ES2665153T3 - Antagonistas del receptor EP3 de prostaglandina - Google Patents
Antagonistas del receptor EP3 de prostaglandina Download PDFInfo
- Publication number
- ES2665153T3 ES2665153T3 ES14799209.3T ES14799209T ES2665153T3 ES 2665153 T3 ES2665153 T3 ES 2665153T3 ES 14799209 T ES14799209 T ES 14799209T ES 2665153 T3 ES2665153 T3 ES 2665153T3
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- Prior art keywords
- compound
- methyl
- mmol
- pharmaceutically acceptable
- compounds
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Classifications
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- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
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- Rheumatology (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361888822P | 2013-10-09 | 2013-10-09 | |
| US201361888822P | 2013-10-09 | ||
| PCT/IB2014/064836 WO2015052610A1 (en) | 2013-10-09 | 2014-09-25 | Antagonists of prostaglandin ep3 receptor |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2665153T3 true ES2665153T3 (es) | 2018-04-24 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES14799209.3T Active ES2665153T3 (es) | 2013-10-09 | 2014-09-25 | Antagonistas del receptor EP3 de prostaglandina |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US9278953B2 (OSRAM) |
| EP (1) | EP3055300B1 (OSRAM) |
| JP (1) | JP6348582B2 (OSRAM) |
| AR (1) | AR097963A1 (OSRAM) |
| CA (1) | CA2926568C (OSRAM) |
| ES (1) | ES2665153T3 (OSRAM) |
| TW (1) | TW201527297A (OSRAM) |
| UY (1) | UY35776A (OSRAM) |
| WO (1) | WO2015052610A1 (OSRAM) |
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| JP2017538769A (ja) * | 2014-12-22 | 2017-12-28 | ファイザー・インク | プロスタグランジンｅｐ３受容体の拮抗薬 |
| US10399944B2 (en) | 2017-08-10 | 2019-09-03 | Janssen Pharmaceutica Nv | Pyridin-2-one derivatives of formula (III) useful as EP3 receptor antagonists |
| US10590083B2 (en) | 2017-08-10 | 2020-03-17 | Janssen Pharmaceutica Nv | Pyridin-2-one derivatives of formula (I) useful as EP3 receptor antagonists |
| US10336701B2 (en) * | 2017-08-10 | 2019-07-02 | Janssen Pharmaceutica Nv | Pyridin-2-one derivatives of formula (II) useful as EP3 receptor antagonists |
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| WO2021094208A1 (en) | 2019-11-12 | 2021-05-20 | Bayer Aktiengesellschaft | Substituted imidazo pyrimidine ep3 antagonists |
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| CN1149196C (zh) | 1998-07-06 | 2004-05-12 | 布里斯托尔-迈尔斯斯奎布公司 | 作为血管紧张肽和内皮肽受体双重拮抗剂的联苯基磺酰胺 |
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| PA8660701A1 (es) | 2005-02-04 | 2006-09-22 | Pfizer Prod Inc | Agonistas de pyy y sus usos |
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| TW201038580A (en) | 2009-02-02 | 2010-11-01 | Pfizer | 4-amino-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6(5H)-yl)phenyl derivatives |
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| WO2011005611A1 (en) | 2009-07-09 | 2011-01-13 | Merck Sharp & Dohme Corp. | Neuromedin u receptor agonists and uses thereof |
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- 2014-09-25 EP EP14799209.3A patent/EP3055300B1/en not_active Not-in-force
- 2014-09-25 CA CA2926568A patent/CA2926568C/en not_active Expired - Fee Related
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- 2014-10-06 TW TW103134754A patent/TW201527297A/zh unknown
- 2014-10-06 US US14/506,752 patent/US9278953B2/en not_active Expired - Fee Related
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| CA2926568C (en) | 2017-09-05 |
| AR097963A1 (es) | 2016-04-20 |
| EP3055300A1 (en) | 2016-08-17 |
| US20150099782A1 (en) | 2015-04-09 |
| EP3055300B1 (en) | 2018-03-07 |
| JP6348582B2 (ja) | 2018-06-27 |
| UY35776A (es) | 2015-05-29 |
| WO2015052610A1 (en) | 2015-04-16 |
| JP2016532647A (ja) | 2016-10-20 |
| US9278953B2 (en) | 2016-03-08 |
| CA2926568A1 (en) | 2015-04-16 |
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