ES8504743A1 - Un procedimiento para la preparacion de nuevos derivados de triazol - Google Patents

Un procedimiento para la preparacion de nuevos derivados de triazol

Info

Publication number
ES8504743A1
ES8504743A1 ES527232A ES527232A ES8504743A1 ES 8504743 A1 ES8504743 A1 ES 8504743A1 ES 527232 A ES527232 A ES 527232A ES 527232 A ES527232 A ES 527232A ES 8504743 A1 ES8504743 A1 ES 8504743A1
Authority
ES
Spain
Prior art keywords
alkyl
formula
triazolyl
aryl
bis
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES527232A
Other languages
English (en)
Other versions
ES527232A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp Belgium
Pfizer Corp
Original Assignee
Pfizer Corp Belgium
Pfizer Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp Belgium, Pfizer Corp filed Critical Pfizer Corp Belgium
Publication of ES8504743A1 publication Critical patent/ES8504743A1/es
Publication of ES527232A0 publication Critical patent/ES527232A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

PROCEDIMIENTO DE PREPARACION DE DERIVADOS DE TRIAZOL, DE FORMULA (I), O SUS SALES FARMACEUTICA O AGRICOLAMENTE ACEPTABLES, DONDE R ES FENILO, OPCIONALMENTE SUSTITUIDO O UN GRUPO 5-CLOROPIRID-2-ILO; Y X ES -NH2, -NH (ALQUILO C1-4), -N(ALQUILO C1-4)2 O -NHCOO (ALQUILO C1-4).SE OBTIENEN POR PREPARACION DE COMPUESTOS DE FORMULA (II), DONDE Q ES UN GRUPO SALIENTE COMO CL, BR, I, METANOSULFONILOXI, TRIFLUORMETANOSULFONILOXI O P-TOLUENSULFONILOXI, CON 1,2,4-TRIAZOL. EL PRODUCTO OBTENIDO RESPONDE A LA FORMULA (I) CON X IGUAL A NH2 Y PUEDE, OPCIONALMENTE, SOMETERSE A ALQUILACION, REACCION CON BASE FUERTE Y CLOROFORMIATO DE ALQUILO, O CONVERTIRSE EN SAL POR REACCION CON EL ACIDO ADECUADO.DE APLICACION COMO FUNGICIDAS AGRICOLAS Y PARA EL TRATAMIENTO DE INFECCIONES FUNGICAS EN LOS ANIMALES, INCLUIDO EL HOMBRE.
ES527232A 1982-11-16 1983-11-14 Un procedimiento para la preparacion de nuevos derivados de triazol Granted ES527232A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8232705 1982-11-16

Publications (2)

Publication Number Publication Date
ES8504743A1 true ES8504743A1 (es) 1985-05-01
ES527232A0 ES527232A0 (es) 1985-05-01

Family

ID=10534301

Family Applications (1)

Application Number Title Priority Date Filing Date
ES527232A Granted ES527232A0 (es) 1982-11-16 1983-11-14 Un procedimiento para la preparacion de nuevos derivados de triazol

Country Status (8)

Country Link
US (1) US4466974A (es)
EP (1) EP0113509B1 (es)
JP (1) JPS59104369A (es)
DE (1) DE3369986D1 (es)
DK (1) DK157928C (es)
ES (1) ES527232A0 (es)
GR (1) GR79071B (es)
IE (1) IE56258B1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE58738B1 (en) * 1984-09-05 1993-11-03 Ici Plc Antifungal azole compounds
US5252594A (en) * 1992-06-17 1993-10-12 Rohm And Haas Company Fungicidal (2-aryl-2-substituted)ethyl-1,2,4-triazoles
US5358939A (en) * 1992-06-25 1994-10-25 Rohm And Haas Company Fungicidal 2-aryl-2,2-disubstituted ethyl-1,2,4-triazoles
CN100451007C (zh) * 2006-10-12 2009-01-14 杭州宇龙化工有限公司 含芳醚双三氮唑类化合物及其用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2908378A1 (de) * 1979-03-03 1980-09-11 Hoechst Ag Derivate des 1,2,4-triazols
GB2078719B (en) * 1980-06-02 1984-04-26 Ici Ltd Heterocyclic compounds
CA1189857A (en) * 1981-03-27 1985-07-02 Janssen Pharmaceutica Naamloze Vennootschap Antimicrobial triazole derivatives
EP0069442B1 (en) * 1981-06-06 1985-02-20 Pfizer Limited Antifungal agents, processes for their preparation, and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
DK157928C (da) 1990-08-06
JPS6346071B2 (es) 1988-09-13
IE832677L (en) 1984-05-16
US4466974A (en) 1984-08-21
DK521683A (da) 1984-05-17
DK157928B (da) 1990-03-05
ES527232A0 (es) 1985-05-01
GR79071B (es) 1984-10-02
DK521683D0 (da) 1983-11-15
IE56258B1 (en) 1991-06-05
DE3369986D1 (en) 1987-04-09
JPS59104369A (ja) 1984-06-16
EP0113509B1 (en) 1987-03-04
EP0113509A3 (en) 1984-10-17
EP0113509A2 (en) 1984-07-18

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20040601