ES388758A1 - Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas. - Google Patents

Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas.

Info

Publication number
ES388758A1
ES388758A1 ES388758A ES388758A ES388758A1 ES 388758 A1 ES388758 A1 ES 388758A1 ES 388758 A ES388758 A ES 388758A ES 388758 A ES388758 A ES 388758A ES 388758 A1 ES388758 A1 ES 388758A1
Authority
ES
Spain
Prior art keywords
alkyl
amino
alkylamino
alkoxy
isopropyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES388758A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sandoz AG
Original Assignee
Sandoz AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz AG filed Critical Sandoz AG
Publication of ES388758A1 publication Critical patent/ES388758A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/80Oxygen atoms
    • C07D239/82Oxygen atoms with an aryl radical attached in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • GPHYSICS
    • G02OPTICS
    • G02BOPTICAL ELEMENTS, SYSTEMS OR APPARATUS
    • G02B27/00Optical systems or apparatus not provided for by any of the groups G02B1/00 - G02B26/00, G02B30/00
    • G02B27/02Viewing or reading apparatus

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Physics & Mathematics (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Physics & Mathematics (AREA)
  • Optics & Photonics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ES388758A 1968-07-01 1971-03-01 Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas. Expired ES388758A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US74180768A 1968-07-01 1968-07-01
US78725468A 1968-12-26 1968-12-26
US81943569A 1969-04-25 1969-04-25

Publications (1)

Publication Number Publication Date
ES388758A1 true ES388758A1 (es) 1974-03-01

Family

ID=27419280

Family Applications (6)

Application Number Title Priority Date Filing Date
ES368949A Expired ES368949A1 (es) 1968-07-01 1969-06-30 Procedimiento para la obtencion de 3,4-dihidroquinazolino- nas.
ES388761A Expired ES388761A1 (es) 1968-07-01 1971-03-01 Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas.
ES388758A Expired ES388758A1 (es) 1968-07-01 1971-03-01 Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas.
ES388760A Expired ES388760A1 (es) 1968-07-01 1971-03-01 Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas.
ES388759A Expired ES388759A1 (es) 1968-07-01 1971-03-01 Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas.
ES388762A Expired ES388762A1 (es) 1968-07-01 1971-03-01 Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas.

Family Applications Before (2)

Application Number Title Priority Date Filing Date
ES368949A Expired ES368949A1 (es) 1968-07-01 1969-06-30 Procedimiento para la obtencion de 3,4-dihidroquinazolino- nas.
ES388761A Expired ES388761A1 (es) 1968-07-01 1971-03-01 Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas.

Family Applications After (3)

Application Number Title Priority Date Filing Date
ES388760A Expired ES388760A1 (es) 1968-07-01 1971-03-01 Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas.
ES388759A Expired ES388759A1 (es) 1968-07-01 1971-03-01 Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas.
ES388762A Expired ES388762A1 (es) 1968-07-01 1971-03-01 Procedimiento para la obtencion de 3,4-dihidro-quinazolino-nas.

Country Status (7)

Country Link
BE (1) BE735439A (es)
CH (1) CH515911A (es)
DE (1) DE1932396A1 (es)
ES (6) ES368949A1 (es)
FR (1) FR2012062A1 (es)
GB (1) GB1256593A (es)
NL (1) NL6909864A (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE759671A (fr) * 1969-12-01 1971-06-01 Sandoz Sa Derives de la quinazolinone, leur preparation et medicaments contenant ces derives
DK129348B (da) * 1970-07-13 1974-09-30 Sumitomo Chemical Co Analogifremgangsmåde til fremstilling af 1-substituerede 3,4-dihydro-2(1H)-quinazolinonderivater.
AU438472B2 (en) * 1970-12-23 1973-08-09 Sumitomo Chemical Company, Limited Quinazolinone derivatives anda process for production thereof
WO1993004047A1 (en) * 1991-08-16 1993-03-04 Merck & Co., Inc. Quinazoline derivatives as inhibitors of hiv reverse transcriptase
IL102764A0 (en) * 1991-08-16 1993-01-31 Merck & Co Inc Quinazoline derivatives,and pharmaceutical compositions containing them
ATE174908T1 (de) * 1993-05-26 1999-01-15 Sumitomo Pharma Chinazolinonderivate
EP3102567B1 (en) * 2014-02-04 2019-07-17 University of Tennessee Research Foundation Inhibitors of paxillin function and related compositions and methods

Also Published As

Publication number Publication date
ES368949A1 (es) 1971-07-16
ES388760A1 (es) 1974-03-01
FR2012062A1 (es) 1970-03-13
GB1256593A (es) 1971-12-08
ES388761A1 (es) 1974-03-01
ES388759A1 (es) 1974-03-01
NL6909864A (es) 1970-01-05
BE735439A (es) 1969-12-30
ES388762A1 (es) 1974-03-01
DE1932396A1 (de) 1970-01-08
CH515911A (de) 1971-11-30

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