ES8404343A1 - Un procedimiento para la prepracion de nuevos derivados de 1,4-diaminociclitol. - Google Patents

Un procedimiento para la prepracion de nuevos derivados de 1,4-diaminociclitol.

Info

Publication number
ES8404343A1
ES8404343A1 ES520337A ES520337A ES8404343A1 ES 8404343 A1 ES8404343 A1 ES 8404343A1 ES 520337 A ES520337 A ES 520337A ES 520337 A ES520337 A ES 520337A ES 8404343 A1 ES8404343 A1 ES 8404343A1
Authority
ES
Spain
Prior art keywords
processes
preparation
pharmaceutical compositions
compositions containing
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES520337A
Other languages
English (en)
Other versions
ES520337A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fujisawa Pharmaceutical Co Ltd
Original Assignee
Fujisawa Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co Ltd filed Critical Fujisawa Pharmaceutical Co Ltd
Publication of ES8404343A1 publication Critical patent/ES8404343A1/es
Publication of ES520337A0 publication Critical patent/ES520337A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H5/00—Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium
    • C07H5/04—Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium to nitrogen
    • C07H5/06—Aminosugars
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/224—Cyclohexane rings substituted by at least two nitrogen atoms with only one saccharide radical directly attached to the cyclohexyl radical, e.g. destomycin, fortimicin, neamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Immunology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DE 1,4-DIAMINOCICLITOL Y DE SUS SALES FISIOLOGICAMENTE COMPATIBLES, DE FORMULA (I), EN LA QUE X, X Y X SON AMINO O AMINO PROTEGIDO; X ES HIDROGENO O HIDROXI; R ES HIDROGENO O ALQUILO INFERIOR; Y R PUEDE SER VARIOS RADICALES.CONSISTE EN LA REACCION DE ACILACION DE UN COMPUESTO DE FORMULA (II), O SU SAL, CON UN AGENTE DE ACILACION DE FORMULA ROH, O SU DERIVADO REACTIVO, FORMULAS EN LAS QUE TODOS LOS SIMBOLOS TIENEN EL MISMO SIGNIFICADO QUE EN LA FORMULA (I). LA REACCION SE EFECTUA EN UN DISOLVENTE INERTE, EN PRESENCIADE UNA BASE EVENTUALMENTE DE UN AGENTE CONDENSANTE, A TEMPERATURAS ENTRE 0JC Y 10JC.ESTOS COMPUESTOS TIENEN APLICACIONES FARMACOLOGICAS POR SU ACTIVIDAD ANTIMICROBIANA E INMUNO-ESTIMULANTE.
ES520337A 1982-03-05 1983-03-04 Un procedimiento para la prepracion de nuevos derivados de 1,4-diaminociclitol. Granted ES520337A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8206609 1982-03-05

Publications (2)

Publication Number Publication Date
ES8404343A1 true ES8404343A1 (es) 1984-04-16
ES520337A0 ES520337A0 (es) 1984-04-16

Family

ID=10528827

Family Applications (1)

Application Number Title Priority Date Filing Date
ES520337A Granted ES520337A0 (es) 1982-03-05 1983-03-04 Un procedimiento para la prepracion de nuevos derivados de 1,4-diaminociclitol.

Country Status (9)

Country Link
US (1) US4504472A (es)
EP (1) EP0088386B1 (es)
JP (2) JPS58164599A (es)
KR (1) KR900006212B1 (es)
AT (1) ATE21908T1 (es)
DE (1) DE3365781D1 (es)
DK (1) DK105183A (es)
ES (1) ES520337A0 (es)
IE (1) IE54288B1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6042394A (ja) * 1983-08-18 1985-03-06 Kowa Co 新規なアミノグリコシド及びその製法
IT1225484B (it) * 1987-11-27 1990-11-14 Pierrel Spa Procedimento di sintesi dell'amikacina

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4091032A (en) * 1976-09-23 1978-05-23 Abbott Laboratories 4-N-acylfortimicin B derivatives and the chemical conversion of fortimicin B to fortimicin A
JPS6011718B2 (ja) * 1976-09-23 1985-03-27 協和醗酵工業株式会社 新規なホ−テイマイシンｂの誘導体およびその製法
US4187297A (en) * 1977-12-21 1980-02-05 Abbott Laboratories 3-De-O-methyl-2-N-acyl and alkyl fortimicins A and B
US4276413A (en) * 1977-12-21 1981-06-30 Abbott Laboratories Fortimicin intermediates for producing 2-deoxyfortimicins
SE447386B (sv) * 1978-10-18 1986-11-10 Kowa Co Aminoglykosider, komposition innehallande dem samt forfarande for framstellning av dem
US4226980A (en) * 1978-12-07 1980-10-07 Abbott Laboratories Novel derivatives of fortimicin B and process for preparing same
US4251516A (en) * 1979-09-26 1981-02-17 Abbott Laboratories 2-Deoxy-3-O-Demethylfortimicins
US4360666A (en) * 1979-11-06 1982-11-23 Abbott Laboratories 2-Deoxyfortimicin A, 4-N-alkyl and 4-N-acyl-2-deoxyfortimicin B derivatives and intermediates therefor

Also Published As

Publication number Publication date
DE3365781D1 (en) 1986-10-09
US4504472A (en) 1985-03-12
JPS58164598A (ja) 1983-09-29
ES520337A0 (es) 1984-04-16
EP0088386A1 (en) 1983-09-14
EP0088386B1 (en) 1986-09-03
DK105183D0 (da) 1983-02-28
IE830399L (en) 1983-09-05
KR900006212B1 (ko) 1990-08-25
KR840004125A (ko) 1984-10-06
DK105183A (da) 1983-09-06
JPS58164599A (ja) 1983-09-29
IE54288B1 (en) 1989-08-16
ATE21908T1 (de) 1986-09-15

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