ES8104274A1 - Procedimiento para la preparacion de 4-amino-1-(2-piridil) piperidinas - Google Patents

Procedimiento para la preparacion de 4-amino-1-(2-piridil) piperidinas

Info

Publication number
ES8104274A1
ES8104274A1 ES492484A ES492484A ES8104274A1 ES 8104274 A1 ES8104274 A1 ES 8104274A1 ES 492484 A ES492484 A ES 492484A ES 492484 A ES492484 A ES 492484A ES 8104274 A1 ES8104274 A1 ES 8104274A1
Authority
ES
Spain
Prior art keywords
group
preparation
anorectic
medicaments containing
amino piperidines
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES492484A
Other languages
English (en)
Other versions
ES492484A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
CM Industries SA
Clin Midy
Original Assignee
CM Industries SA
Clin Midy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by CM Industries SA, Clin Midy filed Critical CM Industries SA
Publication of ES492484A0 publication Critical patent/ES492484A0/es
Publication of ES8104274A1 publication Critical patent/ES8104274A1/es
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Obesity (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

PROCEDIMIENTO PARA LA PREPARACION DE 4-AMINO-1(2-PIRIDI)PIPERIDINAS, DE FORMULA (I), Y SUS SALES FARMACEUTICAMENTE ACEPTABLES, DONDE R REPRESENTA HIDROGENO, UN HALOGENO O DISTINTOS GRUPOS DE RADICALES. SE OBTIENE HACIENDO REACCIONAR UNA 2-HALOPIRIDINA DE FORMULA (II), CON UNA 4-AMINO-PIPERIDINA BLOQUEADA DE FORMULA (III), DONDE HAL REPRESENTA UN ATOMO DE HALOGENO X UN ATOMO DE HIDROGENO. DE ESTA FORMA SE OBTIENE (IV), QUE HIDROLIZANDOLO DA LUGAR AL COMPUESTO DESEADO. ESTE PREPARADO PRESENTA ACTIVIDAD ANOREXICA. *FORMULA*
ES492484A 1979-06-21 1980-06-16 Procedimiento para la preparacion de 4-amino-1-(2-piridil) piperidinas Expired ES8104274A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7915974A FR2459240A1 (fr) 1979-06-21 1979-06-21 Aminopiperidines anorexigenes, procede pour leur preparation, intermediaires dans ledit procede et medicaments qui les contiennent

Publications (2)

Publication Number Publication Date
ES492484A0 ES492484A0 (es) 1981-04-16
ES8104274A1 true ES8104274A1 (es) 1981-04-16

Family

ID=9226937

Family Applications (1)

Application Number Title Priority Date Filing Date
ES492484A Expired ES8104274A1 (es) 1979-06-21 1980-06-16 Procedimiento para la preparacion de 4-amino-1-(2-piridil) piperidinas

Country Status (9)

Country Link
US (1) US4409228A (es)
EP (2) EP0021973B1 (es)
JP (1) JPS5636481A (es)
AR (1) AR229088A1 (es)
AT (1) ATE4901T1 (es)
CA (1) CA1142936A (es)
DE (1) DE3061266D1 (es)
ES (1) ES8104274A1 (es)
FR (1) FR2459240A1 (es)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA848275B (en) * 1983-12-28 1985-08-28 Degussa New piridine-2-ethers or pyridine-2-thioethers having a nitrogen-containing cycloaliphatic ring
GB8710494D0 (en) * 1987-05-02 1987-06-03 Pfizer Ltd Antiarrhythmic agents
FR2674752B1 (fr) * 1991-09-03 1995-03-10 Sanofi Elf Utilisation de 4-amino-1-(2-pyridyl)piperidines pour la preparation de medicaments pour le traitement et la prophylaxie des etats decoulant d'un dysfonctionnement du systeme serotoninergique.
FR2674435B1 (fr) * 1991-03-27 1995-03-10 Sanofi Elf Utilisation de 4-amino-1-(2-pyridyl) piperidines pour la preparation d'agents psychotropes.
ATE175113T1 (de) * 1991-03-27 1999-01-15 Sanofi Sa Verwendung von 4-amino-1-(2-pyridyl)piperidinen als 5-ht3-agonisten zur behandlung und verhütung von serotoninergen dysfunktionen
FR2681785B1 (fr) * 1991-09-30 1995-05-24 Sanofi Elf Utilisation de 4-amino-1-(2-pyridyl)piperidines en tant qu'agents anticonvulsivants et antiepileptiques.
ATE219766T1 (de) * 1993-04-07 2002-07-15 Otsuka Pharma Co Ltd N-acylierte 4-aminopiperidin derivate als aktive bestandteile von peripher gefässerweiternden wikstoffen
US6632823B1 (en) * 1997-12-22 2003-10-14 Merck & Co., Inc. Substituted pyridine compounds useful as modulators of acetylcholine receptors
KR100713572B1 (ko) * 1999-05-21 2007-05-02 아보트 러보러터리즈 중추 신경계 제제로서 유용한 헤테로사이클릭 치환된 아미노아자사이클 및 이를 포함하는 약제학적 조성물
US6833370B1 (en) * 1999-05-21 2004-12-21 Abbott Laboratories Heterocycle substituted aminoazacycles useful as central nervous system agents
EP1428824A1 (en) * 1999-05-21 2004-06-16 Abbott Laboratories Heterocyclic substituted aminoazacycles useful as central nervous system agents
EP1235565B1 (en) * 1999-11-23 2005-12-28 Janssen Pharmaceutica N.V. Use of 5ht 3 agonists for relaxing the fundus
HUP0204496A3 (en) * 2000-01-20 2004-07-28 Eisai Co Ltd Novel piperidine compounds and pharmaceutical compositions containing the same and process for preparation the same
TW200738672A (en) * 2001-12-10 2007-10-16 Bristol Myers Squibb Co Intermediated for the preparation of 4,5-dihydro-pyrazolo [3,4-c] pyrid-2-ones
GT200500281A (es) 2004-10-22 2006-04-24 Novartis Ag Compuestos organicos.
PL2013211T3 (pl) 2006-04-21 2012-08-31 Novartis Ag Pochodne puryny do zastosowania jako agoniści receptora adenozyny A2A
CN102452978A (zh) * 2010-11-01 2012-05-16 重庆康丁医药技术有限公司 2-氯-取代或未取代脂族烃氧基吡啶及其制备方法
PL3646886T3 (pl) 2017-06-28 2024-03-04 Osaka University Leczenie bólu agonistą receptora serotoninowego 3

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE738495C (de) * 1941-08-10 1943-08-18 Kastel Tvornica Kemijsko Farma Verfahren zur Darstellung von substituierten 4-Aminopiperidinen

Also Published As

Publication number Publication date
ES492484A0 (es) 1981-04-16
FR2459240B1 (es) 1982-10-22
JPS5636481A (en) 1981-04-09
DE3061266D1 (en) 1983-01-13
AR229088A1 (es) 1983-06-15
EP0021973B1 (fr) 1982-12-08
CA1142936A (en) 1983-03-15
ATE4901T1 (de) 1983-10-15
FR2459240A1 (fr) 1981-01-09
EP0045980B1 (fr) 1983-10-05
EP0045980A1 (fr) 1982-02-17
EP0021973A2 (fr) 1981-01-07
EP0021973A3 (en) 1981-04-29
US4409228A (en) 1983-10-11

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