EG24851A - Crystalline anticholinergic process for the preparation thereof for preparing a medicament - Google Patents

Crystalline anticholinergic process for the preparation thereof for preparing a medicament

Info

Publication number
EG24851A
EG24851A EG2002060698A EG2002060698A EG24851A EG 24851 A EG24851 A EG 24851A EG 2002060698 A EG2002060698 A EG 2002060698A EG 2002060698 A EG2002060698 A EG 2002060698A EG 24851 A EG24851 A EG 24851A
Authority
EG
Egypt
Prior art keywords
medicament
preparing
preparation
anticholinergic
crystalline
Prior art date
Application number
EG2002060698A
Other languages
English (en)
Inventor
Peter Sieger
Ulrike Werthmann
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Application granted granted Critical
Publication of EG24851A publication Critical patent/EG24851A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pulmonology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
EG2002060698A 2001-06-22 2002-06-19 Crystalline anticholinergic process for the preparation thereof for preparing a medicament EG24851A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10129710 2001-06-22
DE10215436 2002-04-08

Publications (1)

Publication Number Publication Date
EG24851A true EG24851A (en) 2010-10-27

Family

ID=26009556

Family Applications (1)

Application Number Title Priority Date Filing Date
EG2002060698A EG24851A (en) 2001-06-22 2002-06-19 Crystalline anticholinergic process for the preparation thereof for preparing a medicament

Country Status (38)

Country Link
EP (1) EP1401445B1 (cs)
JP (1) JP2005504015A (cs)
KR (2) KR100971616B1 (cs)
CN (1) CN100586948C (cs)
AR (1) AR037491A1 (cs)
AT (1) ATE337006T1 (cs)
AU (1) AU2002345016B2 (cs)
BG (1) BG66303B1 (cs)
BR (1) BR0210537A (cs)
CA (1) CA2450961C (cs)
CO (1) CO5550423A2 (cs)
CY (1) CY1105223T1 (cs)
CZ (1) CZ302786B6 (cs)
DE (1) DE50207943D1 (cs)
DK (1) DK1401445T3 (cs)
EA (1) EA005813B1 (cs)
EE (1) EE05316B1 (cs)
EG (1) EG24851A (cs)
ES (1) ES2271280T3 (cs)
HK (1) HK1068540A1 (cs)
HR (1) HRP20031066B1 (cs)
HU (1) HUP0400333A3 (cs)
IL (2) IL159238A0 (cs)
ME (1) ME00412B (cs)
MX (1) MXPA03011718A (cs)
MY (1) MY122779A (cs)
NO (1) NO334301B1 (cs)
NZ (1) NZ530690A (cs)
PE (2) PE20030130A1 (cs)
PL (1) PL208137B1 (cs)
PT (1) PT1401445E (cs)
RS (1) RS50441B (cs)
SA (1) SA02230255B1 (cs)
SI (1) SI1401445T1 (cs)
SK (1) SK287262B6 (cs)
TW (2) TWI261589B (cs)
UY (1) UY27342A1 (cs)
WO (1) WO2003000265A1 (cs)

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US9108962B2 (en) 2005-12-19 2015-08-18 Sicor, Inc. Forms of tiotropium bromide and processes for preparation thereof
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EP1847543A1 (de) 2006-04-19 2007-10-24 Boehringer Ingelheim Pharma GmbH & Co. KG Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen
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GB0716026D0 (en) 2007-08-16 2007-09-26 Norton Healthcare Ltd An inhalable medicament
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JP5658272B2 (ja) 2009-12-17 2015-01-21 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｃｒ２の新規アンタゴニスト及びこれらの使用
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CA2786245A1 (en) 2010-01-29 2011-08-04 Boehringer Ingelheim International Gmbh Substituted naphthyridines and their use as syk kinase inhibitors
EP2569298B1 (en) 2010-05-12 2015-11-25 Boehringer Ingelheim International GmbH Novel ccr2 receptor antagonists, method for producing the same, and use thereof as medicaments
JP5646736B2 (ja) 2010-05-12 2014-12-24 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規ｃｃｒ２受容体アンタゴニスト、これらの製造方法、及び薬物としてのこれらの使用
JP5647339B2 (ja) 2010-05-17 2014-12-24 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｃｒ２アンタゴニスト及びこれらの使用
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JP5721242B2 (ja) 2010-06-01 2015-05-20 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規ｃｃｒ２アンタゴニスト
TR201007108A2 (tr) * 2010-08-25 2012-03-21 B�Lg�� Mahmut Yeni tiotropyum bromür kristali ve üretim yöntemi.@
JP5959537B2 (ja) 2011-01-28 2016-08-02 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 置換ピリジニル−ピリミジン及び医薬としてのその使用
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TR201111589A2 (tr) * 2011-03-03 2012-09-21 Bi̇lgi̇ç Mahmut Tiotropyum bromür susuz kristal formu.
TR201102068A2 (tr) 2011-03-03 2012-09-21 Bi̇lgi̇ç Mahmut Tiotropyum bromür içeren kristal maddeler
WO2012171863A1 (en) 2011-06-16 2012-12-20 Boehringer Ingelheim International Gmbh New selective ccr2 antagonists
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CN106905314A (zh) 2011-11-25 2017-06-30 阿德弗里奥药品有限责任公司 用于制备取代的5‑氟‑1h‑吡唑并吡啶类化合物的方法
CZ304368B6 (cs) 2011-11-28 2014-04-02 Zentiva, K.S. Směsný solvát tiotropium bromidu a způsob jeho přípravy
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Also Published As

Publication number Publication date
CO5550423A2 (es) 2005-08-31
MXPA03011718A (es) 2004-12-06
DE50207943D1 (de) 2006-10-05
CZ302786B6 (cs) 2011-11-09
ES2271280T3 (es) 2007-04-16
CA2450961C (en) 2010-03-30
TWI261589B (en) 2006-09-11
HUP0400333A2 (hu) 2004-12-28
IL159238A (en) 2010-04-15
KR20090031638A (ko) 2009-03-26
EP1401445B1 (de) 2006-08-23
IL159238A0 (en) 2004-06-01
BR0210537A (pt) 2004-06-22
EP1401445A1 (de) 2004-03-31
NO334301B1 (no) 2014-02-03
AU2002345016B2 (en) 2008-04-17
CN1520294A (zh) 2004-08-11
EE200400029A (et) 2004-04-15
CN100586948C (zh) 2010-02-03
EA005813B1 (ru) 2005-06-30
SA02230255B1 (ar) 2006-10-31
ME00412B (me) 2011-10-10
PT1401445E (pt) 2006-10-31
NO20035696D0 (no) 2003-12-19
PE20081305A1 (es) 2008-10-01
ATE337006T1 (de) 2006-09-15
DK1401445T3 (da) 2006-11-27
SI1401445T1 (sl) 2007-02-28
BG108440A (en) 2004-08-31
HRP20031066B1 (en) 2011-10-31
SK522004A3 (en) 2004-06-08
PL364489A1 (en) 2004-12-13
CZ2004120A3 (cs) 2004-05-12
NZ530690A (en) 2005-05-27
JP2005504015A (ja) 2005-02-10
UY27342A1 (es) 2003-02-28
PE20030130A1 (es) 2003-04-02
PL208137B1 (pl) 2011-03-31
KR100971616B1 (ko) 2010-07-22
BG66303B1 (bg) 2013-03-29
HK1068540A1 (en) 2005-04-29
KR20040018285A (ko) 2004-03-02
HRP20031066A2 (en) 2004-04-30
MY122779A (en) 2006-05-31
RS50441B (sr) 2010-03-02
TW200617007A (en) 2006-06-01
AR037491A1 (es) 2004-11-17
EE05316B1 (et) 2010-08-16
HUP0400333A3 (en) 2012-10-29
CA2450961A1 (en) 2003-01-03
YU99703A (sh) 2006-05-25
SK287262B6 (sk) 2010-04-07
KR101011353B1 (ko) 2011-01-28
EA200301293A1 (ru) 2004-08-26
CY1105223T1 (el) 2010-03-03
WO2003000265A1 (de) 2003-01-03
MEP62008A (en) 2011-05-10

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