ES2057901T3 - Derivados de benzotiazol, su preparacion y los medicamentos que les contienen. - Google Patents
Derivados de benzotiazol, su preparacion y los medicamentos que les contienen.Info
- Publication number
- ES2057901T3 ES2057901T3 ES91910896T ES91910896T ES2057901T3 ES 2057901 T3 ES2057901 T3 ES 2057901T3 ES 91910896 T ES91910896 T ES 91910896T ES 91910896 T ES91910896 T ES 91910896T ES 2057901 T3 ES2057901 T3 ES 2057901T3
- Authority
- ES
- Spain
- Prior art keywords
- pct
- preparation
- radical
- benzotiazole
- medicines
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Hospice & Palliative Care (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Psychiatry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
SE DESCRIBEN COMPUESTOS DE LA FORMULA (I), EN LA CUAL R1 REPRESENTA UN RADICAL POLIFLUOROALCOXI; R2 REPRESENTA UN ATOMO DE AZUFRE O DE NITROGENO SUSTITUIDO POR UN RADICAL ALQUILO O UN RADICAL SULFONILO O SULFINILO; R3 REPRESENTA UN RADICAL FENILO, BENZOILO, - NR4R5 O PIPERIDINIL - 4 SUSTITUIDO EN POSICION - 1 POR UN RADICAL FENILALQUILO; R4 REPRESENTA UN RADICAL ALQUILO; R5 REPRESENTA UN RADICAL FENILALQUILO, N ES IGUAL A 1,2 O 3; M ES IGUAL A 0,1,2 O 3. EL INVENTO TAMBIEN DESCRIBE LAS SALES DE DICHOS COMPUESTOS, PROCESOS PARA SU PREPARACION Y MEDICAMENTOS QUE LOS CONTIENEN.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9007068A FR2663029B1 (fr) | 1990-06-07 | 1990-06-07 | Derives de benzothiazole, leur preparation et les medicaments les contenant. |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2057901T3 true ES2057901T3 (es) | 1994-10-16 |
Family
ID=9397359
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES91910896T Expired - Lifetime ES2057901T3 (es) | 1990-06-07 | 1991-05-31 | Derivados de benzotiazol, su preparacion y los medicamentos que les contienen. |
Country Status (10)
Country | Link |
---|---|
US (1) | US5340824A (es) |
EP (1) | EP0532602B1 (es) |
JP (1) | JPH05507918A (es) |
AT (1) | ATE109475T1 (es) |
CA (1) | CA2080005A1 (es) |
DE (1) | DE69103271T2 (es) |
DK (1) | DK0532602T3 (es) |
ES (1) | ES2057901T3 (es) |
FR (1) | FR2663029B1 (es) |
WO (1) | WO1991018892A1 (es) |
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5824662A (en) | 1996-09-27 | 1998-10-20 | Guilford Pharmaceuticals Inc. | Treatment of global and focal ischemia using naaladase inhibitors |
US6017903A (en) | 1996-09-27 | 2000-01-25 | Guilford Pharmaceuticals Inc. | Pharmaceutical compositions and methods of treating a glutamate abnormality and effecting a neuronal activity in an animal using NAALADase inhibitors |
US6413948B1 (en) | 1996-09-27 | 2002-07-02 | Guilford Pharmaceuticals Inc. | Pharmaceutical compositions and methods of effecting a neuronal activity in an animal using naaladase inhibitors |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2688138B1 (fr) * | 1992-03-06 | 1995-05-05 | Rhone Poulenc Rorer Sa | Application de l'amino-2 trifluoromethoxy-6 benzothiazole pour obtenir un medicament destine au traitement de la sclerose laterale amyotrophique. |
DE4310523A1 (de) * | 1993-03-31 | 1994-10-06 | Basf Ag | Imidazolo-chinoxalinone zur Behandlung zentralnervöser Erkrankungen |
ATE291015T1 (de) * | 1997-11-05 | 2005-04-15 | Mitsubishi Chem Corp | Alkylaminoderivate |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2492258A1 (fr) * | 1980-10-17 | 1982-04-23 | Pharmindustrie | Nouveau medicament a base d'amino-2 trifluoromethoxy-6 benzothiazole |
GB8820231D0 (en) * | 1988-08-25 | 1988-09-28 | Fujisawa Pharmaceutical Co | New benzazole compounds processes for preparation thereof & pharmaceutical composition comprising same |
DE68903484T2 (de) * | 1988-12-15 | 1993-03-18 | Rhone Poulenc Sante | 2-imino-6-polyfluoralkoxy-benzothiazol-derivate, verfahren zu deren herstellung und arzneimittel, die sie enthalten. |
FR2649701B2 (fr) * | 1988-12-15 | 1991-11-22 | Rhone Poulenc Sante | Derives d'imino-2 benzothiazoline, leurs procedes de preparation et les medicaments les contenant |
-
1990
- 1990-06-07 FR FR9007068A patent/FR2663029B1/fr not_active Expired - Lifetime
-
1991
- 1991-05-31 EP EP91910896A patent/EP0532602B1/fr not_active Expired - Lifetime
- 1991-05-31 WO PCT/FR1991/000437 patent/WO1991018892A1/fr active IP Right Grant
- 1991-05-31 DE DE69103271T patent/DE69103271T2/de not_active Expired - Fee Related
- 1991-05-31 DK DK91910896.9T patent/DK0532602T3/da active
- 1991-05-31 CA CA002080005A patent/CA2080005A1/fr not_active Abandoned
- 1991-05-31 AT AT91910896T patent/ATE109475T1/de active
- 1991-05-31 JP JP91510727A patent/JPH05507918A/ja active Pending
- 1991-05-31 ES ES91910896T patent/ES2057901T3/es not_active Expired - Lifetime
- 1991-05-31 US US07/938,153 patent/US5340824A/en not_active Expired - Fee Related
Cited By (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5824662A (en) | 1996-09-27 | 1998-10-20 | Guilford Pharmaceuticals Inc. | Treatment of global and focal ischemia using naaladase inhibitors |
US5985855A (en) | 1996-09-27 | 1999-11-16 | Guilford Pharmaceuticals Inc. | Treatment of global and focal ischemia using NAALADase inhibitors |
US6004946A (en) | 1996-09-27 | 1999-12-21 | Guilford Pharmaceuticals Inc. | Treatment of global and focal ischemia using naaladase inhibitors |
US6017903A (en) | 1996-09-27 | 2000-01-25 | Guilford Pharmaceuticals Inc. | Pharmaceutical compositions and methods of treating a glutamate abnormality and effecting a neuronal activity in an animal using NAALADase inhibitors |
US6413948B1 (en) | 1996-09-27 | 2002-07-02 | Guilford Pharmaceuticals Inc. | Pharmaceutical compositions and methods of effecting a neuronal activity in an animal using naaladase inhibitors |
Also Published As
Publication number | Publication date |
---|---|
DE69103271T2 (de) | 1994-12-22 |
JPH05507918A (ja) | 1993-11-11 |
FR2663029A1 (fr) | 1991-12-13 |
WO1991018892A1 (fr) | 1991-12-12 |
ATE109475T1 (de) | 1994-08-15 |
EP0532602A1 (fr) | 1993-03-24 |
DK0532602T3 (da) | 1994-09-12 |
US5340824A (en) | 1994-08-23 |
DE69103271D1 (de) | 1994-09-08 |
EP0532602B1 (fr) | 1994-08-03 |
FR2663029B1 (fr) | 1992-07-31 |
CA2080005A1 (fr) | 1991-12-08 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG2A | Definitive protection |
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