ES2570385T3 - N-(1H-pirazolil-metil)-formamidas, procedimiento para su producción y su uso como inhibidores de la nitrificación - Google Patents

N-(1H-pirazolil-metil)-formamidas, procedimiento para su producción y su uso como inhibidores de la nitrificación

Info

Publication number
ES2570385T3
ES2570385T3 ES12795740T ES12795740T ES2570385T3 ES 2570385 T3 ES2570385 T3 ES 2570385T3 ES 12795740 T ES12795740 T ES 12795740T ES 12795740 T ES12795740 T ES 12795740T ES 2570385 T3 ES2570385 T3 ES 2570385T3
Authority
ES
Spain
Prior art keywords
formamides
pyrazolyl
methyl
production
nitrification inhibitors
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
ES12795740T
Other languages
English (en)
Inventor
Ute Radics
Hans-Joachim Niclas
Christoph Bender
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SKW Stickstoffwerke Piesteritz GmbH
Original Assignee
SKW Stickstoffwerke Piesteritz GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SKW Stickstoffwerke Piesteritz GmbH filed Critical SKW Stickstoffwerke Piesteritz GmbH
Application granted granted Critical
Publication of ES2570385T3 publication Critical patent/ES2570385T3/es
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C05—FERTILISERS; MANUFACTURE THEREOF
    • C05G—MIXTURES OF FERTILISERS COVERED INDIVIDUALLY BY DIFFERENT SUBCLASSES OF CLASS C05; MIXTURES OF ONE OR MORE FERTILISERS WITH MATERIALS NOT HAVING A SPECIFIC FERTILISING ACTIVITY, e.g. PESTICIDES, SOIL-CONDITIONERS, WETTING AGENTS; FERTILISERS CHARACTERISED BY THEIR FORM
    • C05G3/00—Mixtures of one or more fertilisers with additives not having a specially fertilising activity
    • C05G3/90—Mixtures of one or more fertilisers with additives not having a specially fertilising activity for affecting the nitrification of ammonium compounds or urea in the soil
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P60/00—Technologies relating to agriculture, livestock or agroalimentary industries
    • Y02P60/20—Reduction of greenhouse gas [GHG] emissions in agriculture, e.g. CO2
    • Y02P60/21—Dinitrogen oxide [N2O], e.g. using aquaponics, hydroponics or efficiency measures

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Soil Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Fertilizers (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

N-(1H-Pirazolil-metil)-formamidas de fórmula general I:**Fórmula** caracterizadas porque R4 es >= H, halógeno, alquilo C1-C4 o cicloalquilo C3-C8, R1 y R2 independientemente entre sí representan H, alquilo C1-C4 o cicloalquilo C3-C8, R3 representa alquilo C1-C4, cicloalquilo C3-C8 o arilo C6-C10 o H.
ES12795740T 2011-12-02 2012-11-28 N-(1H-pirazolil-metil)-formamidas, procedimiento para su producción y su uso como inhibidores de la nitrificación Active ES2570385T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102011120098.7A DE102011120098B4 (de) 2011-12-02 2011-12-02 N-(1H-Pyrazolyl-methyl)formamide, Verfahren zu ihrer Herstellung und ihre Verwendung als Nitrifikationsinhibitoren
PCT/EP2012/004918 WO2013079197A1 (de) 2011-12-02 2012-11-28 N-(1h-pyrazolyl-methyl)formamide, verfahren zu ihrer herstellung und ihre verwendung als nitrifikationsinhibitoren

Publications (1)

Publication Number Publication Date
ES2570385T3 true ES2570385T3 (es) 2016-05-18

Family

ID=47294835

Family Applications (1)

Application Number Title Priority Date Filing Date
ES12795740T Active ES2570385T3 (es) 2011-12-02 2012-11-28 N-(1H-pirazolil-metil)-formamidas, procedimiento para su producción y su uso como inhibidores de la nitrificación

Country Status (4)

Country Link
EP (1) EP2785697B1 (es)
DE (1) DE102011120098B4 (es)
ES (1) ES2570385T3 (es)
WO (1) WO2013079197A1 (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102013021933A1 (de) 2013-12-20 2015-06-25 Skw Stickstoffwerke Piesteritz Gmbh Verwendung von Pyrazol-Derivaten als Mittel zur Verbesserung der Trockenstresstoleranz
RU2731051C2 (ru) 2014-11-14 2020-08-28 Басф Се Бензилпропаргиловые простые эфиры в качестве ингибиторов нитрификации
AU2015366289B2 (en) 2014-12-18 2020-04-02 Basf Se Alkynylpyrazoles as nitrification inhibitors
EP3253209A1 (en) 2015-02-06 2017-12-13 Basf Se Pyrazole compounds as nitrification inhibitors
US11053175B2 (en) 2015-05-12 2021-07-06 Basf Se Thioether compounds as nitrification inhibitors
TW201705955A (zh) 2015-05-14 2017-02-16 輝瑞大藥廠 包含吡咯啶－２，５－二酮ｉｄｏ１抑制劑及抗－ｐｄ１／抗－ｐｄ－ｌ１抗體之組合療法
DE102016106592A1 (de) 2016-04-11 2017-10-12 Skw Stickstoffwerke Piesteritz Gmbh Verfahren zur Herstellung von N-((3(5)-Methyl-1H-pyrazol-1-yl)methyl)acetamid (MPA)
BR112018073298A2 (pt) 2016-05-18 2019-02-19 Basf Se cápsula, suspensão de cápsula, mistura, uso das cápsulas e método para reduzir a nitrificação
EP3652133A4 (en) 2017-07-10 2021-04-21 Basf Se MIXTURES WITH A UREA INHIBITOR (UI) AND A NITRIFICATION INHIBITOR SUCH AS 2- (3,4-DIMETHYL-1H-PYRAZOL-1-YL) SUCCIC ACID (DMPSA) OR 3,4-DIMETHYLPYRAZOLYL GLYCOLATE (DMPG)
AU2019226359B2 (en) 2018-02-28 2023-08-17 Basf Se Use of N-functionalized alkoxy pyrazole compounds as nitrification inhibitors
CN111683528B (zh) * 2018-02-28 2022-12-13 巴斯夫欧洲公司 吡唑炔丙基醚作为硝化抑制剂的用途
BR112022013894A2 (pt) 2020-01-16 2023-01-10 Basf Se Mistura, composição agroquímica, método para aumentar a eficiência de uso de fertilizante e uso da mistura
CA3163984A1 (en) 2020-01-16 2021-07-22 Basf Se Mixtures comprising nitrification inhibitors and carriers
EP4341248A1 (en) 2021-05-21 2024-03-27 Basf Se Use of an n-functionalized alkoxy pyrazole compound as nitrification inhibitor

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3635690A (en) 1968-05-16 1972-01-18 Dow Chemical Co Soil treating method and composition for conserving nitrogen in soil by addition of a pyrazole thereto
US3697244A (en) 1968-10-15 1972-10-10 Dow Chemical Co Crop culture with 4h-1,2,4-triazoles
DE2745833C2 (de) 1977-10-12 1986-10-16 VEB Fahlberg-List Chemische und pharmazeutische Fabriken, DDR 3013 Magdeburg Mittel zur Hemmung bzw. Regelung der Nitrifikation von Ammoniumstickstoff in Kulturböden
DE3409317A1 (de) 1984-03-14 1985-09-19 Basf Ag, 6700 Ludwigshafen Nitrifikationsinhibierende 1-hydroxipyrazol-derivate
US4523940A (en) 1984-06-25 1985-06-18 The Dow Chemical Company Soil treating method and composition for conserving nitrogen in soil
AU4348285A (en) 1984-06-25 1986-01-02 Dow Chemical Company, The Pyrazole growth enhancer
US4969946A (en) 1986-01-29 1990-11-13 The Dow Chemical Company Soil treating method and composition for conserving nitrogen in naturally alkaline soil
SU1470737A1 (ru) 1986-09-19 1989-04-07 Предприятие П/Я Г-4302 Способ ингибировани нитрификации карбамида в почве
DE3704359A1 (de) 1987-02-12 1988-08-25 Basf Ag Azolhalbaminal-derivate und ihre verwendung als nitrifikationsinhibitoren
DD292232A5 (de) 1988-10-17 1991-07-25 Stickstoffwerke Ag Wittenberg-Piesteritz,De Mittel zur hemmung bzw. regelung der nitrifikation von ammoniumstickstoff in kulturboeden
DE4018395A1 (de) 1990-06-08 1992-02-20 Wittenberg Stickstoff Ag Mittel zur hemmung bzw. regelung der nitrifikation von ammoniumstickstoff in kulturboeden
DE4111922A1 (de) 1991-04-12 1992-10-15 Basf Ag Verfahren zur herstellung von 1-carbamoyl-pyrazolen
DE4128828A1 (de) 1991-08-30 1993-03-04 Basf Ag Ammonium- oder harnstoffhaltige duengemittel und verfahren zu ihrer herstellung
JPH07104135A (ja) 1993-10-06 1995-04-21 Sanyo Electric Co Ltd 立体画像表示装置
DE4446194A1 (de) 1994-12-23 1996-06-27 Basf Ag Verwendung von Pyrazolderivaten mit hydrophoben Resten als Nitrifikationsinhibitoren
DE19503827A1 (de) 1995-02-06 1996-08-08 Basf Ag Verwendung von schwerflüchtigen Pyrazolderivaten mit hydrophilen Gruppen als Nitrifikationsinhibitoren
DE19631764A1 (de) 1996-08-06 1998-02-12 Basf Ag Neue Nitrifikationsinhibitoren sowie die Verwendung von Polysäuren zur Behandlung von Mineraldüngemitteln die einen Nitrifikationsinhibitor enthalten
DE19822340B4 (de) 1998-05-19 2008-02-28 Skw Stickstoffwerke Piesteritz Gmbh Thermostabile schwerflüchtige Alkyl-1H-1-pyrazolylmethanamin-Derivate und deren Verwendung als Nitrifikationsinhibitoren
DE50105621D1 (de) 2000-04-14 2005-04-21 Piesteritz Stickstoff 1h-pyrazol-derivate, verfahren zu ihrer herstellung und deren verwendung zur hemmung und steuerung der nitrifikation
DE10135423A1 (de) 2000-08-08 2002-02-21 Piesteritz Stickstoff 1H-Pyrazol-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Nitrifikationsinhibitoren
DE10343277A1 (de) 2003-09-18 2005-04-21 Piesteritz Stickstoff N-(1H-Azolyl-methyl)amide, Verfahren zu ihrer Herstellung und ihre Verwendung als Nitrifikationsinhibitoren

Also Published As

Publication number Publication date
DE102011120098B4 (de) 2021-02-11
WO2013079197A1 (de) 2013-06-06
EP2785697B1 (de) 2016-02-03
EP2785697A1 (de) 2014-10-08
DE102011120098A1 (de) 2013-06-06

Similar Documents

Publication Publication Date Title
ES2570385T3 (es) N-(1H-pirazolil-metil)-formamidas, procedimiento para su producción y su uso como inhibidores de la nitrificación
EA201190227A1 (ru) Оксазолзамещенные индазолы в качестве ингибиторов pi3-киназ
CU20140110A7 (es) Compuestos heterocíclicos como inhibidores de mek
ECSP14033037A (es) Síntesis de compuestos heterocíclicos
UA116920C2 (uk) Інгібітори fgfr4
UY32631A (es) Derivados de ciclopenta[c]pirrol-2-carboxilatos, su preparación y su aplicación en terapéutica.
MX2013008212A (es) Derivados de 7-azaindol.
EA201490474A1 (ru) Аминохиназолины в качестве ингибиторов киназ
GT201200322A (es) Derivados de carbamato de hexafluoroisoprofilo, su preparacion y su aplicacion en terapeutica
UY33946A (es) Derivados de c4-monometil triterpenoides y sus métodos de uso
MX2020005498A (es) Inhibidores de cdk.
MX341456B (es) Amino-quinolinas como inhibidores de cinasa.
EA201400338A1 (ru) Производные аминопиримидина для применения в качестве модуляторов киназной активности
EA201400333A1 (ru) Бензонитрильные производные в качестве ингибиторов киназ
DOP2014000036A (es) Compuestos de piridazinona y su uso como inhibidores daao
ECSP14013251A (es) Derivados de 5-flúor-4-imino-3-(sustituido)-3,4-dihidropirimidin-2(1h)ona
UY32630A (es) Derivados de 7-aza-espiro[3.5]nonano-7-carboxilatos, su preparación y su aplicación en terapéutica.
UY34541A (es) ?derivados de dihidro-benzo-oxazina y dihidro-pirido-oxazina?.
CO7151502A2 (es) Compuestos que inhiben la actividad de catecol o- metiltransferasa
UY34006A (es) Imidazopiridazinas
UY33549A (es) Quinolil aminas como agentes inhibidores de las quinasas
EA201301301A1 (ru) Производные тиазола
EA201490643A1 (ru) Новые производные бетулиновой кислоты с противовирусной активностью
EA201590561A1 (ru) Пролекарства аминохиназолинового ингибитора киназы
CR20150257A (es) Derivados de n-(piridin-2-il)pirimidin-4-amina que contiene un grupo sulfoximina