FI50119B - - Google Patents

Info

Publication number
FI50119B
FI50119B FI659/69A FI65969A FI50119B FI 50119 B FI50119 B FI 50119B FI 659/69 A FI659/69 A FI 659/69A FI 65969 A FI65969 A FI 65969A FI 50119 B FI50119 B FI 50119B
Authority
FI
Finland
Application number
FI659/69A
Other languages
Finnish (fi)
Other versions
FI50119C (fi
Inventor
Laszlo Beregi
Pierre Hugon
Michel Laubie
Original Assignee
Science Union & Cie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Science Union & Cie filed Critical Science Union & Cie
Publication of FI50119B publication Critical patent/FI50119B/fi
Application granted granted Critical
Publication of FI50119C publication Critical patent/FI50119C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/08Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
FI690659A 1968-03-06 1969-03-05 Menetelmä uusien terapeuttisesti tehokkaiden N-(3-sulfamyyli-4-kloorib entsamido)-indoliinijohdannaisten valmistamiseksi. FI50119C (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB00906/68A GB1203691A (en) 1968-03-06 1968-03-06 New disubstituted n-amino indoline derivatives and process for preparing them

Publications (2)

Publication Number Publication Date
FI50119B true FI50119B (https=) 1975-09-01
FI50119C FI50119C (fi) 1975-12-10

Family

ID=9976474

Family Applications (1)

Application Number Title Priority Date Filing Date
FI690659A FI50119C (fi) 1968-03-06 1969-03-05 Menetelmä uusien terapeuttisesti tehokkaiden N-(3-sulfamyyli-4-kloorib entsamido)-indoliinijohdannaisten valmistamiseksi.

Country Status (13)

Country Link
US (1) US3565911A (https=)
BE (1) BE728658A (https=)
CH (1) CH507940A (https=)
DE (1) DE1909180A1 (https=)
DK (1) DK126193B (https=)
ES (1) ES364421A1 (https=)
FI (1) FI50119C (https=)
FR (1) FR2003311A1 (https=)
GB (1) GB1203691A (https=)
IT (1) IT8049196A0 (https=)
NL (1) NL145226B (https=)
NO (1) NO128068B (https=)
SE (1) SE334887B (https=)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4112111A (en) * 1975-02-26 1978-09-05 Sandoz Ltd. Indolinylguanidines
IT1113879B (it) * 1979-03-15 1986-01-27 Farmatis Spa Derivato isoindolinico,processo per la sua preparazione e composizioni terapeutiche che lo comprendono come principio attivo
LU82949A1 (fr) * 1980-11-20 1981-06-04 Usv Pharma Corp Nouveaux amino-benzamides,leur procede de preparation et leur application au traitement de l'hypertension
DE3172386D1 (en) * 1980-12-22 1985-10-24 Usv Pharma Corp Synthesis of indolines
JPS57206657A (en) * 1981-06-16 1982-12-18 Mitsui Toatsu Chem Inc Sulfamoylbenzoic acid derivative and remedying composition containing said derivative as active component
FR2529785A1 (fr) * 1982-07-09 1984-01-13 Adir Composition pharmaceutique a base d'indapamide et de 8-(3-tertbutylamino 2-hydroxypropoxy)-thiachromanne
FR2663324B1 (fr) * 1990-06-14 1992-09-04 Adir Nouveau procede de preparation industrielle du 4-chloro 3-sulfamoyl n-(2,3-dihydro 2-methyl 1h-indol-1-yl) benzamide.
FR2663325B1 (fr) * 1990-06-14 1992-09-04 Adir Nouveau procede de preparation industrielle du 4-chloro 3-sulfamoyl n-(2,3-dihydro 2-methyl 1h-indol-1-yl) benzamide a partir de la 2,3-dihydro 2-methyl 1h-indole et de l'acide hydroxylamine-o-sulfonique.
FR2677886B1 (fr) * 1991-06-18 1995-03-31 Adir Comprime matriciel permettant la liberation prolongee d'indapamide apres administration par voie orale.
US5319096A (en) * 1992-04-03 1994-06-07 Hoechst-Roussel Pharmaceuticals Inc. (1H-indol-1-yl)-2-(amino) acetamides and related (1H-indol-1-yl)-(aminoalkyl)amides, pharmaceutical composition and use
IT1288123B1 (it) * 1996-09-04 1998-09-10 Nicox Sa Uso di nitroderivati per l'incontinenza urinaria
CA2495962A1 (en) 2002-08-19 2004-03-04 Pfizer Products Inc. Combination therapy for hyperproliferative diseases
US20060063803A1 (en) * 2004-09-23 2006-03-23 Pfizer Inc 4-Amino substituted-2-substituted-1,2,3,4-tetrahydroquinoline compounds
CA2574535A1 (en) * 2004-11-15 2006-05-26 Nitromed, Inc. Diuretic compounds comprising heterocyclic nitric oxide donor groups, compositions and methods of use
US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
CN101663262B (zh) 2006-12-01 2014-03-26 百时美施贵宝公司 用于治疗动脉粥样硬化和心血管疾病的作为cetp抑制剂的n-(3-苄基)-2,2-(二苯基)-丙-1胺衍生物
FR2924713B1 (fr) * 2007-12-11 2010-01-29 Servier Lab Nouveaux derives diazeniumdiolates, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
EP2575808A1 (en) 2010-05-28 2013-04-10 Mahmut Bilgic Combination of antihypertensive agents
MX2015014666A (es) 2013-04-17 2016-03-01 Pfizer Derivados de n-piperidin-3-ilbenzamida para tratar enfermedades cardiovasculares.
WO2016055901A1 (en) 2014-10-08 2016-04-14 Pfizer Inc. Substituted amide compounds
SG11202107614PA (en) 2019-01-18 2021-08-30 Astrazeneca Ab Pcsk9 inhibitors and methods of use thereof
TW202314018A (zh) * 2021-06-21 2023-04-01 荷蘭商Asm Ip私人控股有限公司 用於形成包含氧化銦鎵鋅的層之反應器系統及方法
EP4373474A1 (en) 2021-07-22 2024-05-29 KRKA, D.D., Novo Mesto Bilayer tablet comprising telmisartan and indapamide
EP4295839A1 (en) 2022-06-20 2023-12-27 KRKA, d.d., Novo mesto Combination of valsartan and indapamide
EP4374855A1 (en) 2022-11-22 2024-05-29 KRKA, D.D., Novo Mesto Pharmaceutical dosage form of candesartan and indapamide
EP4559899B1 (en) 2023-11-21 2026-04-01 KRKA, d.d., Novo mesto Synthesis of 1-amino-2-methyl-2,3-dihydroindole by nitrosating 2-methyl-2,3-dihydro-1h-indole and then reducing the obtained 1-nitroso-2-methyl-2,3-dihydroindole with thiourea dioxide

Also Published As

Publication number Publication date
US3565911A (en) 1971-02-23
NO128068B (https=) 1973-09-24
NL6903421A (https=) 1969-09-09
CH507940A (fr) 1971-05-31
IT8049196A0 (it) 1980-07-09
NL145226B (nl) 1975-03-17
FR2003311A1 (https=) 1969-11-07
DK126193B (da) 1973-06-18
SE334887B (https=) 1971-05-10
DE1909180A1 (de) 1970-07-02
BE728658A (https=) 1969-08-19
FI50119C (fi) 1975-12-10
GB1203691A (en) 1970-09-03
ES364421A1 (es) 1971-02-01

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