ES8206547A1 - Analogue of lincomycin and clindamycin - Google Patents

Analogue of lincomycin and clindamycin

Info

Publication number
ES8206547A1
ES8206547A1 ES507345A ES507345A ES8206547A1 ES 8206547 A1 ES8206547 A1 ES 8206547A1 ES 507345 A ES507345 A ES 507345A ES 507345 A ES507345 A ES 507345A ES 8206547 A1 ES8206547 A1 ES 8206547A1
Authority
ES
Spain
Prior art keywords
formula
lincomycin
clindamycin
analogue
lincosamide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES507345A
Other languages
Spanish (es)
Other versions
ES507345A0 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of ES507345A0 publication Critical patent/ES507345A0/en
Publication of ES8206547A1 publication Critical patent/ES8206547A1/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
    • C07H15/16—Lincomycin; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

PROCEDURE FOR OBTAINING ANALOGS OF LINCOMYCIN AND CLINDAMYCIN OF FORMULA (I), IN WHICH R1, R2 AND R3 MAY BE SEVERAL TYPES OF RADICALS. IT CONSISTS IN THE REACTION OF AN AMINO ACID OF FORMULA (II), IN WHICH R1 AND R3 HAVE THE SAME MEANING THAT IN FORMULA (I) AND IS VALUE OF 1 TO 4, WITH A DERIVATIVE OF A-LINCOSAMIDE, IN AN INERT ORGANIC SOLVENT, AT A TEMPERATURE BETWEEN 10 AND 100 C. THESE COMPOUNDS HAVE PHARMACOLOGICAL APPLICATIONS FOR THEIR ANTIBACTERIAL ACTIVITY (Machine-translation by Google Translate, not legally binding)
ES507345A 1979-11-23 1981-11-20 Analogue of lincomycin and clindamycin Expired ES8206547A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US9665279A 1979-11-23 1979-11-23

Publications (2)

Publication Number Publication Date
ES507345A0 ES507345A0 (en) 1982-09-01
ES8206547A1 true ES8206547A1 (en) 1982-09-01

Family

ID=22258400

Family Applications (2)

Application Number Title Priority Date Filing Date
ES507345A Expired ES8206547A1 (en) 1979-11-23 1981-11-20 Analogue of lincomycin and clindamycin
ES507346A Granted ES507346A0 (en) 1979-11-23 1981-11-20 PROCEDURE FOR THE PREPARATION OF NEW USEFUL ANALOGS OF LINCOMYCIN AND CLINDAMYCIN.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES507346A Granted ES507346A0 (en) 1979-11-23 1981-11-20 PROCEDURE FOR THE PREPARATION OF NEW USEFUL ANALOGS OF LINCOMYCIN AND CLINDAMYCIN.

Country Status (4)

Country Link
JP (2) JPS5687597A (en)
BE (1) BE886301A (en)
ES (2) ES8206547A1 (en)
ZA (1) ZA806438B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI0411537A (en) * 2003-06-17 2006-08-01 Vicuron Pharm Inc lincomycin derivatives that have antibacterial activity

Also Published As

Publication number Publication date
ZA806438B (en) 1981-10-28
JPH0141157B2 (en) 1989-09-04
ES8206548A1 (en) 1982-08-16
JPS63225392A (en) 1988-09-20
JPS6338037B2 (en) 1988-07-28
BE886301A (en) 1981-05-21
ES507346A0 (en) 1982-08-16
JPS5687597A (en) 1981-07-16
ES507345A0 (en) 1982-09-01

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Legal Events

Date Code Title Description
PC1A Transfer granted