ES2428697T3 - Uso de agentes de enlace del receptor EDG en el cáncer - Google Patents
Uso de agentes de enlace del receptor EDG en el cáncer Download PDFInfo
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- ES2428697T3 ES2428697T3 ES08152489T ES08152489T ES2428697T3 ES 2428697 T3 ES2428697 T3 ES 2428697T3 ES 08152489 T ES08152489 T ES 08152489T ES 08152489 T ES08152489 T ES 08152489T ES 2428697 T3 ES2428697 T3 ES 2428697T3
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- VBEQCZHXXJYVRD-GACYYNSASA-N uroanthelone Chemical compound C([C@@H](C(=O)N[C@H](C(=O)N[C@@H](CS)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CS)C(=O)N[C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)NCC(=O)N[C@@H](CC=1C=CC(O)=CC=1)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CS)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC=1C2=CC=CC=C2NC=1)C(=O)N[C@@H](CC=1C2=CC=CC=C2NC=1)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(O)=O)C(C)C)[C@@H](C)O)NC(=O)[C@H](CO)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](NC(=O)[C@H](CC=1NC=NC=1)NC(=O)[C@H](CCSC)NC(=O)[C@H](CS)NC(=O)[C@@H](NC(=O)CNC(=O)CNC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CS)NC(=O)[C@H](CC=1C=CC(O)=CC=1)NC(=O)CNC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CC=1C=CC(O)=CC=1)NC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)[C@H]1N(CCC1)C(=O)[C@H](CS)NC(=O)CNC(=O)[C@H]1N(CCC1)C(=O)[C@H](CC=1C=CC(O)=CC=1)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(N)=O)C(C)C)[C@@H](C)CC)C1=CC=C(O)C=C1 VBEQCZHXXJYVRD-GACYYNSASA-N 0.000 description 1
- 210000001215 vagina Anatomy 0.000 description 1
- 229960002004 valdecoxib Drugs 0.000 description 1
- LNPDTQAFDNKSHK-UHFFFAOYSA-N valdecoxib Chemical compound CC=1ON=C(C=2C=CC=CC=2)C=1C1=CC=C(S(N)(=O)=O)C=C1 LNPDTQAFDNKSHK-UHFFFAOYSA-N 0.000 description 1
- MSRILKIQRXUYCT-UHFFFAOYSA-M valproate semisodium Chemical compound [Na+].CCCC(C(O)=O)CCC.CCCC(C([O-])=O)CCC MSRILKIQRXUYCT-UHFFFAOYSA-M 0.000 description 1
- 229960000604 valproic acid Drugs 0.000 description 1
- 229960000241 vandetanib Drugs 0.000 description 1
- 201000011531 vascular cancer Diseases 0.000 description 1
- 206010055031 vascular neoplasm Diseases 0.000 description 1
- JXLYSJRDGCGARV-CFWMRBGOSA-N vinblastine Chemical compound C([C@H](C[C@]1(C(=O)OC)C=2C(=CC3=C([C@]45[C@H]([C@@]([C@H](OC(C)=O)[C@]6(CC)C=CCN([C@H]56)CC4)(O)C(=O)OC)N3C)C=2)OC)C[C@@](C2)(O)CC)N2CCC2=C1NC1=CC=CC=C21 JXLYSJRDGCGARV-CFWMRBGOSA-N 0.000 description 1
- 229960004528 vincristine Drugs 0.000 description 1
- OGWKCGZFUXNPDA-UHFFFAOYSA-N vincristine Natural products C1C(CC)(O)CC(CC2(C(=O)OC)C=3C(=CC4=C(C56C(C(C(OC(C)=O)C7(CC)C=CCN(C67)CC5)(O)C(=O)OC)N4C=O)C=3)OC)CN1CCC1=C2NC2=CC=CC=C12 OGWKCGZFUXNPDA-UHFFFAOYSA-N 0.000 description 1
- 125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 description 1
- 229920002554 vinyl polymer Polymers 0.000 description 1
- XLMPPFTZALNBFS-INIZCTEOSA-N vorozole Chemical compound C1([C@@H](C2=CC=C3N=NN(C3=C2)C)N2N=CN=C2)=CC=C(Cl)C=C1 XLMPPFTZALNBFS-INIZCTEOSA-N 0.000 description 1
- 210000003905 vulva Anatomy 0.000 description 1
- 230000003442 weekly effect Effects 0.000 description 1
- 238000001262 western blot Methods 0.000 description 1
- 229940053867 xeloda Drugs 0.000 description 1
- 229940033942 zoladex Drugs 0.000 description 1
- 229960004276 zoledronic acid Drugs 0.000 description 1
- 229940002005 zometa Drugs 0.000 description 1
- CGTADGCBEXYWNE-JUKNQOCSSA-N zotarolimus Chemical compound N1([C@H]2CC[C@@H](C[C@@H](C)[C@H]3OC(=O)[C@@H]4CCCCN4C(=O)C(=O)[C@@]4(O)[C@H](C)CC[C@H](O4)C[C@@H](/C(C)=C/C=C/C=C/[C@@H](C)C[C@@H](C)C(=O)[C@H](OC)[C@H](O)/C(C)=C/[C@@H](C)C(=O)C3)OC)C[C@H]2OC)C=NN=N1 CGTADGCBEXYWNE-JUKNQOCSSA-N 0.000 description 1
- 229950009819 zotarolimus Drugs 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0211261A GB0211261D0 (en) | 2002-05-16 | 2002-05-16 | Organic compounds |
| GB0211261 | 2002-05-16 | ||
| US39041102P | 2002-06-20 | 2002-06-20 | |
| US390411P | 2002-06-20 | ||
| GB0217150A GB0217150D0 (en) | 2002-07-24 | 2002-07-24 | Organic compounds |
| GB0217150 | 2002-07-24 | ||
| US44973903P | 2003-02-24 | 2003-02-24 | |
| US449739P | 2003-02-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2428697T3 true ES2428697T3 (es) | 2013-11-08 |
Family
ID=43508462
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES08152489T Expired - Lifetime ES2428697T3 (es) | 2002-05-16 | 2003-05-15 | Uso de agentes de enlace del receptor EDG en el cáncer |
Country Status (7)
| Country | Link |
|---|---|
| KR (5) | KR20120025018A (pl) |
| DK (1) | DK1944026T3 (pl) |
| ES (1) | ES2428697T3 (pl) |
| PL (1) | PL396723A1 (pl) |
| PT (1) | PT1944026E (pl) |
| SI (1) | SI1944026T1 (pl) |
| TW (2) | TWI341197B (pl) |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH1180026A (ja) * | 1997-09-02 | 1999-03-23 | Yoshitomi Pharmaceut Ind Ltd | 新規免疫抑制剤、その使用方法およびその同定方法 |
-
2003
- 2003-05-15 PT PT81524894T patent/PT1944026E/pt unknown
- 2003-05-15 KR KR1020127004175A patent/KR20120025018A/ko not_active Withdrawn
- 2003-05-15 KR KR1020117018300A patent/KR101299873B1/ko not_active Expired - Fee Related
- 2003-05-15 PL PL396723A patent/PL396723A1/pl not_active Application Discontinuation
- 2003-05-15 SI SI200332293T patent/SI1944026T1/sl unknown
- 2003-05-15 KR KR1020107027288A patent/KR20100133027A/ko not_active Withdrawn
- 2003-05-15 TW TW097139649A patent/TWI341197B/zh not_active IP Right Cessation
- 2003-05-15 KR KR1020137019570A patent/KR20130088904A/ko not_active Ceased
- 2003-05-15 TW TW092113223A patent/TWI340036B/zh not_active IP Right Cessation
- 2003-05-15 ES ES08152489T patent/ES2428697T3/es not_active Expired - Lifetime
- 2003-05-15 KR KR10-2004-7018417A patent/KR20050003460A/ko not_active Withdrawn
- 2003-05-15 DK DK08152489.4T patent/DK1944026T3/da active
Also Published As
| Publication number | Publication date |
|---|---|
| PL396723A1 (pl) | 2011-12-19 |
| TW200906381A (en) | 2009-02-16 |
| KR20130088904A (ko) | 2013-08-08 |
| KR20110094154A (ko) | 2011-08-19 |
| DK1944026T3 (da) | 2013-09-30 |
| TWI341197B (en) | 2011-05-01 |
| KR101299873B1 (ko) | 2013-08-23 |
| KR20120025018A (ko) | 2012-03-14 |
| TWI340036B (en) | 2011-04-11 |
| TW200307533A (en) | 2003-12-16 |
| SI1944026T1 (sl) | 2013-10-30 |
| KR20100133027A (ko) | 2010-12-20 |
| PT1944026E (pt) | 2013-09-18 |
| KR20050003460A (ko) | 2005-01-10 |
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