ES2071346T3 - Tetrapeptidos que derivan de antibioticos dalbaheptidos. - Google Patents

Tetrapeptidos que derivan de antibioticos dalbaheptidos.

Info

Publication number
ES2071346T3
ES2071346T3 ES91920590T ES91920590T ES2071346T3 ES 2071346 T3 ES2071346 T3 ES 2071346T3 ES 91920590 T ES91920590 T ES 91920590T ES 91920590 T ES91920590 T ES 91920590T ES 2071346 T3 ES2071346 T3 ES 2071346T3
Authority
ES
Spain
Prior art keywords
group
tetrapeptides
antibiotics
carboxyacid
dalbaheptid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES91920590T
Other languages
English (en)
Inventor
Adriano Malabarba
Romeo Ciabatti
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gruppo Lepetit SpA
Original Assignee
Gruppo Lepetit SpA
Lepetit SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruppo Lepetit SpA, Lepetit SpA filed Critical Gruppo Lepetit SpA
Application granted granted Critical
Publication of ES2071346T3 publication Critical patent/ES2071346T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)

Abstract

TETRAPEPTIDOS DE LA FORMULA GENERAL (I) QUE DERIVAN DE ANTIBIOTICOS DALBAHEPTIDOS EN DONDE: W Y Z REPRESENTAN LAS PARTES RELATIVAS DEL AGLICONE DE UN ANTIBIOTICO DEL GRUPO DALBAHEPTIDO (AGLUCODALBAHEPTIDOS); Y REPRESENTA UN GRUPO CARBOXIACIDO O UN DERIVADO FUNCIONAL DE DICHO GRUPO CARBOXIACIDO; R Y R0 REPRESENTAN CADA UNO INDEPENDIENTEMENTE UN GRUPO AMINO O AMINO PROTEGIDO; R1 REPRESENTA HIDROGENO O UN GRUPO DE PROTECCION DE LA FUNCION CARBOXIACIDA; Y SUS SALES CON ACIDOS Y BASES ASI COMO SUS SALES INTERIORES. UN PROCESO PARA LA PRODUCCION DE LOS TETRAPEPTIDOS DE FORMULA (I) A PARTIR DE LOS DALBAHEPTIDOS Y AGLUCODALBAHEPTIDOS CORRESPONDIENTES.
ES91920590T 1990-12-10 1991-11-28 Tetrapeptidos que derivan de antibioticos dalbaheptidos. Expired - Lifetime ES2071346T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP90123672 1990-12-10

Publications (1)

Publication Number Publication Date
ES2071346T3 true ES2071346T3 (es) 1995-06-16

Family

ID=8204819

Family Applications (1)

Application Number Title Priority Date Filing Date
ES91920590T Expired - Lifetime ES2071346T3 (es) 1990-12-10 1991-11-28 Tetrapeptidos que derivan de antibioticos dalbaheptidos.

Country Status (10)

Country Link
EP (1) EP0561827B1 (es)
JP (1) JP3276632B2 (es)
KR (1) KR100202250B1 (es)
AT (1) ATE121101T1 (es)
CA (1) CA2098098C (es)
DE (1) DE69108930T2 (es)
DK (1) DK0561827T3 (es)
ES (1) ES2071346T3 (es)
IE (1) IE914265A1 (es)
WO (1) WO1992010517A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100298136B1 (ko) * 1993-05-19 2001-10-24 클라우디오 쿼르타 합성아글루코달바헵티드항생제

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2110401T3 (es) * 1989-07-18 1998-02-16 Biosearch Italia Spa Antibioticos pentapeptidicos derivados de dalbaheptidos.

Also Published As

Publication number Publication date
JP3276632B2 (ja) 2002-04-22
DE69108930T2 (de) 1995-08-24
DK0561827T3 (da) 1995-07-03
EP0561827B1 (en) 1995-04-12
KR100202250B1 (ko) 1999-06-15
KR930703358A (ko) 1993-11-29
WO1992010517A1 (en) 1992-06-25
CA2098098A1 (en) 1992-06-10
DE69108930D1 (de) 1995-05-18
IE914265A1 (en) 1992-06-17
CA2098098C (en) 2003-04-08
ATE121101T1 (de) 1995-04-15
JPH06503307A (ja) 1994-04-14
EP0561827A1 (en) 1993-09-29

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