EA201700114A1 - Капсаициноиды и их применение в качестве лекарственных средств - Google Patents
Капсаициноиды и их применение в качестве лекарственных средствInfo
- Publication number
- EA201700114A1 EA201700114A1 EA201700114A EA201700114A EA201700114A1 EA 201700114 A1 EA201700114 A1 EA 201700114A1 EA 201700114 A EA201700114 A EA 201700114A EA 201700114 A EA201700114 A EA 201700114A EA 201700114 A1 EA201700114 A1 EA 201700114A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- drug
- applicable
- treatment
- capsaicinoids
- medicines
- Prior art date
Links
- 239000003814 drug Substances 0.000 title abstract 5
- YKPUWZUDDOIDPM-SOFGYWHQSA-N capsaicin Chemical compound COC1=CC(CNC(=O)CCCC\C=C\C(C)C)=CC=C1O YKPUWZUDDOIDPM-SOFGYWHQSA-N 0.000 title abstract 2
- 229940079593 drug Drugs 0.000 abstract 4
- 208000030507 AIDS Diseases 0.000 abstract 1
- 208000036142 Viral infection Diseases 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 230000003110 anti-inflammatory effect Effects 0.000 abstract 1
- 230000000840 anti-viral effect Effects 0.000 abstract 1
- 206010003246 arthritis Diseases 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 230000009385 viral infection Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K36/00—Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
- A61K36/18—Magnoliophyta (angiosperms)
- A61K36/185—Magnoliopsida (dicotyledons)
- A61K36/81—Solanaceae (Potato family), e.g. tobacco, nightshade, tomato, belladonna, capsicum or jimsonweed
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Natural Medicines & Medicinal Plants (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Microbiology (AREA)
- Alternative & Traditional Medicine (AREA)
- Mycology (AREA)
- Medical Informatics (AREA)
- Botany (AREA)
- Biotechnology (AREA)
- Engineering & Computer Science (AREA)
- Virology (AREA)
- Physiology (AREA)
- Nutrition Science (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Communicable Diseases (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- AIDS & HIV (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Plant Substances (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
В настоящем изобретении предложено лекарственное средство, содержащее капсаициноид, обладающее противовирусным действием и применимое для лечения вирусных инфекций и ВИЧ/СПИД. Лекарственное средство также обладает усиливающим нейропластичность действием и применимо для лечения стресса и других психологических состояний. Кроме того, лекарственное средство обладает противовоспалительным действием и применимо для лечения артрита. Лекарственное средство также обладает антибактериальным действием.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
AU2014903253A AU2014903253A0 (en) | 2014-08-19 | Viral therapy | |
PCT/AU2015/000454 WO2016025977A1 (en) | 2014-08-19 | 2015-07-31 | Capsaicinoids and uses thereof as medicaments |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201700114A1 true EA201700114A1 (ru) | 2017-06-30 |
Family
ID=55349992
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201700114A EA201700114A1 (ru) | 2014-08-19 | 2015-07-31 | Капсаициноиды и их применение в качестве лекарственных средств |
Country Status (8)
Country | Link |
---|---|
US (1) | US20170239198A1 (ru) |
EP (1) | EP3182968A4 (ru) |
KR (1) | KR20170066344A (ru) |
AU (1) | AU2015306063A1 (ru) |
CA (1) | CA2961766A1 (ru) |
EA (1) | EA201700114A1 (ru) |
MA (1) | MA40496A (ru) |
WO (1) | WO2016025977A1 (ru) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP3534961A4 (en) | 2016-11-02 | 2020-05-27 | Centrexion Therapeutics Corporation | STABLE AQUEOUS INJECTABLE CAPSAICIN FORMULATIONS AND MEDICAL USES THEREOF |
CN111201015A (zh) | 2017-07-20 | 2020-05-26 | 中枢疗法公司 | 使用辣椒素治疗疼痛的方法和组合物 |
US11447444B1 (en) | 2019-01-18 | 2022-09-20 | Centrexion Therapeutics Corporation | Capsaicinoid prodrug compounds and their use in treating medical conditions |
US11254659B1 (en) | 2019-01-18 | 2022-02-22 | Centrexion Therapeutics Corporation | Capsaicinoid prodrug compounds and their use in treating medical conditions |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4486450B1 (en) * | 1980-07-14 | 1998-07-28 | Joel E Bernstein | Method of treating psoriatic skin and composition |
US4599342A (en) * | 1984-01-16 | 1986-07-08 | The Procter & Gamble Company | Pharmaceutical products providing enhanced analgesia |
US20030082249A1 (en) * | 2001-10-26 | 2003-05-01 | Ovation Pharmaceuticals | Compositions containing capsaicin and its derivatives, and their use in treating mucositis |
FR2849992B1 (fr) * | 2003-01-17 | 2007-03-16 | Inst Phytoceutic | Composition pour une administration par voie orale contenant des capsaicinoides |
US20040224037A1 (en) * | 2003-04-28 | 2004-11-11 | Gonzalo Romero-Matos | Devastating treatment against hiv/aids with capsaicin |
-
2015
- 2015-07-31 AU AU2015306063A patent/AU2015306063A1/en not_active Abandoned
- 2015-07-31 EP EP15833869.9A patent/EP3182968A4/en not_active Withdrawn
- 2015-07-31 EA EA201700114A patent/EA201700114A1/ru unknown
- 2015-07-31 MA MA040496A patent/MA40496A/fr unknown
- 2015-07-31 WO PCT/AU2015/000454 patent/WO2016025977A1/en active Application Filing
- 2015-07-31 KR KR1020177007621A patent/KR20170066344A/ko unknown
- 2015-07-31 US US15/505,152 patent/US20170239198A1/en not_active Abandoned
- 2015-07-31 CA CA2961766A patent/CA2961766A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
MA40496A (fr) | 2017-06-28 |
US20170239198A1 (en) | 2017-08-24 |
AU2015306063A1 (en) | 2017-04-13 |
EP3182968A4 (en) | 2018-05-09 |
CA2961766A1 (en) | 2016-02-25 |
WO2016025977A1 (en) | 2016-02-25 |
EP3182968A1 (en) | 2017-06-28 |
KR20170066344A (ko) | 2017-06-14 |
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