EE200300279A - Toimeaine parendatud vabanemisprofiiliga mikroosakesed ja nende valmistamise meetod - Google Patents

Toimeaine parendatud vabanemisprofiiliga mikroosakesed ja nende valmistamise meetod

Info

Publication number
EE200300279A
EE200300279A EEP200300279A EEP200300279A EE200300279A EE 200300279 A EE200300279 A EE 200300279A EE P200300279 A EEP200300279 A EE P200300279A EE P200300279 A EEP200300279 A EE P200300279A EE 200300279 A EE200300279 A EE 200300279A
Authority
EE
Estonia
Prior art keywords
microparticles
preparation
release profile
improved release
present
Prior art date
Application number
EEP200300279A
Other languages
English (en)
Estonian (et)
Inventor
Kissel Thomas
Fridrich Ruland
Schneider Peter
Original Assignee
Merckle Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE2000161944 external-priority patent/DE10061944A1/de
Priority claimed from DE2001118160 external-priority patent/DE10118160A1/de
Application filed by Merckle Gmbh filed Critical Merckle Gmbh
Publication of EE200300279A publication Critical patent/EE200300279A/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1641Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647Polyesters, e.g. poly(lactide-co-glycolide)

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
EEP200300279A 2000-12-13 2001-12-11 Toimeaine parendatud vabanemisprofiiliga mikroosakesed ja nende valmistamise meetod EE200300279A (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE2000161944 DE10061944A1 (de) 2000-12-13 2000-12-13 Mikropartikel mit verbessertem Freisetzungsprofil
DE2001118160 DE10118160A1 (de) 2001-04-11 2001-04-11 Chitosan enthaltende Mikropartikel
PCT/EP2001/014515 WO2002047664A2 (de) 2000-12-13 2001-12-11 Mikropartikel mit verbessertem freisetzungsprofil und verfahren zu deren herstellung

Publications (1)

Publication Number Publication Date
EE200300279A true EE200300279A (et) 2003-10-15

Family

ID=26007947

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300279A EE200300279A (et) 2000-12-13 2001-12-11 Toimeaine parendatud vabanemisprofiiliga mikroosakesed ja nende valmistamise meetod

Country Status (20)

Country Link
US (1) US20040115277A1 (cs)
EP (1) EP1341522B1 (cs)
JP (1) JP2004515527A (cs)
AT (1) ATE309788T1 (cs)
AU (2) AU2002233239B2 (cs)
BG (1) BG107885A (cs)
BR (1) BR0116077A (cs)
CA (1) CA2431285A1 (cs)
CY (1) CY1105442T1 (cs)
CZ (1) CZ20031559A3 (cs)
DE (1) DE50108114D1 (cs)
DK (1) DK1341522T3 (cs)
EE (1) EE200300279A (cs)
ES (1) ES2250502T3 (cs)
HU (1) HUP0302363A3 (cs)
NO (1) NO20032657L (cs)
PL (1) PL363716A1 (cs)
RU (1) RU2291686C2 (cs)
SK (1) SK7172003A3 (cs)
WO (1) WO2002047664A2 (cs)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1976680A (zh) * 2004-06-28 2007-06-06 康乃尔研究基金会有限公司 从不饱和官能化的多元醇酯得到的可注射微球
GB0416328D0 (en) * 2004-07-21 2004-08-25 Univ Cardiff Use of dry powder compositions for pulmonary delivery
EP1679065A1 (en) * 2005-01-07 2006-07-12 OctoPlus Sciences B.V. Controlled release compositions for interferon based on PEGT/PBT block copolymers
US8628701B2 (en) * 2006-10-31 2014-01-14 Xavier University Of Louisiana Method of micro-encapsulation
UA90013C2 (ru) * 2008-03-19 2010-03-25 Давид Анатолійович Нога Фармацевтическая композиция, содержащая инсулин, и способ его получения
WO2011163469A1 (en) 2010-06-23 2011-12-29 Teva Pharmaceutical Industries Ltd. Hydrated form of anti-inflammatory roflumilast-n-oxide
LT2790675T (lt) * 2011-12-14 2019-11-11 Abraxis Bioscience Llc Polimerinių užpildų panaudojimas dalelių liofilizacijai arba šaldymui
US9308172B2 (en) * 2012-10-26 2016-04-12 Board Of Trustees Of Michigan State University Device and method for encapsulation of hydrophilic materials
JP6151848B2 (ja) * 2013-04-18 2017-06-21 シャンドン ルイ ファーマシューティカル カンパニー リミテッド ゴセレリン徐放性マイクロスフェア医薬組成物
PL3021873T3 (pl) 2013-07-18 2019-01-31 Xalud Therapeutics, Inc. Kompozycja do leczenia choroby zapalnej stawów
WO2015024759A1 (en) * 2013-08-21 2015-02-26 Evonik Industries Ag Process for preparing redispersible powders of water-insoluble, biodegradable polyesters

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3116311B2 (ja) * 1990-06-13 2000-12-11 エーザイ株式会社 マイクロスフィアの製法
IT1243390B (it) * 1990-11-22 1994-06-10 Vectorpharma Int Composizioni farmaceutiche in forma di particelle atte al rilascio controllato di sostanze farmacologicamente attive e procedimento per la loro preparazione.
DE4201179A1 (de) * 1992-01-17 1993-07-22 Alfatec Pharma Gmbh Wirkstoff(e) enthaltendes granulat oder pellet mit einem geruest aus hydrophilen makromolekuelen und verfahren zu seiner herstellung
ATE188375T1 (de) * 1992-11-17 2000-01-15 Yoshitomi Pharmaceutical Ein antipsychotikum enthaltende mikrokugel zur verzögerten freisetzung und verfahren für ihre herstellung
FR2702968B1 (fr) * 1993-03-23 1995-06-23 Lafon Labor Procédé de préparation de particules renfermant un ingrédient actif par extrusion et lyophilisation .
WO1994023699A1 (en) * 1993-04-19 1994-10-27 Medisorb Technologies International L.P. Long-acting treatment by slow-release delivery of antisense oligodeoxyribonucleotides from biodegradable microparticles
US5942253A (en) * 1995-10-12 1999-08-24 Immunex Corporation Prolonged release of GM-CSF
US5792477A (en) * 1996-05-07 1998-08-11 Alkermes Controlled Therapeutics, Inc. Ii Preparation of extended shelf-life biodegradable, biocompatible microparticles containing a biologically active agent
CA2213906A1 (en) * 1996-09-23 1998-03-23 Dusica Maysinger Pharmaceutical composition and method for neuron rescue in ischemic stroke
KR100289471B1 (ko) * 1998-01-19 2001-09-17 김충섭 휀타닐계마취제의이식형서방성제제
US6194006B1 (en) * 1998-12-30 2001-02-27 Alkermes Controlled Therapeutics Inc. Ii Preparation of microparticles having a selected release profile
EP1044683A1 (en) * 1999-04-15 2000-10-18 Debio Recherche Pharmaceutique S.A. One-step dispersion method for the microencapsulation of water soluble substances

Also Published As

Publication number Publication date
WO2002047664A3 (de) 2002-12-27
HK1054689A1 (en) 2003-12-12
CA2431285A1 (en) 2002-06-20
NO20032657D0 (no) 2003-06-12
WO2002047664A2 (de) 2002-06-20
EP1341522B1 (de) 2005-11-16
JP2004515527A (ja) 2004-05-27
AU3323902A (en) 2002-06-24
CZ20031559A3 (cs) 2004-03-17
RU2291686C2 (ru) 2007-01-20
ES2250502T3 (es) 2006-04-16
HUP0302363A2 (hu) 2003-10-28
EP1341522A2 (de) 2003-09-10
NO20032657L (no) 2003-07-18
WO2002047664A8 (de) 2004-03-04
DE50108114D1 (de) 2005-12-22
BG107885A (bg) 2004-01-30
DK1341522T3 (da) 2006-02-13
PL363716A1 (en) 2004-11-29
AU2002233239B2 (en) 2006-05-11
CY1105442T1 (el) 2010-04-28
ATE309788T1 (de) 2005-12-15
US20040115277A1 (en) 2004-06-17
SK7172003A3 (en) 2004-05-04
HUP0302363A3 (en) 2006-07-28
BR0116077A (pt) 2004-02-17

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