ES409942A1 - Procedure for the preparation of an N-arilmidate compound. (Machine-translation by Google Translate, not legally binding) - Google Patents
Procedure for the preparation of an N-arilmidate compound. (Machine-translation by Google Translate, not legally binding)Info
- Publication number
- ES409942A1 ES409942A1 ES0409942A ES409942A ES409942A1 ES 409942 A1 ES409942 A1 ES 409942A1 ES 0409942 A ES0409942 A ES 0409942A ES 409942 A ES409942 A ES 409942A ES 409942 A1 ES409942 A1 ES 409942A1
- Authority
- ES
- Spain
- Prior art keywords
- formula
- compound
- halogen
- cycloalkyl
- general formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
A procedure for the preparation of an N-arylimidate compound of the general formula I **(See formula)** and its pharmaceutically acceptable acid addition salts, in which formula **(See formula)** R1 represents lower alkyl, lower cycloalkyl, aralkyl or aryl, X represents nitro, trifluoromethyl or halogen, Y represents hydrogen, halogen, nitro, lower alkyl, lower alkoxy, lower alkanoyl, polyfluoroalkoxy, polyfluoroalkyl or trifluoromethylthio, A represents (see formula), wherein R2 and R3 independently represent Z-substituted alkyl in which the alkyl moiety is straight-chain or branched and has at most 5 carbon atoms, or R2 and R3, together with the Carbon atoms to which they are attached represent cycloalkyl: Z-substituted wherein the cycloalkyl moiety has 5 carbon atoms at most, and Z represents hydrogen, halogen, or an etherified or esterified free hydroxy group, except that when X and Y are both chlorine, or when X is chlorine and Y is methyl, then R1 is lower alkyl, lower cycloalkyl, or aralkyl, characterized by subjecting an N-arylimidohaline of the general formula II to alcohololysis **(See formula)** by reaction with a hydroxy compound of the general formula III **(See formula)** or with a salt thereof, in which formula X, Y, A and R1 have the meaning indicated above and Z is hydrogen, halogen or an etherified hydroxyl group and isolate the compound thus obtained from the general formula I in free form or in the form of a pharmaceutically acceptable acid addition salt of yours. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US21178071A | 1971-12-23 | 1971-12-23 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES409942A1 true ES409942A1 (en) | 1976-05-16 |
Family
ID=22788341
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES0409942A Expired ES409942A1 (en) | 1971-12-23 | 1972-12-22 | Procedure for the preparation of an N-arilmidate compound. (Machine-translation by Google Translate, not legally binding) |
Country Status (14)
Country | Link |
---|---|
JP (1) | JPS4868535A (en) |
AR (1) | AR199889A1 (en) |
AT (1) | AT321266B (en) |
AU (1) | AU465324B2 (en) |
BE (1) | BE793119A (en) |
CA (1) | CA976559A (en) |
DE (1) | DE2261293A1 (en) |
ES (1) | ES409942A1 (en) |
FR (1) | FR2164833B1 (en) |
GB (1) | GB1414327A (en) |
HU (1) | HU165850B (en) |
IL (1) | IL41138A (en) |
NL (1) | NL7217449A (en) |
ZA (1) | ZA729045B (en) |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3453311A (en) * | 1966-01-20 | 1969-07-01 | Rohm & Haas | Aryl n-(aryl)-alkanoimidates |
-
0
- BE BE793119D patent/BE793119A/en unknown
-
1972
- 1972-12-08 AU AU49849/72A patent/AU465324B2/en not_active Expired
- 1972-12-15 DE DE2261293A patent/DE2261293A1/en active Pending
- 1972-12-20 IL IL41138A patent/IL41138A/en unknown
- 1972-12-21 AT AT1092572A patent/AT321266B/en not_active IP Right Cessation
- 1972-12-21 ZA ZA729045A patent/ZA729045B/en unknown
- 1972-12-21 AR AR245768A patent/AR199889A1/en active
- 1972-12-21 GB GB5916372A patent/GB1414327A/en not_active Expired
- 1972-12-21 NL NL7217449A patent/NL7217449A/xx unknown
- 1972-12-21 HU HUSCHE418*1A patent/HU165850B/hu unknown
- 1972-12-21 CA CA159,624A patent/CA976559A/en not_active Expired
- 1972-12-21 FR FR7245752A patent/FR2164833B1/fr not_active Expired
- 1972-12-22 ES ES0409942A patent/ES409942A1/en not_active Expired
- 1972-12-22 JP JP47128359A patent/JPS4868535A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
BE793119A (en) | 1973-06-21 |
FR2164833B1 (en) | 1975-10-31 |
AU4984972A (en) | 1974-06-13 |
NL7217449A (en) | 1973-06-26 |
JPS4868535A (en) | 1973-09-18 |
ZA729045B (en) | 1973-09-26 |
AT321266B (en) | 1975-03-25 |
CA976559A (en) | 1975-10-21 |
IL41138A0 (en) | 1973-02-28 |
HU165850B (en) | 1974-11-28 |
AR199889A1 (en) | 1974-10-08 |
AU465324B2 (en) | 1975-09-25 |
FR2164833A1 (en) | 1973-08-03 |
GB1414327A (en) | 1975-11-19 |
IL41138A (en) | 1976-04-30 |
DE2261293A1 (en) | 1973-07-05 |
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