ES2879809T3 - Ciertos inhibidores de proteínas quinasas - Google Patents
Ciertos inhibidores de proteínas quinasas Download PDFInfo
- Publication number
- ES2879809T3 ES2879809T3 ES15855878T ES15855878T ES2879809T3 ES 2879809 T3 ES2879809 T3 ES 2879809T3 ES 15855878 T ES15855878 T ES 15855878T ES 15855878 T ES15855878 T ES 15855878T ES 2879809 T3 ES2879809 T3 ES 2879809T3
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- alkyl
- cycloalkyl
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- substituted
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Organic Chemistry (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Transplantation (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462073993P | 2014-11-01 | 2014-11-01 | |
| PCT/CN2015/093551 WO2016066142A1 (en) | 2014-11-01 | 2015-11-01 | Certain protein kinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2879809T3 true ES2879809T3 (es) | 2021-11-23 |
Family
ID=55856639
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES15855878T Active ES2879809T3 (es) | 2014-11-01 | 2015-11-01 | Ciertos inhibidores de proteínas quinasas |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US10328060B2 (enExample) |
| EP (1) | EP3224248B1 (enExample) |
| JP (1) | JP6831324B2 (enExample) |
| CN (1) | CN107207441B (enExample) |
| AU (1) | AU2015341186B2 (enExample) |
| BR (1) | BR112017008867A2 (enExample) |
| CA (1) | CA2966252C (enExample) |
| ES (1) | ES2879809T3 (enExample) |
| WO (1) | WO2016066142A1 (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HK1232227A1 (zh) * | 2014-07-04 | 2018-01-05 | Lupin Limited | 作为pi3k抑制剂的喹嗪酮衍生物 |
| WO2017103825A1 (en) | 2015-12-18 | 2017-06-22 | Lupin Limited | Quinolizinone derivatives as pi3k inhibitors |
| CA3178569A1 (en) * | 2020-05-16 | 2021-11-25 | Zuwen ZHOU | Compounds as protein kinase inhibitors |
| WO2022228387A1 (en) * | 2021-04-26 | 2022-11-03 | Fochon Biosciences, Ltd. | Compounds as parp inhibitors |
| WO2023078401A1 (en) * | 2021-11-05 | 2023-05-11 | Fochon Biosciences, Ltd. | Compounds as protein kinase inhibitors |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS545996A (en) * | 1977-06-15 | 1979-01-17 | Yamanouchi Pharmaceut Co Ltd | Heterocyclic compounds and process for their preparation |
| AU5991699A (en) * | 1998-09-21 | 2000-04-10 | Biochem Pharma Inc. | Quinolizinones as integrin inhibitors |
| US6667300B2 (en) | 2000-04-25 | 2003-12-23 | Icos Corporation | Inhibitors of human phosphatidylinositol 3-kinase delta |
| WO2005113556A1 (en) | 2004-05-13 | 2005-12-01 | Icos Corporation | Quinazolinones as inhibitors of human phosphatidylinositol 3-kinase delta |
| KR20090087027A (ko) * | 2006-11-13 | 2009-08-14 | 일라이 릴리 앤드 캄파니 | 염증 질환 및 암의 치료를 위한 티에노피리미디논 |
| US8557830B2 (en) | 2007-06-07 | 2013-10-15 | Amgen Inc. | RAF kinase modulators and methods of use |
| KR101763656B1 (ko) * | 2009-06-29 | 2017-08-01 | 인사이트 홀딩스 코포레이션 | Ｐｉ3ｋ 저해물질로서의 피리미디논 |
| US8916593B2 (en) | 2010-05-04 | 2014-12-23 | Pfizer Inc. | Alkoxy-substituted 2-aminopyridines as ALK inhibitors |
| EP2518070A1 (en) | 2011-04-29 | 2012-10-31 | Almirall, S.A. | Pyrrolotriazinone derivatives as PI3K inhibitors |
| DK2812004T3 (en) * | 2012-02-10 | 2018-10-15 | Ptc Therapeutics Inc | COMPOUNDS FOR TREATMENT OF SPINAL MUSCLE DROPHY |
| WO2013149362A1 (en) | 2012-04-06 | 2013-10-10 | Glaxosmithkline Llc | 1-(dihydronaphthalenyl)pyridones as melanin-concentrating hormone receptor 1 antagonists |
| HK1232227A1 (zh) * | 2014-07-04 | 2018-01-05 | Lupin Limited | 作为pi3k抑制剂的喹嗪酮衍生物 |
-
2015
- 2015-11-01 ES ES15855878T patent/ES2879809T3/es active Active
- 2015-11-01 WO PCT/CN2015/093551 patent/WO2016066142A1/en not_active Ceased
- 2015-11-01 BR BR112017008867A patent/BR112017008867A2/pt not_active Application Discontinuation
- 2015-11-01 AU AU2015341186A patent/AU2015341186B2/en not_active Ceased
- 2015-11-01 JP JP2017523862A patent/JP6831324B2/ja not_active Expired - Fee Related
- 2015-11-01 US US15/523,315 patent/US10328060B2/en active Active
- 2015-11-01 EP EP15855878.3A patent/EP3224248B1/en active Active
- 2015-11-01 CN CN201580071637.2A patent/CN107207441B/zh not_active Expired - Fee Related
- 2015-11-01 CA CA2966252A patent/CA2966252C/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| US10328060B2 (en) | 2019-06-25 |
| BR112017008867A2 (pt) | 2017-12-26 |
| EP3224248A1 (en) | 2017-10-04 |
| US20180036293A1 (en) | 2018-02-08 |
| EP3224248A4 (en) | 2018-08-08 |
| EP3224248B1 (en) | 2021-05-05 |
| WO2016066142A1 (en) | 2016-05-06 |
| JP6831324B2 (ja) | 2021-02-17 |
| JP2017533232A (ja) | 2017-11-09 |
| AU2015341186B2 (en) | 2019-11-14 |
| CN107207441B (zh) | 2020-11-24 |
| AU2015341186A1 (en) | 2017-06-08 |
| CN107207441A (zh) | 2017-09-26 |
| CA2966252A1 (en) | 2016-05-06 |
| CA2966252C (en) | 2023-10-24 |
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