ES2004693A6 - Un procedimiento para la preparacion de una composicion farmaceutica solida administrable por via oral, que contiene vinburnina como principio activo. - Google Patents
Un procedimiento para la preparacion de una composicion farmaceutica solida administrable por via oral, que contiene vinburnina como principio activo.Info
- Publication number
- ES2004693A6 ES2004693A6 ES8700706A ES8700706A ES2004693A6 ES 2004693 A6 ES2004693 A6 ES 2004693A6 ES 8700706 A ES8700706 A ES 8700706A ES 8700706 A ES8700706 A ES 8700706A ES 2004693 A6 ES2004693 A6 ES 2004693A6
- Authority
- ES
- Spain
- Prior art keywords
- vinburnine
- preparing
- pharmaceutical compositions
- compositions containing
- active principle
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/475—Quinolines; Isoquinolines having an indole ring, e.g. yohimbine, reserpine, strychnine, vinblastine
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
UN PROCEDIMIENTO PARA LA PREPARACION DE UNA COMPOSICION FARMACEUTICA SOLIDA ADMINISTRABLE POR VIA ORAL, QUE CONTIENE VINBURNINA COMO PRINCIPIO ACTIVO. EL PROCEDIMIENTO CONSISTE EN APLICAR EL PRINCIPIO ACTIVO MEZCLADO CON EXCIPIENTE IDONEOS SOBRE GRANULOS INERTES (CONSTITUIDOS POR GRANULOS DE SACAROSA Y DE ALMIDON DE MAIZ) OBTENIENDOSE UNOS GRANULOS QUE SEREVISTEN CON UNA MEMBRANA RETARDANTE CONSTITUIDA POR UN POLIMERO ANIONICO DE ACIDO METACRILICO PARCIALMENTE ESTERIFICADO CON METILO. LAS COMPOSICIONES FARMACEUTICAS ASI OBTENIDAS, EN FORMA DE CAPSULAS O COMPRIMIDOS, ESTAN CONSTITUIDAS POR MICROGRANULOS QUE CONTIENEN EL PRINCIPIO ACTIVO, EXCIPIENTES DE GRANULACION Y UN ACIDO ORGANICO PARA REGULAR EL PH, REVESTIDOS POR UN POLIMERO ANIONICO; TIENEN MEJORADAS FAVORABLEMENTE LA FARMACOCINETICA Y BIO DISPONIBILIDAD DEL PRINCIPIO ACTIVO Y SON UTILES PARA EL TRATAMIENTO DE TRASTORNOS CEREBROVASCULARES.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT19751/86A IT1204839B (it) | 1986-03-14 | 1986-03-14 | Composizioni farmaceutiche contenenti vinburnina e loro procedimento di preparazione |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2004693A6 true ES2004693A6 (es) | 1989-02-01 |
Family
ID=11160928
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES8700706A Expired ES2004693A6 (es) | 1986-03-14 | 1987-03-13 | Un procedimiento para la preparacion de una composicion farmaceutica solida administrable por via oral, que contiene vinburnina como principio activo. |
Country Status (8)
Country | Link |
---|---|
BE (1) | BE1000087A3 (es) |
DE (1) | DE3708068A1 (es) |
ES (1) | ES2004693A6 (es) |
FR (1) | FR2597340B1 (es) |
GR (1) | GR870422B (es) |
IT (1) | IT1204839B (es) |
MY (1) | MY102368A (es) |
PT (1) | PT84465B (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN113402506B (zh) * | 2021-06-17 | 2023-06-16 | 四川大学 | 中间体和制备方法及其在合成长春布宁上的应用 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2313915A1 (fr) * | 1976-01-26 | 1977-01-07 | Corneille Gilbert | Nouvelle forme galenique d'administration de la vincamine et de ses derives, son procede de preparation et medicaments comprenant cette nouvelle forme |
DE2950977A1 (de) * | 1978-12-22 | 1980-07-10 | Donald E Panoz | Neue galenische zubereitungsform fuer die orale verabreichung von medikamenten mit programmierter besetzung, sowie verfahren zu ihrer herstellung |
-
1986
- 1986-03-14 IT IT19751/86A patent/IT1204839B/it active Protection Beyond IP Right Term
-
1987
- 1987-03-12 PT PT84465A patent/PT84465B/pt not_active IP Right Cessation
- 1987-03-13 DE DE19873708068 patent/DE3708068A1/de not_active Withdrawn
- 1987-03-13 GR GR870422A patent/GR870422B/el unknown
- 1987-03-13 FR FR878703446A patent/FR2597340B1/fr not_active Expired - Lifetime
- 1987-03-13 BE BE8700264A patent/BE1000087A3/fr not_active IP Right Cessation
- 1987-03-13 ES ES8700706A patent/ES2004693A6/es not_active Expired
- 1987-09-25 MY MYPI87001939A patent/MY102368A/en unknown
Also Published As
Publication number | Publication date |
---|---|
DE3708068A1 (de) | 1987-09-17 |
BE1000087A3 (fr) | 1988-02-02 |
IT8619751A0 (it) | 1986-03-14 |
IT1204839B (it) | 1989-03-10 |
MY102368A (en) | 1992-06-17 |
FR2597340A1 (fr) | 1987-10-23 |
PT84465A (en) | 1987-04-01 |
GR870422B (en) | 1987-07-10 |
FR2597340B1 (fr) | 1990-04-13 |
PT84465B (pt) | 1989-10-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD1A | Patent lapsed |
Effective date: 20020401 |