ES8600763A1 - Procedimiento de preparacion de nuevos derivados de guarnina. - Google Patents

Procedimiento de preparacion de nuevos derivados de guarnina.

Info

Publication number
ES8600763A1
ES8600763A1 ES533618A ES533618A ES8600763A1 ES 8600763 A1 ES8600763 A1 ES 8600763A1 ES 533618 A ES533618 A ES 533618A ES 533618 A ES533618 A ES 533618A ES 8600763 A1 ES8600763 A1 ES 8600763A1
Authority
ES
Spain
Prior art keywords
guanine
propoxymethyl
preparation
dihydroxy
application
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES533618A
Other languages
English (en)
Spanish (es)
Other versions
ES533618A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of ES533618A0 publication Critical patent/ES533618A0/es
Publication of ES8600763A1 publication Critical patent/ES8600763A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • C07F9/65616Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings containing the ring system having three or more than three double bonds between ring members or between ring members and non-ring members, e.g. purine or analogs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES533618A 1983-06-24 1984-06-22 Procedimiento de preparacion de nuevos derivados de guarnina. Expired ES8600763A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US50732883A 1983-06-24 1983-06-24
US61691084A 1984-06-06 1984-06-06

Publications (2)

Publication Number Publication Date
ES533618A0 ES533618A0 (es) 1985-10-16
ES8600763A1 true ES8600763A1 (es) 1985-10-16

Family

ID=27055802

Family Applications (1)

Application Number Title Priority Date Filing Date
ES533618A Expired ES8600763A1 (es) 1983-06-24 1984-06-22 Procedimiento de preparacion de nuevos derivados de guarnina.

Country Status (10)

Country Link
EP (1) EP0130126B1 (enExample)
AU (1) AU564194B2 (enExample)
CA (1) CA1225400A (enExample)
DE (1) DE3465596D1 (enExample)
DK (1) DK306184A (enExample)
ES (1) ES8600763A1 (enExample)
GR (1) GR82379B (enExample)
IL (1) IL72173A0 (enExample)
NZ (1) NZ208634A (enExample)
PT (1) PT78769A (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3571810D1 (en) * 1984-01-26 1989-08-31 Merck & Co Inc Substituted butyl guanines and their utilization in antiviral compositions
US4579849A (en) * 1984-04-06 1986-04-01 Merck & Co., Inc. N-alkylguanine acyclonucleosides as antiviral agents
MY101126A (en) * 1985-12-13 1991-07-31 Beecham Group Plc Novel compounds
CS264222B1 (en) * 1986-07-18 1989-06-13 Holy Antonin N-phosphonylmethoxyalkylderivatives of bases of pytimidine and purine and method of use them
US4966895A (en) * 1989-02-02 1990-10-30 Merck & Co. Inc. Cyclic monophosphates of purine and pyrimidine acyclonucleosides as anti-retroviral agents
US5216142A (en) * 1989-04-17 1993-06-01 Efamol Holdings Plc Anti-virals
AU2641192A (en) * 1991-09-24 1993-04-27 Wellcome Foundation Limited, The Therapeutic nucleosides
US6057305A (en) 1992-08-05 2000-05-02 Institute Of Organic Chemistry And Biochemistry Of The Academy Of Sciences Of The Czech Republic Antiretroviral enantiomeric nucleotide analogs
US5627185A (en) * 1994-11-23 1997-05-06 Gosselin; Gilles Acyclovir derivatives as antiviral agents

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ201662A (en) * 1981-08-26 1986-07-11 Merck & Co Inc 9-(1,3-(and 2,3)-dihydroxy-1-(and 2)-propoxy-methyl)guanine derivatives and methods for their preparation

Also Published As

Publication number Publication date
EP0130126A1 (en) 1985-01-02
DE3465596D1 (en) 1987-10-01
CA1225400A (en) 1987-08-11
DK306184A (da) 1984-12-25
AU2976384A (en) 1985-01-03
NZ208634A (en) 1988-02-29
EP0130126B1 (en) 1987-08-26
PT78769A (en) 1984-07-01
ES533618A0 (es) 1985-10-16
DK306184D0 (da) 1984-06-22
AU564194B2 (en) 1987-08-06
IL72173A0 (en) 1984-10-31
GR82379B (enExample) 1984-12-13

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