EA202192607A1 - Композиции и способы для лечения глазного заболевания - Google Patents
Композиции и способы для лечения глазного заболеванияInfo
- Publication number
- EA202192607A1 EA202192607A1 EA202192607A EA202192607A EA202192607A1 EA 202192607 A1 EA202192607 A1 EA 202192607A1 EA 202192607 A EA202192607 A EA 202192607A EA 202192607 A EA202192607 A EA 202192607A EA 202192607 A1 EA202192607 A1 EA 202192607A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- methods
- compositions
- treatment
- once
- eye disease
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- 239000000203 mixture Substances 0.000 title abstract 2
- 208000030533 eye disease Diseases 0.000 title 1
- 238000002347 injection Methods 0.000 abstract 3
- 239000007924 injection Substances 0.000 abstract 3
- 102000008186 Collagen Human genes 0.000 abstract 1
- 108010035532 Collagen Proteins 0.000 abstract 1
- 206010061218 Inflammation Diseases 0.000 abstract 1
- 208000022873 Ocular disease Diseases 0.000 abstract 1
- 230000003592 biomimetic effect Effects 0.000 abstract 1
- 229920001436 collagen Polymers 0.000 abstract 1
- 230000004054 inflammatory process Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
- 108090000765 processed proteins & peptides Proteins 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 230000008728 vascular permeability Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/39—Connective tissue peptides, e.g. collagen, elastin, laminin, fibronectin, vitronectin, cold insoluble globulin [CIG]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/78—Connective tissue peptides, e.g. collagen, elastin, laminin, fibronectin, vitronectin or cold insoluble globulin [CIG]
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Ophthalmology & Optometry (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Zoology (AREA)
- Gastroenterology & Hepatology (AREA)
- Dermatology (AREA)
- Immunology (AREA)
- Biomedical Technology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Toxicology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Medicinal Preparation (AREA)
Abstract
В различных аспектах и вариантах реализации изобретения предложены способы и фармацевтические композиции для лечения глазного заболевания, связанного с сосудистой проницаемостью или воспалением глаз. В различных аспектах и вариантах реализации изобретение включает введение от около 1 мкг до около 1 мг биомиметического пептида, полученного из коллагена IV или его соли пациенту путем внутриглазной инъекции. Инъекции проводятся с частотой от около одного раза в месяц до около одного раза в два года. В различных вариантах реализации способы и композиции могут обеспечивать мощное действие и длительную продолжительность действия при нечастых интравитреальных инъекциях небольшого объема.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201962824017P | 2019-03-26 | 2019-03-26 | |
PCT/US2020/024972 WO2020198481A1 (en) | 2019-03-26 | 2020-03-26 | Compositions and methods for treating ocular disease |
Publications (1)
Publication Number | Publication Date |
---|---|
EA202192607A1 true EA202192607A1 (ru) | 2022-03-03 |
Family
ID=72609544
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA202192607A EA202192607A1 (ru) | 2019-03-26 | 2020-03-26 | Композиции и способы для лечения глазного заболевания |
Country Status (12)
Country | Link |
---|---|
US (1) | US20230054032A1 (ru) |
EP (1) | EP3946418A4 (ru) |
JP (1) | JP2022527276A (ru) |
KR (1) | KR20210146352A (ru) |
CN (1) | CN113710264A (ru) |
AU (1) | AU2020248438A1 (ru) |
CA (1) | CA3134816A1 (ru) |
EA (1) | EA202192607A1 (ru) |
IL (1) | IL286625A (ru) |
MX (1) | MX2021011727A (ru) |
WO (1) | WO2020198481A1 (ru) |
ZA (1) | ZA202107235B (ru) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN117126233A (zh) * | 2022-05-20 | 2023-11-28 | 杭州禾泰健宇生物科技有限公司 | 一种类肽化合物及其应用 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20100144641A1 (en) * | 2005-09-12 | 2010-06-10 | Popel Aleksander S | Compositions Having Antiangiogenic Activity and Uses Thereof |
EP2649095B1 (en) * | 2010-12-10 | 2021-10-06 | Aleksander S. Popel | Mimetic peptides derived from collagen type iv and their use for treating angiogenesis- and lymphangiogenesis- dependent diseases |
WO2014197892A1 (en) * | 2013-06-07 | 2014-12-11 | The Johns Hopkins University | A biomimetic peptide and biodegradable delivery platform for the treatment of angiogenesis- and lymphangiogenesis-dependent diseases |
US20180339024A1 (en) * | 2015-11-19 | 2018-11-29 | Asclepix Therapeutics, Llc | Peptides with anti-angiogenic, anti-lymphangiogenic, and anti-edemic properties and nanoparticle formulations |
CN110177563A (zh) * | 2016-10-04 | 2019-08-27 | 阿斯克雷佩西治疗公司 | 用于激活tie2信号传导的化合物和方法 |
AU2018266690A1 (en) * | 2017-05-08 | 2019-12-12 | Asclepix Therapeutics, Inc. | Biodegradable microparticles for sustained delivery of anti-angiogenic peptide |
US11674959B2 (en) * | 2017-08-03 | 2023-06-13 | The Johns Hopkins University | Methods for identifying and preparing pharmaceutical agents for activating Tie1 and/or Tie2 receptors |
-
2020
- 2020-03-26 US US17/442,682 patent/US20230054032A1/en active Pending
- 2020-03-26 JP JP2021557369A patent/JP2022527276A/ja active Pending
- 2020-03-26 CN CN202080030026.4A patent/CN113710264A/zh active Pending
- 2020-03-26 CA CA3134816A patent/CA3134816A1/en active Pending
- 2020-03-26 MX MX2021011727A patent/MX2021011727A/es unknown
- 2020-03-26 WO PCT/US2020/024972 patent/WO2020198481A1/en unknown
- 2020-03-26 AU AU2020248438A patent/AU2020248438A1/en active Pending
- 2020-03-26 EA EA202192607A patent/EA202192607A1/ru unknown
- 2020-03-26 KR KR1020217034683A patent/KR20210146352A/ko unknown
- 2020-03-26 EP EP20776493.7A patent/EP3946418A4/en active Pending
-
2021
- 2021-09-23 IL IL286625A patent/IL286625A/en unknown
- 2021-09-27 ZA ZA2021/07235A patent/ZA202107235B/en unknown
Also Published As
Publication number | Publication date |
---|---|
WO2020198481A1 (en) | 2020-10-01 |
MX2021011727A (es) | 2022-01-24 |
EP3946418A4 (en) | 2023-02-22 |
ZA202107235B (en) | 2023-10-25 |
AU2020248438A1 (en) | 2021-10-28 |
CN113710264A (zh) | 2021-11-26 |
KR20210146352A (ko) | 2021-12-03 |
CA3134816A1 (en) | 2020-10-01 |
JP2022527276A (ja) | 2022-06-01 |
EP3946418A1 (en) | 2022-02-09 |
US20230054032A1 (en) | 2023-02-23 |
IL286625A (en) | 2021-12-01 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
JP2020528082A (ja) | 加齢黄斑変性と他の眼疾患の治療用の細胞透過性ペプチドを使用する治療薬の局所送達 | |
JP2017515811A5 (ru) | ||
ES2706059T3 (es) | Composición farmacéutica acuosa que contiene un agente terapéutico biológico y derivado de L-arginina y una inyección que incluye la composición | |
RU2012140704A (ru) | Способ профилактики и/или лечения фиброза и/или помутнения роговицы (варианты), способ получения фармацевтической композиции для профилактики и/или лечения фиброза и/или помутнения роговицы и глазная фармацевтическая композиция | |
RU2006142861A (ru) | Применение вязкоупругой композиции по новому назначению | |
MX2017012506A (es) | Composicion farmaceutica para la prevencion y tratamiento de enfermedades del ojo que contiene, como ingrediente activo, una proteina de fusion en la cual el peptido que penetra el tejido y la preparacion del factor de crecimiento endotelial antivascular se fusionan. | |
NO980195L (no) | Cyklosporinderivater med anti-HIV-effekt | |
WO2006119128A8 (en) | Vascular targeting of ocular neovascularization | |
MX2021009526A (es) | Composiciones para suministro farmacologico, para la administracion ocular de agentes terapeuticos, y metodos de uso de las mismas. | |
GB0716600D0 (en) | Ophthalmic medicine composition | |
JP2018504984A5 (ru) | ||
PH12021551232A1 (en) | Haloallylamine compounds and application thereof | |
ES2672099T3 (es) | Antagonistas del receptor NK-1 para el tratamiento de la neovascularización corneal | |
RU2018145017A (ru) | Применение сиролимуса для лечения экссудативной возрастной макулярной дегенерации с персистирующим отеком | |
AU2016258001B2 (en) | Injectable depot formulations | |
EA202192607A1 (ru) | Композиции и способы для лечения глазного заболевания | |
AR123570A1 (es) | Tratamientos para el edema macular diabético y la agudeza visual disminuida | |
MX2022003820A (es) | Metodos de tratamiento para modificar la hermodinamica. | |
MX2021005077A (es) | Peptidos y composiciones farmaceuticas para tratar enfermedades oculares. | |
EA202191130A1 (ru) | Фармацевтическая композиция для лечения апластической анемии | |
RU2012127869A (ru) | Устойчивые водные композиции пролекарств агонистов простагладина и способы их применения | |
JP6944463B2 (ja) | 眼疾患の治療のための組成物及び方法 | |
MX2022003051A (es) | Formulaciones para la administracion de farmacos. | |
MX2021015796A (es) | Composiciones y metodos para tratar enfermedades oculares. | |
MD722Z (ru) | Устройство и метод лечения старческой катаракты |