FI47487C - Uudet 3-asyyliamido-5-aryyli-1,3-dihydro-2H-1,4-bentsodiatsepiini-2-on it, jotka ovat välituotteita valmistettaessa vastaavia 3-amino-1,4-ben tsodiatsepiini-2-oneja. - Google Patents

Uudet 3-asyyliamido-5-aryyli-1,3-dihydro-2H-1,4-bentsodiatsepiini-2-on it, jotka ovat välituotteita valmistettaessa vastaavia 3-amino-1,4-ben tsodiatsepiini-2-oneja.

Info

Publication number
FI47487C
FI47487C FI642542A FI254264A FI47487C FI 47487 C FI47487 C FI 47487C FI 642542 A FI642542 A FI 642542A FI 254264 A FI254264 A FI 254264A FI 47487 C FI47487 C FI 47487C
Authority
FI
Finland
Prior art keywords
benzodiazepin
ones
acylamido
dihydro
intermediates
Prior art date
Application number
FI642542A
Other languages
English (en)
Swedish (sv)
Other versions
FI47487B (fi
Inventor
Childress
Bell
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Prod filed Critical American Home Prod
Priority to FI237372A priority Critical patent/FI49042C/fi
Priority to FI97473A priority patent/FI49618C/fi
Publication of FI47487B publication Critical patent/FI47487B/fi
Application granted granted Critical
Publication of FI47487C publication Critical patent/FI47487C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Furan Compounds (AREA)
  • Pyridine Compounds (AREA)
FI642542A 1963-12-03 1964-12-02 Uudet 3-asyyliamido-5-aryyli-1,3-dihydro-2H-1,4-bentsodiatsepiini-2-on it, jotka ovat välituotteita valmistettaessa vastaavia 3-amino-1,4-ben tsodiatsepiini-2-oneja. FI47487C (fi)

Priority Applications (2)

Application Number Priority Date Filing Date Title
FI237372A FI49042C (fi) 1963-12-03 1972-08-28 Menetelmä 3-amino-5-aryyli-1,3-dihydro-2H-1,4-bentsodiatsepiini-2-onie n valmistamiseksi.
FI97473A FI49618C (fi) 1963-12-03 1973-03-29 Menetelmä uusien 3-asyyliamido-5-aryyli-1,3-dihydro-2H-1,4-bentsodiats epiini-2-onien valmistamiseksi, jotka ovat välituotteita valmistettaes sa vastaavia 3-amino-5-aryyli-1,3-dihydro-2H-1,4-bentsodiatsepiini-2-o neja.

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32767463A 1963-12-03 1963-12-03
US414583A US3344136A (en) 1963-12-03 1964-11-30 Process for producing 3-acetamido-1, 3-dihydro-5-phenyl-2h-1, 4-benzodiazepin-2-ones

Publications (2)

Publication Number Publication Date
FI47487B FI47487B (fi) 1973-08-31
FI47487C true FI47487C (fi) 1973-12-10

Family

ID=26986000

Family Applications (1)

Application Number Title Priority Date Filing Date
FI642542A FI47487C (fi) 1963-12-03 1964-12-02 Uudet 3-asyyliamido-5-aryyli-1,3-dihydro-2H-1,4-bentsodiatsepiini-2-on it, jotka ovat välituotteita valmistettaessa vastaavia 3-amino-1,4-ben tsodiatsepiini-2-oneja.

Country Status (12)

Country Link
US (1) US3344136A (fi)
BE (1) BE656606A (fi)
BR (1) BR6464985D0 (fi)
CH (1) CH451173A (fi)
DE (2) DE1645920A1 (fi)
DK (1) DK120492B (fi)
FI (1) FI47487C (fi)
GB (2) GB1082213A (fi)
IL (1) IL22545A (fi)
IT (1) IT1044774B (fi)
NL (2) NL6414066A (fi)
SE (2) SE316187B (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3423459A (en) * 1966-04-19 1969-01-21 American Home Prod Acetanilido derivatives and method for preparing same
US3903103A (en) * 1971-09-15 1975-09-02 Upjohn Co 4-Amino-s-triazolo-{8 4,3-a{9 {8 1,4{9 benzodiazepine
CA1332410C (en) * 1984-06-26 1994-10-11 Roger M. Freidinger Benzodiazepine analogs
US4820834A (en) * 1984-06-26 1989-04-11 Merck & Co., Inc. Benzodiazepine analogs
US4628084A (en) * 1986-01-02 1986-12-09 Merck & Co., Inc. Process for 3-acylamino benzodiazepines
US5428157A (en) * 1993-11-22 1995-06-27 Merck & Co., Inc. 3-acylaminobenzodiazepines
BR0314595A (pt) * 2002-09-20 2005-08-09 Arrow Therapeutics Ltd Uso de um derivado de benzodiazepina ou um sal farmaceuticamente aceitável deste, inalador ou nebulisador, produto, usos de um produto e de um composto ou sal farmaceuticamente aceitável deste, derivado de benzodiazepina, composto, e, composição farmacêutica
MX2008003369A (es) * 2005-09-19 2008-03-27 Arrow Therapeutics Ltd Derivados de benzodiazepina para tratar infeccion de hepatitis c.

Also Published As

Publication number Publication date
DK120492B (da) 1971-06-07
SE317978B (fi) 1969-12-01
BE656606A (fi)
FI47487B (fi) 1973-08-31
GB1082213A (en) 1967-09-06
DE1445467A1 (de) 1969-02-13
BR6464985D0 (pt) 1973-08-02
US3344136A (en) 1967-09-26
GB1082212A (en) 1967-09-06
IL22545A (en) 1968-09-26
NL6414066A (fi) 1965-06-04
NL134421C (fi)
DE1645920A1 (de) 1970-09-24
SE316187B (fi) 1969-10-20
IT1044774B (it) 1980-04-21
CH451173A (de) 1968-05-15

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