EA201891102A1 - Термодинамически стабильная кристаллическая модификация 2-метил-n-(5-метил-1,3,4-оксадиазол-2-ил)-3-(метилсульфонил)-4-(трифторметил)бензамида - Google Patents

Термодинамически стабильная кристаллическая модификация 2-метил-n-(5-метил-1,3,4-оксадиазол-2-ил)-3-(метилсульфонил)-4-(трифторметил)бензамида

Info

Publication number
EA201891102A1
EA201891102A1 EA201891102A EA201891102A EA201891102A1 EA 201891102 A1 EA201891102 A1 EA 201891102A1 EA 201891102 A EA201891102 A EA 201891102A EA 201891102 A EA201891102 A EA 201891102A EA 201891102 A1 EA201891102 A1 EA 201891102A1
Authority
EA
Eurasian Patent Office
Prior art keywords
methyl
oxadiazol
methylsulfonyl
benzamide
trifluoromethyl
Prior art date
Application number
EA201891102A
Other languages
English (en)
Inventor
Арним Кён
Кристофер Хью Розингер
Кристиан Вальдрафф
Бритта Оленик
Биргит Кайль
Бенедикт Мель
Original Assignee
Байер Кропсайенс Акциенгезельшафт
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Байер Кропсайенс Акциенгезельшафт filed Critical Байер Кропсайенс Акциенгезельшафт
Publication of EA201891102A1 publication Critical patent/EA201891102A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C07D271/113—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Toxicology (AREA)
  • Medicinal Preparation (AREA)

Abstract

Описана термодинамически стабильная кристаллическая модификация 2-метил-N-(5-метил-1,3,4-оксадиазол-2-ил)-3-(метилсульфонил)-4-(трифторметил)бензамида. Эта термодинамически стабильная кристаллическая модификация имеет особые преимущества в стабильности суспензионных составов.
EA201891102A 2015-11-09 2016-11-04 Термодинамически стабильная кристаллическая модификация 2-метил-n-(5-метил-1,3,4-оксадиазол-2-ил)-3-(метилсульфонил)-4-(трифторметил)бензамида EA201891102A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP15193615 2015-11-09
PCT/EP2016/076620 WO2017080912A1 (de) 2015-11-09 2016-11-04 Thermodynamisch stabile kristallmodifikation von 2-methyl-n-(5-methyl-1,3,4-oxadiazol-2-yl)-3-(methylsulfonyl)-4-(trifluoromethyl)benzamid

Publications (1)

Publication Number Publication Date
EA201891102A1 true EA201891102A1 (ru) 2018-11-30

Family

ID=54541996

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201891102A EA201891102A1 (ru) 2015-11-09 2016-11-04 Термодинамически стабильная кристаллическая модификация 2-метил-n-(5-метил-1,3,4-оксадиазол-2-ил)-3-(метилсульфонил)-4-(трифторметил)бензамида

Country Status (12)

Country Link
US (1) US10336716B2 (ru)
EP (1) EP3374351A1 (ru)
JP (1) JP2018534294A (ru)
CN (1) CN108349916A (ru)
AU (1) AU2016352566A1 (ru)
BR (1) BR112018009386A8 (ru)
CA (1) CA3004360A1 (ru)
EA (1) EA201891102A1 (ru)
MX (1) MX2018005818A (ru)
UY (1) UY36982A (ru)
WO (1) WO2017080912A1 (ru)
ZA (1) ZA201802523B (ru)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10152459A1 (de) 2001-10-24 2003-05-08 Bayer Cropscience Ag Neue thermodynamisch stabile Kristallmodifikation von [2-(2-Chloro-4-mesyl-benzoyl)cyclohexane-1,3-dione]
HUE029871T2 (en) * 2011-03-22 2017-04-28 Bayer Ip Gmbh N- (1,3,4-oxadiazol-2-yl) -arylcarboxylic acids and their use as herbicides

Also Published As

Publication number Publication date
ZA201802523B (en) 2019-01-30
MX2018005818A (es) 2018-08-01
WO2017080912A1 (de) 2017-05-18
CN108349916A (zh) 2018-07-31
AU2016352566A1 (en) 2018-05-10
JP2018534294A (ja) 2018-11-22
US10336716B2 (en) 2019-07-02
EP3374351A1 (de) 2018-09-19
BR112018009386A2 (pt) 2018-11-13
BR112018009386A8 (pt) 2019-02-26
UY36982A (es) 2017-06-30
US20180319754A1 (en) 2018-11-08
CA3004360A1 (en) 2017-05-18

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