FI47192C - Tapa valmistaa kardiovaskulaarisesti vaikuttavia 2,7-dimorfoliino-4-am ino-6-aryyli-pteridiinejä. - Google Patents

Tapa valmistaa kardiovaskulaarisesti vaikuttavia 2,7-dimorfoliino-4-am ino-6-aryyli-pteridiinejä.

Info

Publication number
FI47192C
FI47192C FI660913A FI91366A FI47192C FI 47192 C FI47192 C FI 47192C FI 660913 A FI660913 A FI 660913A FI 91366 A FI91366 A FI 91366A FI 47192 C FI47192 C FI 47192C
Authority
FI
Finland
Prior art keywords
dimorpholino
pteridines
aryl
amino
preparation
Prior art date
Application number
FI660913A
Other languages
English (en)
Swedish (sv)
Other versions
FI47192B (fi
Inventor
Roch
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of FI47192B publication Critical patent/FI47192B/fi
Application granted granted Critical
Publication of FI47192C publication Critical patent/FI47192C/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D475/00Heterocyclic compounds containing pteridine ring systems
    • C07D475/06Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D475/00Heterocyclic compounds containing pteridine ring systems
    • C07D475/06Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4
    • C07D475/08Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4 with a nitrogen atom directly attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI660913A 1965-04-15 1966-04-07 Tapa valmistaa kardiovaskulaarisesti vaikuttavia 2,7-dimorfoliino-4-am ino-6-aryyli-pteridiinejä. FI47192C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DET0028408 1965-04-15
JP2360067 1967-04-18

Publications (2)

Publication Number Publication Date
FI47192B FI47192B (fi) 1973-07-02
FI47192C true FI47192C (fi) 1973-10-10

Family

ID=26000021

Family Applications (1)

Application Number Title Priority Date Filing Date
FI660913A FI47192C (fi) 1965-04-15 1966-04-07 Tapa valmistaa kardiovaskulaarisesti vaikuttavia 2,7-dimorfoliino-4-am ino-6-aryyli-pteridiinejä.

Country Status (10)

Country Link
US (1) US3475425A (fi)
BE (1) BE679537A (fi)
CH (1) CH468395A (fi)
DK (2) DK123981B (fi)
FI (1) FI47192C (fi)
FR (3) FR1485627A (fi)
GB (2) GB1130956A (fi)
IE (1) IE32453B1 (fi)
NL (3) NL6605126A (fi)
SE (2) SE324575B (fi)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7276506B2 (en) * 1998-12-28 2007-10-02 4 Aza Bioscience Nv Immunosuppressive effects of pteridine derivatives
US6946465B2 (en) * 1999-02-02 2005-09-20 4 Aza Bioscience Nv Immunosuppressive effects of pteridine derivatives
DK1663244T3 (da) * 2003-09-12 2007-12-03 4 Aza Ip Nv Pteridin-derivater til behandling af TNF-alpha-beslægtede sygdomme
US20070032477A1 (en) * 2003-10-17 2007-02-08 Waer Mark J A Pteridine derivatives useful for making pharmaceutical compositions
US10144736B2 (en) * 2006-07-20 2018-12-04 Gilead Sciences, Inc. Substituted pteridines useful for the treatment and prevention of viral infections
CN107108615B (zh) 2015-03-04 2020-11-20 吉利德科学公司 Toll样受体调节性4,6-二氨基-吡啶并[3,2-D]嘧啶化合物
EP3507276B1 (en) 2016-09-02 2021-11-03 Gilead Sciences, Inc. Toll like receptor modulator compounds
US10640499B2 (en) 2016-09-02 2020-05-05 Gilead Sciences, Inc. Toll like receptor modulator compounds
TW202212339A (zh) 2019-04-17 2022-04-01 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TW202210480A (zh) 2019-04-17 2022-03-16 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TW202115056A (zh) 2019-06-28 2021-04-16 美商基利科學股份有限公司 類鐸受體調節劑化合物的製備方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1915334A (en) * 1930-10-16 1933-06-27 Du Pont Fluosilicate of organic heterocyclic bases and process of making it
US2075359A (en) * 1930-10-16 1937-03-30 Du Pont Insecticide
US2362614A (en) * 1940-03-11 1944-11-14 Jose B Calva Insecticides
US2940972A (en) * 1957-06-27 1960-06-14 Thomae Gmbh Dr K Tri-and tetra-substituted pteridine derivatives

Also Published As

Publication number Publication date
SE324575B (fi) 1970-06-08
FR1485627A (fr) 1967-06-23
FR5876M (fi) 1968-03-18
GB1130956A (en) 1968-10-16
SE334160B (fi) 1971-04-19
FI47192B (fi) 1973-07-02
GB1223461A (en) 1971-02-24
DK123981B (da) 1972-08-28
DK126254B (da) 1973-06-25
IE32453L (en) 1968-10-18
DE1620498A1 (de) 1970-06-25
CH468395A (de) 1969-02-15
FR328F (fi) 1970-10-05
NL131481C (fi)
IE32453B1 (en) 1973-08-08
NL6605126A (fi) 1966-10-17
US3475425A (en) 1969-10-28
NL6805515A (fi) 1968-10-21
BE679537A (fi) 1966-10-14

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