ES467482A1 - 1,2,6-thiadiazin-4-one derivatives - Google Patents
1,2,6-thiadiazin-4-one derivativesInfo
- Publication number
- ES467482A1 ES467482A1 ES467482A ES467482A ES467482A1 ES 467482 A1 ES467482 A1 ES 467482A1 ES 467482 A ES467482 A ES 467482A ES 467482 A ES467482 A ES 467482A ES 467482 A1 ES467482 A1 ES 467482A1
- Authority
- ES
- Spain
- Prior art keywords
- carbon atoms
- alcohol
- phenyl
- cyano
- nitro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/15—Six-membered rings
- C07D285/16—Thiadiazines; Hydrogenated thiadiazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Abstract
Procedure for the preparation of 1,2,6-thiadiszinones of the formula **(See formula)** wherein R1 represents a saturated or unsaturated, straight or branched chain, aliphatic radical with up to 12 carbon atoms, which may be substituted with 1-3 fluorine, chlorine or bromine atoms, with cyano, nitro, hydroxy groups, C 1-4 alkoxy, C 1-4 chloroalkoxy, C 1-4 alcoholylthio, C 3-6 cycloalkoxy, phenyl, a phenyl substituted with 1-3 halogen atoms, cyano, nitro, carboxy, carbamoyl, -CO-O (alcohol with 1-4 carbon atoms); phenoxy, (see formula), -CO-O (alcohol with 1-4 carbon atoms), tetrahydrofuryl, quinoline or 2,2-dimethyl-1,3-dioxolanyl; or a cycloalkoxy radical with 3-6 carbon atoms; or a phenyl radical which may be substituted with 1-3 halogen atoms and/or with alcohol with 1-4 carbon atoms, cycloalkoxy with 3-6 carbon atoms, alkoxy with 1-4 carbon atoms, alcoholylthio with 1- 4 carbon atoms, cyano, trifluoromethyl, formyl, 1-2 nitro, COR2 or phenyl groups; or -N = C (CH3) 2, or -CH (CN) -C6H5; or naphthyl; R2 alkoxy with 1-4 carbon atoms, hydroxy or -NR3R4; R3 and R4 hydrogen or alcohol with 1-4 carbon atoms; n 1 or 2, characterized in that the solution or suspension of 3,5-dichloro-1,2,6-thiadiazin-4-one in the alcohol R1OH is reacted, possibly with the addition of water, with an equivalent of a hydroxide, bicarbonate or carbonate of an alkali or alkaline earth metal, preferably with sodium or potassium hydroxide. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19762619090 DE2619090A1 (en) | 1976-05-03 | 1976-05-03 | 1.2.6-THIADIAZINONE, THEIR PRODUCTION AND USE |
Publications (1)
Publication Number | Publication Date |
---|---|
ES467482A1 true ES467482A1 (en) | 1978-10-16 |
Family
ID=5976731
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES458381A Expired ES458381A1 (en) | 1976-05-03 | 1977-05-02 | 1,2,6-thiadiazin-4-one derivatives |
ES467482A Expired ES467482A1 (en) | 1976-05-03 | 1978-03-03 | 1,2,6-thiadiazin-4-one derivatives |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES458381A Expired ES458381A1 (en) | 1976-05-03 | 1977-05-02 | 1,2,6-thiadiazin-4-one derivatives |
Country Status (14)
Country | Link |
---|---|
JP (1) | JPS52133995A (en) |
AT (1) | AT355036B (en) |
AU (1) | AU500386B2 (en) |
BE (1) | BE854184A (en) |
DE (1) | DE2619090A1 (en) |
ES (2) | ES458381A1 (en) |
FR (1) | FR2375223A1 (en) |
GB (1) | GB1577055A (en) |
HU (1) | HU176649B (en) |
IL (1) | IL51981A (en) |
IT (1) | IT1079620B (en) |
NL (1) | NL7704711A (en) |
SE (1) | SE7705086L (en) |
ZA (1) | ZA772643B (en) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4196284A (en) | 1977-03-30 | 1980-04-01 | Fmc Corporation | 5-Substituted-thio-3-chloro-4H-1,2,6-thiadiazin-4-ones |
US4097594A (en) * | 1977-03-30 | 1978-06-27 | Fmc Corporation | Mono-5-substituted-3-chloro-4H-1,2,6-thiadiazin-4-one antifungal agents |
US4201780A (en) | 1977-03-30 | 1980-05-06 | Fmc Corporation | Mono-5-substituted-3-chloro-4H-1,2,6-thiadiazin-4-one antifungal agents |
US4497807A (en) * | 1978-03-31 | 1985-02-05 | E. I. Du Pont De Nemours And Company | Thiadiazinone plant disease control agents |
US4143138A (en) | 1978-05-08 | 1979-03-06 | Fmc Corporation | 3-chloro-5-(optionally substituted heterocycloxy)-4h-1,2,6-thiadiazin-4-one antifungal agents |
ES2045545T3 (en) * | 1988-09-30 | 1994-01-16 | Ciba Geigy Ag | BIOCIDES FOR THE PROTECTION OF MATERIALS AND FOR AQUEOUS SYSTEMS. |
RU2624846C1 (en) * | 2016-10-10 | 2017-07-07 | федеральное государственное бюджетное учреждение "Федеральный научно-исследовательский центр эпидемиологии и микробиологии имени почетного академика Н.Ф. Гамалеи" Министерства здравоохранения Российской Федерации | Application of 4-(3-ethoxy-4-hydroxybenzyl)-5-oxo-5,6-dihydro-4h-[1,3,4]-thiadiazine-2-(2,4-difluorophenyl)-carboxamide to suppress infection, caused by antibiotic-resistant pseudomonas aeruginosa strains, and method of suppression of this infection |
-
1976
- 1976-05-03 DE DE19762619090 patent/DE2619090A1/en not_active Withdrawn
-
1977
- 1977-04-25 AT AT286877A patent/AT355036B/en not_active IP Right Cessation
- 1977-04-26 JP JP4832577A patent/JPS52133995A/en active Pending
- 1977-04-29 NL NL7704711A patent/NL7704711A/en not_active Application Discontinuation
- 1977-05-02 ES ES458381A patent/ES458381A1/en not_active Expired
- 1977-05-02 IT IT49225/77A patent/IT1079620B/en active
- 1977-05-02 IL IL51981A patent/IL51981A/en unknown
- 1977-05-02 BE BE177201A patent/BE854184A/en unknown
- 1977-05-02 GB GB18263/77A patent/GB1577055A/en not_active Expired
- 1977-05-02 HU HU77CE1129A patent/HU176649B/en unknown
- 1977-05-02 AU AU24770/77A patent/AU500386B2/en not_active Expired
- 1977-05-02 SE SE7705086A patent/SE7705086L/en not_active Application Discontinuation
- 1977-05-03 ZA ZA00772643A patent/ZA772643B/en unknown
- 1977-05-03 FR FR7713362A patent/FR2375223A1/en active Granted
-
1978
- 1978-03-03 ES ES467482A patent/ES467482A1/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
NL7704711A (en) | 1977-11-07 |
ZA772643B (en) | 1979-01-31 |
FR2375223A1 (en) | 1978-07-21 |
BE854184A (en) | 1977-11-03 |
AT355036B (en) | 1980-02-11 |
SE7705086L (en) | 1977-11-04 |
AU2477077A (en) | 1978-11-09 |
IL51981A (en) | 1981-07-31 |
HU176649B (en) | 1981-04-28 |
IT1079620B (en) | 1985-05-13 |
JPS52133995A (en) | 1977-11-09 |
ES458381A1 (en) | 1978-08-16 |
ATA286877A (en) | 1979-07-15 |
AU500386B2 (en) | 1979-05-17 |
FR2375223B1 (en) | 1979-05-11 |
GB1577055A (en) | 1980-10-15 |
DE2619090A1 (en) | 1977-11-17 |
IL51981A0 (en) | 1977-07-31 |
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