ES435403A1 - A procedure for the preparation of N- (1'-alylprolrolinin-2'-methyl) -2-metoxy-4,5-azimido-benzamine (Machine-translation by Google Translate, not legally binding)
- Google Patents
A procedure for the preparation of N- (1'-alylprolrolinin-2'-methyl) -2-metoxy-4,5-azimido-benzamine (Machine-translation by Google Translate, not legally binding)
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Societe dEtudes Scientifiques et Industrielles de lIle de France SA
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Societe dEtudes Scientifiques et Industrielles de lIle de France SA
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Publication of ES435403A1publicationCriticalpatent/ES435403A1/en
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Nitrogen Condensed Heterocyclic Rings
(AREA)
Abstract
A process for the preparation of N- (1-allylpyrrolidinyl-2-methyl) -2-methoxy-4,5-azimido-benzamide, as well as its pharmaceutically acceptable acid addition salts, its quaternary ammonium salts, and its isomers levorotatory and dextrorotatory, characterized by nitrating a compound of formula ** (see formula) ** Wherein x is a hydroxyl or alkoxy radical containing from 1 to 5 carbon atoms, r and r 'are hydrogen or an acyl radical, hydrogenate the nitrated compound in 5- formed, diazotize the obtained 5-diamine compound, and acidify by direct reaction of the 4,5-azimido compound thus obtained with l-allyl-2-aminomethylpyrrolidine, or by reaction of one of its activated derivatives. (Machine-translation by Google Translate, not legally binding)
ES0435403A1975-03-071975-03-07A procedure for the preparation of N- (1'-alylprolrolinin-2'-methyl) -2-metoxy-4,5-azimido-benzamine (Machine-translation by Google Translate, not legally binding)
ExpiredES435403A1
(en)
A procedure for the preparation of N- (1'-alylprolrolinin-2'-methyl) -2-metoxy-4,5-azimido-benzamine (Machine-translation by Google Translate, not legally binding)
A procedure for the preparation of N- (1'-alylprolrolinin-2'-methyl) -2-metoxy-4,5-azimido-benzamine (Machine-translation by Google Translate, not legally binding)
A procedure for the preparation of N- (1'-alylprolrolinin-2'-methyl) -2-metoxy-4,5-azimido-benzamine (Machine-translation by Google Translate, not legally binding)
A procedure for the preparation of N- (1'-alylprolrolinin-2'-methyl) -2-metoxy-4,5-azimido-benzamine (Machine-translation by Google Translate, not legally binding)
New procedure for the preparation of benz derivatives (f) indazol -4, 9-diona, with citostatic activity (Machine-translation by Google Translate, not legally binding)