EE200300078A - 2,5-dihüdropürasolo-[3,4-D]pürimidin-4-oonid, nende saamine ja kasutamine epilepsiaravimite valmistamiseks ning neid sisaldav farmatseutiline kompositsioon - Google Patents

2,5-dihüdropürasolo-[3,4-D]pürimidin-4-oonid, nende saamine ja kasutamine epilepsiaravimite valmistamiseks ning neid sisaldav farmatseutiline kompositsioon

Info

Publication number
EE200300078A
EE200300078A EEP200300078A EEP200300078A EE200300078A EE 200300078 A EE200300078 A EE 200300078A EE P200300078 A EEP200300078 A EE P200300078A EE P200300078 A EEP200300078 A EE P200300078A EE 200300078 A EE200300078 A EE 200300078A
Authority
EE
Estonia
Prior art keywords
preparation
dihydropyrazolo
pyrimidin
ones
pharmaceutical composition
Prior art date
Application number
EEP200300078A
Other languages
English (en)
Estonian (et)
Inventor
Arnold Thomas
Lankau Hans-Joachim
Unverferth Klaus
Tober Christine
Rundfeldt Chris
Dost Rita
Bern�ster Katrin
Gasparic Antje
Original Assignee
Elbion Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Elbion Ag filed Critical Elbion Ag
Publication of EE200300078A publication Critical patent/EE200300078A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
EEP200300078A 2000-08-26 2001-08-24 2,5-dihüdropürasolo-[3,4-D]pürimidin-4-oonid, nende saamine ja kasutamine epilepsiaravimite valmistamiseks ning neid sisaldav farmatseutiline kompositsioon EE200300078A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10042092A DE10042092A1 (de) 2000-08-26 2000-08-26 Antikonvulsiv wirkende 2,5-Dihydro-pyrazolo(3,4-d)pyrimidin-4-one und Verfahren zu deren Darstellung
PCT/EP2001/009811 WO2002018387A1 (de) 2000-08-26 2001-08-24 Antikonvulsiv wirkende 2,5-dihydro-pyrazolo[3,4-d]pyrimidin-4-one und verfahren zu deren darstellung

Publications (1)

Publication Number Publication Date
EE200300078A true EE200300078A (et) 2004-12-15

Family

ID=7653967

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200300078A EE200300078A (et) 2000-08-26 2001-08-24 2,5-dihüdropürasolo-[3,4-D]pürimidin-4-oonid, nende saamine ja kasutamine epilepsiaravimite valmistamiseks ning neid sisaldav farmatseutiline kompositsioon

Country Status (16)

Country Link
US (1) US20030186997A1 (de)
EP (1) EP1311510A1 (de)
JP (1) JP2004507547A (de)
KR (1) KR20030036734A (de)
CN (1) CN1449397A (de)
AU (1) AU2001282124A1 (de)
BG (1) BG107561A (de)
BR (1) BR0113517A (de)
CA (1) CA2420288A1 (de)
DE (1) DE10042092A1 (de)
EE (1) EE200300078A (de)
HR (1) HRP20030226A2 (de)
IL (1) IL154070A0 (de)
NO (1) NO20030687D0 (de)
RU (1) RU2003108258A (de)
WO (1) WO2002018387A1 (de)

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3165520A (en) * 1965-01-12 Certificate of correction
US3939161A (en) * 1973-10-29 1976-02-17 Abbott Laboratories 1,3-Dimethyl- 1H-pyrazolo(4,3-D) pyrimidine-7 (6H)-ones
US5721356A (en) * 1989-09-15 1998-02-24 Gensia, Inc. Orally active adenosine kinase inhibitors
US5763596A (en) * 1989-09-15 1998-06-09 Metabasis Therapeutics, Inc. C-4' modified adenosine kinase inhibitors
EP0729758A3 (de) * 1995-03-02 1997-10-29 Pfizer Pyrazolopyrimidine und Pyrrolopyrimidine zur Behandlung von neuronalen und anderen Krankheiten
DE19827679A1 (de) * 1998-06-22 1999-12-23 Dresden Arzneimittel Adenosinrezeptoraffine, antikonvulsiv und antiallergisch/antiasthmatisch wirkende Pyrazolo[3,4-d]pyrimidine und Verfahren zu deren Herstellung

Also Published As

Publication number Publication date
DE10042092A1 (de) 2002-03-07
BR0113517A (pt) 2003-07-29
JP2004507547A (ja) 2004-03-11
BG107561A (en) 2003-10-31
WO2002018387A1 (de) 2002-03-07
HRP20030226A2 (en) 2003-06-30
NO20030687L (no) 2003-02-12
KR20030036734A (ko) 2003-05-09
CA2420288A1 (en) 2002-03-07
AU2001282124A1 (en) 2002-03-13
NO20030687D0 (no) 2003-02-12
RU2003108258A (ru) 2005-01-27
EP1311510A1 (de) 2003-05-21
IL154070A0 (en) 2003-07-31
US20030186997A1 (en) 2003-10-02
CN1449397A (zh) 2003-10-15

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