ECSP003476A - SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL - Google Patents

SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL

Info

Publication number
ECSP003476A
ECSP003476A ECSP003476A ECSP003476A EC SP003476 A ECSP003476 A EC SP003476A EC SP003476 A ECSP003476 A EC SP003476A EC SP003476 A ECSP003476 A EC SP003476A
Authority
EC
Ecuador
Prior art keywords
useful
pirimidinones
heteroaril
substituted
selective inhibition
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Ashton Hamme
William Neumann
Darin Jones
Melvin L Rueppel
Michael S South
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Priority to ECSP003476 priority Critical patent/ECSP003476A/en
Publication of ECSP003476A publication Critical patent/ECSP003476A/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

El invento se relaciona con los compuestos sustitutos del arilo policíclico y pirimidinonas heteroarilos útiles como inhibidores de las proteasas de serina de la cascada de coagulación y compuestos, composiciones y métodos utilizados para terapias anticuagulantes para el tratamiento y prevención de una variedad de condiciones trombóticas, incluyendo la arteria coronaria y enfermedades cerebrovasculares.The invention relates to polycyclic aryl and heteroaryl pyrimidinones substitute compounds useful as inhibitors of coagulation cascade serine proteases and compounds, compositions and methods used for anticoagulant therapies for the treatment and prevention of a variety of thrombotic conditions, including coronary artery and cerebrovascular diseases.

ECSP003476 2000-05-19 2000-05-19 SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL ECSP003476A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ECSP003476 ECSP003476A (en) 2000-05-19 2000-05-19 SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ECSP003476 ECSP003476A (en) 2000-05-19 2000-05-19 SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL

Publications (1)

Publication Number Publication Date
ECSP003476A true ECSP003476A (en) 2000-10-24

Family

ID=42041102

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP003476 ECSP003476A (en) 2000-05-19 2000-05-19 SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL

Country Status (1)

Country Link
EC (1) ECSP003476A (en)

Similar Documents

Publication Publication Date Title
UY26154A1 (en) ARIL AND HETEROARIL REPLACED POLYCYCLIC PYRIDONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL
UY26157A1 (en) SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL USEFUL FOR THE SELECTIVE I NHIBITION OF THE COAGULATION WATERFALL
UY26156A1 (en) ARIL AND HETEROARIL POLYCYCLIC PIRIMIDONES SUBSTITUTED USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL
CL2022000751A1 (en) shp2 phosphatase inhibitors and methods for their use (divisional application no. 202002419)
EA200801530A1 (en) ANALOGUES OF ARYLPROPIONAMID, ARYLACRYLAMIDE, ARYLPROPINAMIDE OR ARYLMETHYLMANE AS A FACTOR XIA INHIBITORS
UY26155A1 (en) ARIL AND HETEROARIL POLYCLIC SUBSTITUTED PIRAZINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL.
DE60107687D1 (en) CYCLPENTANOINDOLE, MIXTURES CONTAINING SUCH COMPOUNDS AND TREATMENT METHODS
PA8559101A1 (en) INHIBITORS OF THE XA FACTOR AND THE OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION WATERFALL
AR022427A1 (en) PEPTIDIL KETONES HETEROCICLICAS USEFUL AS INHIBITORS OF TRIPTASE
UY27774A1 (en) METALOPROTEIN INHIBITORS OF TRIARIL-OXI-ARIL-ESPIROPIRIMIDINA-2,4,6-TRIONA
PA8619901A1 (en) USEFUL KINOLINES IN THE TREATMENT OF CARDIOVASCULAR DISEASES
EA200400971A1 (en) Fluorine-substituted cycloalkanoylindoles, compositions containing such compounds, and methods of treatment
DE602005014621D1 (en) 3-A4-HETEROCYCLYL-1,2,3-TRIAZOL-1-YLÜ-N-ARYLBENZAMIDES AS INHIBITORS OF CYTOKIN PRODUCTION FOR THE TREATMENT OF CHRONIC INFLAMMATORY DISEASES
EA200600465A1 (en) CASPASE INHIBITORS CONTAINING THE ISOXASOLINE CYCLE
ECSP056106A (en) NEW PHOSPHONIC ACID COMPOUNDS AS INHIBITORS OF SERINA PROTEASAS
ATE367380T1 (en) PIPERAZINYLQUINOLINE DERIVATIVES SUITABLE FOR THE TREATMENT OF CNS DISEASES
AR019477A1 (en) TRIAZOLOPIRIDINS FOR THE TREATMENT OF THROMBOSIS DISORDERS
PT1268463E (en) 4-PYRONES SUBSTITUTED WITH USUAL POLYCYCLIC AERIAL AND HETEROARYL FOR THE SELECTIVE INHIBITION OF COAGULACAO CASCADE
ECSP003476A (en) SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL
MEP48708A (en) Phosphonic acid compounds as inhibitors of serine proteases
ECSP003478A (en) SUBSTITUTED POLYCLIC ARYL AND HETEROARIL URACILS USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL
ECSP003480A (en) SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRAZONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL
ECSP003477A (en) SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PYRIDONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL
CO5160331A1 (en) PIRIDONAS ARILO AND HETEROARILO POLICICLICO SUBSTITUTES USEFUL FOR SELECTIVE INHIBITION OF THE CASCADA DE COAGULACION
WO2001077079A3 (en) Polycyclic aryl and heteroaryl substituted 4-pyridones useful for selective inhibition of the coagulation cascade