EE9900524A - N-Triazolyl-2-indolecarboxamides and their Use as CCK-A Agonists - Google Patents
N-Triazolyl-2-indolecarboxamides and their Use as CCK-A AgonistsInfo
- Publication number
- EE9900524A EE9900524A EEP199900524A EEP9900524A EE9900524A EE 9900524 A EE9900524 A EE 9900524A EE P199900524 A EEP199900524 A EE P199900524A EE P9900524 A EEP9900524 A EE P9900524A EE 9900524 A EE9900524 A EE 9900524A
- Authority
- EE
- Estonia
- Prior art keywords
- indolecarboxamides
- cck
- triazolyl
- agonists
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4196—1,2,4-Triazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D249/14—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurology (AREA)
- Endocrinology (AREA)
- Cardiology (AREA)
- Hematology (AREA)
- Psychiatry (AREA)
- Biomedical Technology (AREA)
- Obesity (AREA)
- Neurosurgery (AREA)
- Nutrition Science (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9705850A FR2763337B1 (en) | 1997-05-13 | 1997-05-13 | NOVEL TRIAZOLE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| PCT/FR1998/000905 WO1998051686A1 (en) | 1997-05-13 | 1998-05-06 | N-triazolyl-2-indolecarboxamides and their use as cck-a agonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| EE9900524A true EE9900524A (en) | 2000-06-15 |
Family
ID=9506830
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EEP199900524A EE9900524A (en) | 1997-05-13 | 1998-05-06 | N-Triazolyl-2-indolecarboxamides and their Use as CCK-A Agonists |
Country Status (35)
| Country | Link |
|---|---|
| EP (1) | EP0984960B1 (en) |
| JP (1) | JP2001524980A (en) |
| KR (1) | KR20010012541A (en) |
| CN (1) | CN1263528A (en) |
| AR (1) | AR011729A1 (en) |
| AT (1) | ATE232207T1 (en) |
| AU (1) | AU725530B2 (en) |
| BR (1) | BR9811465A (en) |
| CA (1) | CA2289573A1 (en) |
| CO (1) | CO4940485A1 (en) |
| CZ (1) | CZ289484B6 (en) |
| DE (1) | DE69811223T2 (en) |
| DK (1) | DK0984960T3 (en) |
| DZ (1) | DZ2486A1 (en) |
| EE (1) | EE9900524A (en) |
| ES (1) | ES2190081T3 (en) |
| FR (1) | FR2763337B1 (en) |
| GT (1) | GT199800068A (en) |
| HR (1) | HRP980258B1 (en) |
| HU (1) | HUP0002763A3 (en) |
| ID (1) | ID22911A (en) |
| IL (1) | IL132903A0 (en) |
| IS (1) | IS5235A (en) |
| NO (1) | NO995513L (en) |
| NZ (1) | NZ500637A (en) |
| PL (1) | PL336772A1 (en) |
| RU (1) | RU2175323C2 (en) |
| SI (1) | SI0984960T1 (en) |
| SK (1) | SK154299A3 (en) |
| TR (1) | TR199902795T2 (en) |
| TW (1) | TW396155B (en) |
| UY (1) | UY24997A1 (en) |
| WO (1) | WO1998051686A1 (en) |
| YU (1) | YU57999A (en) |
| ZA (1) | ZA983997B (en) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2802530B1 (en) | 1999-12-17 | 2002-02-22 | Sanofi Synthelabo | NOVEL BRANCHED SUBSTITUTED AMINO DERIVATIVES OF 3-AMINO-1-PHENYL-1H [1,2,4] TRIAZOLE, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| EP1335914A1 (en) * | 2000-10-26 | 2003-08-20 | Sanofi-Synthelabo | Triazole derivatives and pharmaceutical compositions comprising them |
| FR2815963B1 (en) * | 2000-10-26 | 2003-02-28 | Sanofi Synthelabo | NOVEL TRIAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| HUP0004741A2 (en) * | 2000-11-28 | 2002-12-28 | Sanofi-Synthelabo | Chemical process for the preparation of thiazole derivatives and new intermediate |
| CA2463441A1 (en) * | 2001-10-12 | 2003-05-08 | Bayer Pharmaceuticals Corporation | Phenyl substituted 5-membered nitrogen containing heterocycles for the treatment of obesity |
| EP1314733A1 (en) * | 2001-11-22 | 2003-05-28 | Aventis Pharma Deutschland GmbH | Indole-2-carboxamides as factor Xa inhibitors |
| EP1479677A1 (en) * | 2003-05-19 | 2004-11-24 | Aventis Pharma Deutschland GmbH | New indole derivatives as factor xa inhibitors |
| EP1532980A1 (en) | 2003-11-24 | 2005-05-25 | Novo Nordisk A/S | N-heteroaryl indole carboxamides and analogues thereof, for use as glucokinase activators in the treatment of diabetes |
| GB0403038D0 (en) * | 2004-02-11 | 2004-03-17 | Novartis Ag | Organic compounds |
| CA2676222A1 (en) * | 2007-01-26 | 2008-07-31 | Merck & Co., Inc. | Substituted aminopyrimidines as cholecystokinin-1 receptor modulators |
| US8703761B2 (en) * | 2008-07-15 | 2014-04-22 | Novartis Ag | Organic compounds |
| EP2440555B1 (en) * | 2009-06-09 | 2016-05-18 | Actelion Pharmaceuticals Ltd | Fluorinated aminotriazole derivatives |
| EP2490656B1 (en) * | 2009-10-22 | 2017-01-18 | Henkel AG & Co. KGaA | Composition for the treatment of keratinic fibres comprising a nonionic propyleneoxide-modified starch and an anionic polymer |
| CN106928147A (en) * | 2017-03-14 | 2017-07-07 | 华东师范大学 | Tricyclic diterpene analog and preparation method thereof and its application in antiprostate cancer is prepared |
| CN107271623A (en) * | 2017-07-27 | 2017-10-20 | 青岛啤酒股份有限公司 | Beer potableness evaluation method based on human body satiety |
| KR20220150270A (en) | 2019-10-07 | 2022-11-10 | 칼리오페, 인크. | GPR119 agonists |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2701708B1 (en) * | 1993-02-19 | 1995-05-19 | Sanofi Elf | Polysubstituted 2-amido-4-phenylthiazole derivatives, process for their preparation, pharmaceutical composition and use of these derivatives for the preparation of a medicament. |
| FR2703995B1 (en) * | 1993-04-16 | 1995-07-21 | Sanofi Elf | 5-ACYLAMINO 1,2,4-THIADIAZOLES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. |
-
1997
- 1997-05-13 FR FR9705850A patent/FR2763337B1/en not_active Expired - Fee Related
-
1998
- 1998-05-06 ES ES98924383T patent/ES2190081T3/en not_active Expired - Lifetime
- 1998-05-06 WO PCT/FR1998/000905 patent/WO1998051686A1/en not_active Application Discontinuation
- 1998-05-06 TR TR1999/02795T patent/TR199902795T2/en unknown
- 1998-05-06 BR BR9811465-4A patent/BR9811465A/en not_active IP Right Cessation
- 1998-05-06 SI SI9830372T patent/SI0984960T1/en unknown
- 1998-05-06 CA CA002289573A patent/CA2289573A1/en not_active Abandoned
- 1998-05-06 SK SK1542-99A patent/SK154299A3/en unknown
- 1998-05-06 EP EP98924383A patent/EP0984960B1/en not_active Expired - Lifetime
- 1998-05-06 DK DK98924383T patent/DK0984960T3/en active
- 1998-05-06 KR KR1019997010496A patent/KR20010012541A/en not_active Application Discontinuation
- 1998-05-06 AT AT98924383T patent/ATE232207T1/en not_active IP Right Cessation
- 1998-05-06 CZ CZ19994006A patent/CZ289484B6/en not_active IP Right Cessation
- 1998-05-06 YU YU57999A patent/YU57999A/en unknown
- 1998-05-06 PL PL98336772A patent/PL336772A1/en unknown
- 1998-05-06 IL IL13290398A patent/IL132903A0/en unknown
- 1998-05-06 AU AU76599/98A patent/AU725530B2/en not_active Ceased
- 1998-05-06 DZ DZ980096A patent/DZ2486A1/en active
- 1998-05-06 DE DE69811223T patent/DE69811223T2/en not_active Expired - Fee Related
- 1998-05-06 ID IDW991374A patent/ID22911A/en unknown
- 1998-05-06 EE EEP199900524A patent/EE9900524A/en unknown
- 1998-05-06 JP JP54885398A patent/JP2001524980A/en not_active Ceased
- 1998-05-06 NZ NZ500637A patent/NZ500637A/en unknown
- 1998-05-06 HU HU0002763A patent/HUP0002763A3/en unknown
- 1998-05-06 CN CN98807175A patent/CN1263528A/en active Pending
- 1998-05-06 CO CO98024703A patent/CO4940485A1/en unknown
- 1998-05-06 RU RU99125773/04A patent/RU2175323C2/en not_active IP Right Cessation
- 1998-05-11 AR ARP980102152A patent/AR011729A1/en active IP Right Grant
- 1998-05-12 ZA ZA9803997A patent/ZA983997B/en unknown
- 1998-05-12 TW TW087107326A patent/TW396155B/en active
- 1998-05-12 UY UY24997A patent/UY24997A1/en not_active IP Right Cessation
- 1998-05-13 HR HR980258A patent/HRP980258B1/en not_active IP Right Cessation
- 1998-05-20 GT GT199800068A patent/GT199800068A/en unknown
-
1999
- 1999-10-29 IS IS5235A patent/IS5235A/en unknown
- 1999-11-11 NO NO995513A patent/NO995513L/en not_active Application Discontinuation
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