ES424851A1 (es) 1976-06-01
NO142221C (no) 1980-07-16
SE416051B (sv) 1980-11-24
NO142221B (no) 1980-04-08
ATA277774A (de) 1977-05-15
CA1066701A (en) 1979-11-20
IE39102L (en) 1974-10-03
AR204003A1 (es) 1975-11-12
AT340931B (de) 1978-01-10

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