ECSP014053A - Nuevos retinoides selectivos gamma - Google Patents
Nuevos retinoides selectivos gammaInfo
- Publication number
- ECSP014053A ECSP014053A EC2001004053A ECSP014053A ECSP014053A EC SP014053 A ECSP014053 A EC SP014053A EC 2001004053 A EC2001004053 A EC 2001004053A EC SP014053 A ECSP014053 A EC SP014053A EC SP014053 A ECSP014053 A EC SP014053A
- Authority
- EC
- Ecuador
- Prior art keywords
- agonist
- formula
- retinoic acid
- new gamma
- gamma selective
- Prior art date
Links
- 239000000556 agonist Substances 0.000 abstract 2
- SHGAZHPCJJPHSC-YCNIQYBTSA-N all-trans-retinoic acid Chemical compound OC(=O)\C=C(/C)\C=C\C=C(/C)\C=C\C1=C(C)CCCC1(C)C SHGAZHPCJJPHSC-YCNIQYBTSA-N 0.000 abstract 2
- 229930002330 retinoic acid Natural products 0.000 abstract 2
- 229960001727 tretinoin Drugs 0.000 abstract 2
- 206010014561 Emphysema Diseases 0.000 abstract 1
- 208000019693 Lung disease Diseases 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 230000004075 alteration Effects 0.000 abstract 1
- 150000001735 carboxylic acids Chemical class 0.000 abstract 1
- 210000003679 cervix uteri Anatomy 0.000 abstract 1
- 210000001072 colon Anatomy 0.000 abstract 1
- 230000009841 epithelial lesion Effects 0.000 abstract 1
- 210000003238 esophagus Anatomy 0.000 abstract 1
- 210000000867 larynx Anatomy 0.000 abstract 1
- 230000003211 malignant effect Effects 0.000 abstract 1
- 210000000214 mouth Anatomy 0.000 abstract 1
- 210000004400 mucous membrane Anatomy 0.000 abstract 1
- 238000011321 prophylaxis Methods 0.000 abstract 1
- 239000000018 receptor agonist Substances 0.000 abstract 1
- 229940044601 receptor agonist Drugs 0.000 abstract 1
- 150000004492 retinoid derivatives Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
- 210000002105 tongue Anatomy 0.000 abstract 1
- 238000011282 treatment Methods 0.000 abstract 1
- 210000003932 urinary bladder Anatomy 0.000 abstract 1
Landscapes
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Nuevos agonista retinoides selectivos de RAR de la fórmula I: en la que los símbolos tienen os significados definidos en la especificación, y las sales farmacéuticamente activas de los ácidos carboxílicos de la fórmula I, además la invención se refiere al uso de tales agonista receptores de ácido retinoico, en particular a agonista selectivos del receptor y de ácido retinoico (RARy) para el tratamiento del enfisema y de enfermedades pulmonares asociadas, así como la terapia y profilaxis de lesiones epiteliales malignas y premalignas, tumores y alteraciones precancerosas de la membrana mucosa de la boca, lengua, laringe, esófago, vejiga, cuello de la matriz y colon.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10934600 | 2000-05-02 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP014053A true ECSP014053A (es) | 2002-02-25 |
Family
ID=40410320
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2001004053A ECSP014053A (es) | 2000-05-02 | 2001-05-02 | Nuevos retinoides selectivos gamma |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP014053A (es) |
-
2001
- 2001-05-02 EC EC2001004053A patent/ECSP014053A/es unknown
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