ES8600260A1 - Un procedimiento para preparar derivados de propinilaminotiazol - Google Patents
Un procedimiento para preparar derivados de propinilaminotiazolInfo
- Publication number
- ES8600260A1 ES8600260A1 ES527795A ES527795A ES8600260A1 ES 8600260 A1 ES8600260 A1 ES 8600260A1 ES 527795 A ES527795 A ES 527795A ES 527795 A ES527795 A ES 527795A ES 8600260 A1 ES8600260 A1 ES 8600260A1
- Authority
- ES
- Spain
- Prior art keywords
- derivatives
- propynylaminothiazole
- propynylamino
- thiazole
- microbial
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- HICLNPXFONCGNV-UHFFFAOYSA-N n-prop-1-ynyl-1,3-thiazol-2-amine Chemical class CC#CNC1=NC=CS1 HICLNPXFONCGNV-UHFFFAOYSA-N 0.000 title 1
- 230000000845 anti-microbial effect Effects 0.000 abstract 2
- 239000004480 active ingredient Substances 0.000 abstract 1
- 239000004599 antimicrobial Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- BKMDBXYRKHFLET-UHFFFAOYSA-N n-(3-iodoprop-2-ynyl)-1,3-thiazol-2-amine Chemical class IC#CCNC1=NC=CS1 BKMDBXYRKHFLET-UHFFFAOYSA-N 0.000 abstract 1
- LCCRDGYJMCVCDL-UHFFFAOYSA-N n-prop-2-ynyl-1,3-thiazol-2-amine Chemical compound C#CCNC1=NC=CS1 LCCRDGYJMCVCDL-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
PROCEDIMIENTO PARA PREPARAR DERIVADOS DE PROPINILAMINOTIAZOL.COMPRENDE SOMETER A UNA REACCION DE YODACCION A UN COMPUESTO DE FORMULA (II) PARA OBTENER DERIVADOS DE PROPINILAMINOTIAZOL DE FORMULA (I) DONDE R1 ES H, ALQUILO C 1 A 4, CARBOXI, FORMILO Y OTROS; R1 Y R2, CUANDO SE CONSIDERAN JUNTO CON LOS CARBONOS UNIDOS, SON UN ANILLO DE BENCENO CONDENSADO OPCIONALMENTE SUSTITUIDO CON 1 O 2 GRUPOS ELEGIDOS DEL GRUPO QUE CONSTA DE ALQUILO C 1 A 4 Y ALCOXI C 1 A 4; Y R3 ES H O ALQUILO C 1 A 4. LA REACCION SE REALIZA CON YODO Y EN UN COMPUESTO DE METAL ALCALINO, EN UN DISOLVENTE INERTE, A UNA TEMPERATURA AMBIENTE O BAJO ENFRIAMIENTO.TIENEN APLICACIONES MEDICO-AGRICOLAS CON SU COMPOSICION ANTIMICROBIANA.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP57225271A JPS59112978A (ja) | 1982-12-21 | 1982-12-21 | プロピニルアミノチアゾ−ル誘導体 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8600260A1 true ES8600260A1 (es) | 1985-10-01 |
| ES527795A0 ES527795A0 (es) | 1985-10-01 |
Family
ID=16826703
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES527795A Granted ES527795A0 (es) | 1982-12-21 | 1983-12-05 | Un procedimiento para preparar derivados de propinilaminotiazol |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US4535088A (es) |
| EP (1) | EP0111904A3 (es) |
| JP (1) | JPS59112978A (es) |
| KR (1) | KR880001049B1 (es) |
| AU (1) | AU565850B2 (es) |
| CA (1) | CA1212117A (es) |
| DK (1) | DK587283A (es) |
| ES (1) | ES527795A0 (es) |
| GB (1) | GB2132617B (es) |
| ZA (1) | ZA839037B (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8610432D0 (en) * | 1986-04-29 | 1986-06-04 | Akzo Nv | Amino-thiazole & oxazole derivatives |
| USRE34242E (en) * | 1986-04-29 | 1993-05-04 | Akzo N.V. | Amino-oxazole compounds having dopaminergic activity |
| CA2023176A1 (en) * | 1989-08-25 | 1991-02-26 | Margaret M. Bowers-Daines | Preparation and use of iodopropargyl esters of a-amino acid derivatives as antimicrobial agents |
| US5252745A (en) * | 1989-08-25 | 1993-10-12 | Rohm And Haas Company | Preparation and use of iodopropargyl esters of α-amino acid derivatives as antimicrobial agents |
| US5243055A (en) * | 1990-12-19 | 1993-09-07 | Givaudan Corporation | Heterocyclic formamidines useful as ultraviolet light absorbers |
| WO1994001423A1 (fr) * | 1992-07-07 | 1994-01-20 | Nippon Soda Co., Ltd. | Derive de thiazol |
| US20040176430A1 (en) * | 2002-11-21 | 2004-09-09 | Jeffrey Sterling | Propargyl-trifluoromethoxy-amino-benzothiazole derivatives |
| ZA200504988B (en) * | 2002-11-21 | 2006-08-30 | Teva Pharma | Propargyl-trifluoromethoxy-amino-benzothiazole derivatives |
| US20050197365A1 (en) * | 2004-02-27 | 2005-09-08 | Jeffrey Sterling | Diamino thiazoloindan derivatives and their use |
| WO2010012793A1 (en) * | 2008-08-01 | 2010-02-04 | Bayer Cropscience Sa | Fungicide aminothiazole derivatives |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3106553A (en) * | 1961-01-16 | 1963-10-08 | Miles Lab | Nu-2-propynyl alkylenediamines |
| BE754783A (fr) * | 1969-08-15 | 1971-02-12 | May & Baker Ltd | Derives thiazolyl a usage herbicide leur preparation et les compositions qui les contiennent |
| JPS4825494B1 (es) * | 1970-08-27 | 1973-07-30 | ||
| DE2206575A1 (de) * | 1971-02-26 | 1972-09-14 | Agripat S.A., Basel (Schweiz) | Schädlingsbekämpfungsmittel |
| US4378426A (en) * | 1981-11-12 | 1983-03-29 | Eastman Kodak Company | Photographic speed increasing and latent image stabilizing compounds, silver halide emulsions, and photographic elements |
-
1982
- 1982-12-21 JP JP57225271A patent/JPS59112978A/ja active Pending
-
1983
- 1983-12-02 US US06/557,365 patent/US4535088A/en not_active Expired - Lifetime
- 1983-12-05 ZA ZA839037A patent/ZA839037B/xx unknown
- 1983-12-05 ES ES527795A patent/ES527795A0/es active Granted
- 1983-12-06 AU AU22110/83A patent/AU565850B2/en not_active Ceased
- 1983-12-15 EP EP83112646A patent/EP0111904A3/en not_active Withdrawn
- 1983-12-20 DK DK587283A patent/DK587283A/da not_active Application Discontinuation
- 1983-12-21 CA CA000443876A patent/CA1212117A/en not_active Expired
- 1983-12-21 KR KR1019830006083A patent/KR880001049B1/ko not_active Expired
- 1983-12-21 GB GB08333982A patent/GB2132617B/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| GB8333982D0 (en) | 1984-02-01 |
| AU565850B2 (en) | 1987-10-01 |
| AU2211083A (en) | 1984-06-28 |
| DK587283A (da) | 1984-06-22 |
| KR880001049B1 (ko) | 1988-06-18 |
| EP0111904A2 (en) | 1984-06-27 |
| JPS59112978A (ja) | 1984-06-29 |
| KR840006982A (ko) | 1984-12-04 |
| ES527795A0 (es) | 1985-10-01 |
| DK587283D0 (da) | 1983-12-20 |
| GB2132617A (en) | 1984-07-11 |
| GB2132617B (en) | 1986-05-29 |
| CA1212117A (en) | 1986-09-30 |
| EP0111904A3 (en) | 1986-01-22 |
| ZA839037B (en) | 1984-07-25 |
| US4535088A (en) | 1985-08-13 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| ES8503344A1 (es) | Un procedimiento para preparar derivados de propinilaminoisoxazol | |
| ATE167357T1 (de) | Synergistische mikrobizide kombinationen | |
| BG60102B2 (bg) | Метод за получаване на 5-флуор-2(((4-циклопропил- метокси-2-пиридинил)метил)тионил)-1н-бензимидазол | |
| PL268927A1 (en) | Method of obtaining novel derivatives of benzimidazole | |
| EG17996A (en) | Benzimidazole derivative,process for its preparation,and insecticidal and/or acaricidal composition containing it as an active ingredient | |
| AU531878B2 (en) | Medicated animal feed based on liver meal | |
| EE9900428A (et) | Köhavastased ravimkoostised | |
| ES8600260A1 (es) | Un procedimiento para preparar derivados de propinilaminotiazol | |
| AU591046B2 (en) | Physiologically active agent for agricultural use | |
| DK0613368T3 (da) | Hudregenererende kosmetisk sammensætning | |
| GB2021409A (en) | Pharmaceutical composition | |
| ZA845682B (en) | Benzamidine derivatives having an antimicrobial activity process for their preparation and use as disinfectant drugs or preservatives | |
| IL67975A (en) | Derivatives of n,n-disubstituted azolecarboxamide and agricultural and horticultural fungicidal or nematicidal compositions containing same as active ingredient | |
| IT1229223B (it) | Composizioni veterinarie sinergisticamente attive e procedimento per la loro preparazione. | |
| ZA791765B (en) | New benzodioxole derivatives,processes for their preparation and their use as synergistic agents in insecticidal and acaricidal compositions | |
| PH14497A (en) | Fungicidal composition for agricultural use comprising 5-methyl-s-triazolo-(3,4-b)benzothiazole and method of use thereof | |
| DE3268609D1 (en) | Hair rinse composition | |
| HUT56692A (en) | Fungicidal composition comprising arylpropyl amines as active ingredient and process for preparing the active ingredients | |
| IL57058A (en) | Dichlorobenzodioxole derivatives,their preparation and their use as synergistic agents in insecticidal and acaricidal compositions | |
| IL61417A0 (en) | 2-(thi)oxo-1,3,2-oxazaphospholanes, their preparation and their use as synergistic agents in pesticidal compositions | |
| ES8407031A1 (es) | "procedimiento para la preparacion de n-(2-metil--5-cloro-fenil)-n-metoxiacetil-3-amino-1,3-oxazilidin-urea" | |
| FR2526432B1 (fr) | Derive de tetrahydrobenzothiazole et composition herbicide contenant celui-ci, a titre d'ingredient actif | |
| EP0132772A3 (en) | Fr-900216 substance obtainable by cultivating atcc 20577 for use as an active therapeutic substance and pharmaceutical antitumor composition comprising fr-900216 substance | |
| SU1697314A1 (ru) | Средство для профилактики спаечной болезни "изонидез" | |
| HUT41228A (en) | Microbicide compositions containing new 2,4-dichloro-5-nitro-thiazole as active ingredient and process for preparing the active substance |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19970519 |