ES369570A1 - New thiadiazolyl-ureas, their production and composition containing same - Google Patents

New thiadiazolyl-ureas, their production and composition containing same

Info

Publication number
ES369570A1
ES369570A1 ES369570A ES369570A ES369570A1 ES 369570 A1 ES369570 A1 ES 369570A1 ES 369570 A ES369570 A ES 369570A ES 369570 A ES369570 A ES 369570A ES 369570 A1 ES369570 A1 ES 369570A1
Authority
ES
Spain
Prior art keywords
formula
ureas
thiadiazolyl
aliphatic
hydrocarbon radical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES369570A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Agripat SA
Original Assignee
Agripat SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Agripat SA filed Critical Agripat SA
Publication of ES369570A1 publication Critical patent/ES369570A1/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C07D285/135—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/36—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< directly attached to at least one heterocyclic ring; Thio analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Procedure for the preparation of 1,3,4-thiadiazolyl- (2) -ureas of the formula ** (see formula) ** in which R1 means a hydrocarbon radical with at most 6 carbon atoms, aliphatic or cycloaliphatic, saturated or unsaturated, optionally substituted by ether or halogen, R2 means hydrogen, a lower aliphatic or cycloaliphatic hydrocarbon radical, R3 means hydrogen or a lower alkyl radical, R4 means a saturated or unsaturated aliphatic or cycloaliphatic hydrocarbon radical, optionally substituted etherically or by halogen or a lower alkoxy radical, characterized in that a 2-amino-1,3,4-thiadiazole of formula II ** (see formula) ** it is transformed either with an ester of halocarbonic acid or with phosgene in the presence of an acid binding agent, into a derivative of carbamic acid and this is reacted with an amine of formula III ** (see formula) ** where in formulas II and III, the symbols R1 to R4 have the meanings indicated under formula I. (Machine-translation by Google Translate, not legally binding)
ES369570A 1968-07-17 1969-07-16 New thiadiazolyl-ureas, their production and composition containing same Expired ES369570A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH1069168A CH498859A (en) 1968-07-17 1968-07-17 Process for the production of thiadiazolyl ureas

Publications (1)

Publication Number Publication Date
ES369570A1 true ES369570A1 (en) 1971-06-01

Family

ID=4365813

Family Applications (4)

Application Number Title Priority Date Filing Date
ES369569A Expired ES369569A1 (en) 1968-07-17 1969-07-16 New thiadiazolyl-ureas, their production and composition containing same
ES369570A Expired ES369570A1 (en) 1968-07-17 1969-07-16 New thiadiazolyl-ureas, their production and composition containing same
ES369572A Expired ES369572A1 (en) 1968-07-17 1969-07-16 New thiadiazolyl-ureas, their production and composition containing same
ES369571A Expired ES369571A1 (en) 1968-07-17 1969-07-16 New thiadiazolyl-ureas, their production and composition containing same

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES369569A Expired ES369569A1 (en) 1968-07-17 1969-07-16 New thiadiazolyl-ureas, their production and composition containing same

Family Applications After (2)

Application Number Title Priority Date Filing Date
ES369572A Expired ES369572A1 (en) 1968-07-17 1969-07-16 New thiadiazolyl-ureas, their production and composition containing same
ES369571A Expired ES369571A1 (en) 1968-07-17 1969-07-16 New thiadiazolyl-ureas, their production and composition containing same

Country Status (15)

Country Link
JP (1) JPS5440610B1 (en)
AT (1) AT291668B (en)
BE (1) BE736171A (en)
BG (1) BG16312A3 (en)
CH (2) CH498859A (en)
CS (1) CS157651B2 (en)
DE (1) DE1936241A1 (en)
DK (1) DK139357B (en)
ES (4) ES369569A1 (en)
FR (1) FR2013116A1 (en)
GB (1) GB1282308A (en)
IL (1) IL32632A (en)
NL (1) NL6910940A (en)
PL (1) PL80180B1 (en)
RO (1) RO61084A (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH498859A (en) * 1968-07-17 1970-11-15 Agripat Sa Process for the production of thiadiazolyl ureas
DE2044442C2 (en) * 1970-09-03 1983-11-03 Schering AG, 1000 Berlin und 4709 Bergkamen 1,1,3-Trimethyl-3 - (- 5-Ethylsulfonyl-1,3,4-Thiadiazol-2-yl) -urea with herbicidal action
DE2059328C2 (en) * 1970-11-24 1984-02-23 Schering AG, 1000 Berlin und 4709 Bergkamen 1,1,3-Trimethyl-3- (5-ethylsulfinyl-1,3,4-thiadiazol-2-YL) urea
DE2719810A1 (en) 1977-04-28 1978-11-02 Schering Ag 1,2,3-THIADIAZOLINE-2-ID DERIVATIVES, METHOD FOR THE PRODUCTION OF THESE COMPOUNDS AND THEIR CONTAINING AGENTS WITH GROWTH REGULATORY EFFECT FOR PLANTS
DE3151017A1 (en) * 1981-12-23 1983-06-30 W. Antpöhler GmbH & Co KG, 4795 Delbrück Machine for cutting dough strands into slices and method for making baked products using the machine
DE19542721A1 (en) * 1995-11-16 1997-05-22 Sgl Technik Gmbh Process for the production of moldings from plastic-filler mixtures with a high filler content
PL215132B1 (en) 2002-06-27 2013-10-31 Novo Nordisk As Aryl carbonyl derivatives as therapeutic agents
KR101196313B1 (en) 2004-01-06 2012-11-07 노보 노르디스크 에이/에스 Heteroaryl-ureas and their use as glucokinase activators
JP2009500378A (en) 2005-07-08 2009-01-08 ノボ・ノルデイスク・エー／エス Dicycloalkylcarbamoylureas as glucokinase activators
WO2007006760A1 (en) 2005-07-08 2007-01-18 Novo Nordisk A/S Dicycloalkyl urea glucokinase activators
CA2615938C (en) * 2005-07-14 2014-04-29 Novo-Nordisk A/S Urea glucokinase activators
US8138185B2 (en) 2007-01-09 2012-03-20 Novo Nordisk A/S Urea glucokinase activators
JP5226008B2 (en) 2007-01-11 2013-07-03 ノボ・ノルデイスク・エー／エス Urea glucokinase activator
AU2019287437A1 (en) 2018-06-12 2020-09-10 Vtv Therapeutics Llc Therapeutic uses of glucokinase activators in combination with insulin or insulin analogs

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1670925B2 (en) * 1967-09-19 1977-03-10 Bayer Ag, 5090 Leverkusen 1,3,4-THIADIAZOLYL URENE
GB1195672A (en) * 1968-02-01 1970-06-17 Mobil Oil Corp Novel Urea Derivatives and Herbicides containing the same
CH498859A (en) * 1968-07-17 1970-11-15 Agripat Sa Process for the production of thiadiazolyl ureas
CH521711A (en) * 1968-12-23 1972-04-30 Bayer Ag Herbicidal agent
GB1290223A (en) * 1969-04-21 1972-09-20

Also Published As

Publication number Publication date
JPS5440610B1 (en) 1979-12-04
RO61084A (en) 1976-10-15
AT291668B (en) 1971-07-26
ES369569A1 (en) 1971-06-01
BG16312A3 (en) 1972-08-20
NL6910940A (en) 1970-01-20
CH502762A (en) 1971-02-15
CS157651B2 (en) 1974-09-16
CH498859A (en) 1970-11-15
PL80180B1 (en) 1975-08-30
IL32632A0 (en) 1969-09-25
ES369572A1 (en) 1971-06-01
GB1282308A (en) 1972-07-19
IL32632A (en) 1973-03-30
BE736171A (en) 1970-01-16
FR2013116A1 (en) 1970-03-27
DE1936241A1 (en) 1970-02-12
ES369571A1 (en) 1971-06-01
DK139357B (en) 1979-02-05
DK139357C (en) 1979-07-16

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