CO5160331A1 - PIRIDONAS ARILO AND HETEROARILO POLICICLICO SUBSTITUTES USEFUL FOR SELECTIVE INHIBITION OF THE CASCADA DE COAGULACION - Google Patents

PIRIDONAS ARILO AND HETEROARILO POLICICLICO SUBSTITUTES USEFUL FOR SELECTIVE INHIBITION OF THE CASCADA DE COAGULACION

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Publication number
CO5160331A1
CO5160331A1 CO00040189A CO00040189A CO5160331A1 CO 5160331 A1 CO5160331 A1 CO 5160331A1 CO 00040189 A CO00040189 A CO 00040189A CO 00040189 A CO00040189 A CO 00040189A CO 5160331 A1 CO5160331 A1 CO 5160331A1
Authority
CO
Colombia
Prior art keywords
policiclico
piridonas
coagulacion
cascada
heteroarilo
Prior art date
Application number
CO00040189A
Other languages
Spanish (es)
Inventor
Michael S South
Zeng Qingpeng
Melvin L Rueppel
Original Assignee
Monsanto Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Monsanto Co filed Critical Monsanto Co
Priority to CO00040189A priority Critical patent/CO5160331A1/en
Publication of CO5160331A1 publication Critical patent/CO5160331A1/en

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  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Compuestos de piridona de arilo y heteroarilo policíclicos sustituidos con la fórmula:<EMI FILE="00040189_1" ID="1" IMF=JPEG >que son útiles como inhibidores de proteasas de serina de la cascada de coagulación y a compuestos, composiciones y métodos para terapéutica anticoagulante para el tratamiento y prevención de una diversidad de estados trombóticos entre los que se incluyen enfermedades cerebrovasculares y de las arterias coronarias.Polycyclic aryl and heteroaryl pyridone compounds substituted with the formula: <EMI FILE = "00040189_1" ID = "1" MFI = JPEG> which are useful as inhibitors of coagulation cascade serine proteases and compounds, compositions and methods for anticoagulant therapy for the treatment and prevention of a variety of thrombotic states, including cerebrovascular and coronary artery diseases.

CO00040189A 2000-05-30 2000-05-30 PIRIDONAS ARILO AND HETEROARILO POLICICLICO SUBSTITUTES USEFUL FOR SELECTIVE INHIBITION OF THE CASCADA DE COAGULACION CO5160331A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CO00040189A CO5160331A1 (en) 2000-05-30 2000-05-30 PIRIDONAS ARILO AND HETEROARILO POLICICLICO SUBSTITUTES USEFUL FOR SELECTIVE INHIBITION OF THE CASCADA DE COAGULACION

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CO00040189A CO5160331A1 (en) 2000-05-30 2000-05-30 PIRIDONAS ARILO AND HETEROARILO POLICICLICO SUBSTITUTES USEFUL FOR SELECTIVE INHIBITION OF THE CASCADA DE COAGULACION

Publications (1)

Publication Number Publication Date
CO5160331A1 true CO5160331A1 (en) 2002-05-30

Family

ID=40943531

Family Applications (1)

Application Number Title Priority Date Filing Date
CO00040189A CO5160331A1 (en) 2000-05-30 2000-05-30 PIRIDONAS ARILO AND HETEROARILO POLICICLICO SUBSTITUTES USEFUL FOR SELECTIVE INHIBITION OF THE CASCADA DE COAGULACION

Country Status (1)

Country Link
CO (1) CO5160331A1 (en)

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