ES427163A1 - Tertiary-alkylamino-lower acyl-xylidide local anesthetics - Google Patents
Tertiary-alkylamino-lower acyl-xylidide local anestheticsInfo
- Publication number
- ES427163A1 ES427163A1 ES427163A ES427163A ES427163A1 ES 427163 A1 ES427163 A1 ES 427163A1 ES 427163 A ES427163 A ES 427163A ES 427163 A ES427163 A ES 427163A ES 427163 A1 ES427163 A1 ES 427163A1
- Authority
- ES
- Spain
- Prior art keywords
- formula
- compound
- lower acyl
- tertiary
- xylidide
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
A procedure for the preparation of tertiary alcohol-amino-lower acyl-xylidides of the structural formula: ** (See formula) ** and its pharmaceutically acceptable salts, characterized in that a compound of the formula is reacted ** (See formula) ** wherein X is halogen such as Cl, Br or I, with a compound of the formula ** (See formula) ** until the formation of a compound of the formula I after which the compound of the formula I thus obtained, if desired, is reacted with a pharmaceutically acceptable acid. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US369146A US3925469A (en) | 1972-02-28 | 1973-06-12 | Tetiary-alkylamino-lower-acyl-xylidide local anaesthetics |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES427163A1 true ES427163A1 (en) | 1976-07-16 |
Family
ID=23454269
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES427163A Expired ES427163A1 (en) | 1973-06-12 | 1974-06-11 | Tertiary-alkylamino-lower acyl-xylidide local anesthetics |
Country Status (18)
| Country | Link |
|---|---|
| JP (1) | JPS5035121A (en) |
| AR (1) | AR204834A1 (en) |
| AT (1) | AT334346B (en) |
| AU (1) | AU6993274A (en) |
| BE (1) | BE816213A (en) |
| CA (1) | CA1027140A (en) |
| CH (1) | CH592610A5 (en) |
| DD (1) | DD115114A5 (en) |
| DE (1) | DE2427789C3 (en) |
| ES (1) | ES427163A1 (en) |
| FR (1) | FR2233042B1 (en) |
| GB (1) | GB1475774A (en) |
| HU (1) | HU167981B (en) |
| LU (1) | LU70303A1 (en) |
| NL (1) | NL7407852A (en) |
| PL (1) | PL91706B1 (en) |
| SU (1) | SU568360A3 (en) |
| ZA (1) | ZA743766B (en) |
-
1974
- 1974-01-01 AR AR254187A patent/AR204834A1/en active
- 1974-06-08 DE DE2427789A patent/DE2427789C3/en not_active Expired
- 1974-06-10 AU AU69932/74A patent/AU6993274A/en not_active Expired
- 1974-06-11 FR FR7420218A patent/FR2233042B1/fr not_active Expired
- 1974-06-11 ES ES427163A patent/ES427163A1/en not_active Expired
- 1974-06-12 SU SU7402031564A patent/SU568360A3/en active
- 1974-06-12 NL NL7407852A patent/NL7407852A/xx unknown
- 1974-06-12 CA CA202,246A patent/CA1027140A/en not_active Expired
- 1974-06-12 BE BE145319A patent/BE816213A/en unknown
- 1974-06-12 JP JP49067019A patent/JPS5035121A/ja active Pending
- 1974-06-12 DD DD179118A patent/DD115114A5/xx unknown
- 1974-06-12 ZA ZA00743766A patent/ZA743766B/en unknown
- 1974-06-12 LU LU70303A patent/LU70303A1/xx unknown
- 1974-06-12 PL PL1974171847A patent/PL91706B1/en unknown
- 1974-06-12 HU HUAA778A patent/HU167981B/hu unknown
- 1974-06-12 GB GB2608874A patent/GB1475774A/en not_active Expired
- 1974-06-12 CH CH805574A patent/CH592610A5/xx not_active IP Right Cessation
- 1974-06-12 AT AT484874A patent/AT334346B/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| FR2233042B1 (en) | 1977-11-10 |
| PL91706B1 (en) | 1977-03-31 |
| CH592610A5 (en) | 1977-10-31 |
| GB1475774A (en) | 1977-06-10 |
| JPS5035121A (en) | 1975-04-03 |
| DE2427789B2 (en) | 1978-05-03 |
| ATA484874A (en) | 1976-05-15 |
| DE2427789C3 (en) | 1979-01-18 |
| AR204834A1 (en) | 1976-03-05 |
| DE2427789A1 (en) | 1975-01-16 |
| SU568360A3 (en) | 1977-08-05 |
| FR2233042A1 (en) | 1975-01-10 |
| CA1027140A (en) | 1978-02-28 |
| LU70303A1 (en) | 1976-04-13 |
| AT334346B (en) | 1976-01-10 |
| HU167981B (en) | 1976-02-28 |
| NL7407852A (en) | 1974-12-16 |
| DD115114A5 (en) | 1975-09-12 |
| AU6993274A (en) | 1975-12-11 |
| ZA743766B (en) | 1975-06-25 |
| BE816213A (en) | 1974-12-12 |
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