EA201491165A1 - Вагинальное кольцо, содержащее dhea или сульфат dhea и возможно агент, модулирующий высвобождение активного ингредиента, полезное для увеличения овариального резерва у женщин и для облегчения симптомов, связанных с менопаузой - Google Patents
Вагинальное кольцо, содержащее dhea или сульфат dhea и возможно агент, модулирующий высвобождение активного ингредиента, полезное для увеличения овариального резерва у женщин и для облегчения симптомов, связанных с менопаузойInfo
- Publication number
- EA201491165A1 EA201491165A1 EA201491165A EA201491165A EA201491165A1 EA 201491165 A1 EA201491165 A1 EA 201491165A1 EA 201491165 A EA201491165 A EA 201491165A EA 201491165 A EA201491165 A EA 201491165A EA 201491165 A1 EA201491165 A1 EA 201491165A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- mans
- dhea
- man
- active ingredient
- women
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
- A61K31/5685—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone having an oxo group in position 17, e.g. androsterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
- A61K9/0036—Devices retained in the vagina or cervix for a prolonged period, e.g. intravaginal rings, medicated tampons, medicated diaphragms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Reproductive Health (AREA)
- Epidemiology (AREA)
- Gynecology & Obstetrics (AREA)
- Urology & Nephrology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Endocrinology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Inorganic Chemistry (AREA)
- Pregnancy & Childbirth (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Infusion, Injection, And Reservoir Apparatuses (AREA)
- Orthopedics, Nursing, And Contraception (AREA)
Abstract
Вагинальное кольцо с длительным высвобождением, содержащее дегидроэпиандростерон (DHEA), сульфат дегидроэпиандростерона (DHEA-S) или его фармацевтически приемлемую соль в качестве активного агента и возможно агент, модулирующий высвобождение активного ингредиента, где количество активного ингредиента составляет от 1 до 32 мас.% относительно общей массы композиции, и модулятор выбран из поливинилпирролидона K-30, лактозы, микрокристаллической целлюлозы и лаурилсульфата натрия. Вагинальное кольцо по настоящему изобретению может быть использовано для увеличения овариального резерва у женщин, для применения в качестве лекарственного средства во вспомогательных репродуктивных программах и для облегчения симптомов, связанных с менопаузой, таких как симптомы атрофии вульвы и влагалища, и половой дисфункции у женщин в постменопаузе.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/IB2011/056023 WO2013098592A1 (es) | 2011-12-29 | 2011-12-29 | Anillo vaginal que comprende dhea o dhea sulfato y opcionalmente un agente modulador de la liberación del principio activo, útil para aumentar la reserva ovárica en mujeres y para aliviar síntomas asociados a la menopausia |
Publications (2)
Publication Number | Publication Date |
---|---|
EA201491165A1 true EA201491165A1 (ru) | 2014-12-30 |
EA027633B1 EA027633B1 (ru) | 2017-08-31 |
Family
ID=48696405
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201491165A EA027633B1 (ru) | 2011-12-29 | 2011-12-29 | Вагинальное кольцо, содержащее dhea или сульфат dhea и возможно агент, модулирующий высвобождение активного ингредиента, полезное для увеличения овариального резерва у женщин и для облегчения симптомов, связанных с менопаузой |
Country Status (12)
Country | Link |
---|---|
US (1) | US9066956B2 (ru) |
EP (1) | EP2799042A4 (ru) |
JP (1) | JP5887424B2 (ru) |
KR (1) | KR101622861B1 (ru) |
CN (1) | CN104271084B (ru) |
BR (1) | BR112014014308A2 (ru) |
CA (1) | CA2860133C (ru) |
CR (1) | CR20140270A (ru) |
EA (1) | EA027633B1 (ru) |
MX (1) | MX350336B (ru) |
NI (1) | NI201400067A (ru) |
WO (1) | WO2013098592A1 (ru) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP3272333A1 (en) | 2016-07-22 | 2018-01-24 | Chemo Research, S.L. | Vaginal composition comprising a combination of estrogen and vitamin d |
CN108537785B (zh) * | 2018-04-04 | 2021-04-30 | 北京大学人民医院 | 一种子宫超声微蠕动视频处理方法 |
US10918649B2 (en) * | 2019-06-21 | 2021-02-16 | The Population Council, Inc. | System for providing birth control |
WO2021111385A2 (en) | 2019-12-06 | 2021-06-10 | Prathima Chowdary | Sustained release estrogen vaginal ring pessary for treatment of atrophy, cystitis and uterovaginal prolapse |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5776923A (en) | 1993-01-19 | 1998-07-07 | Endorecherche, Inc. | Method of treating or preventing osteoporosis by adminstering dehydropiandrosterone |
ATE275957T1 (de) | 1993-01-19 | 2004-10-15 | Endorech Inc | Therapeutische verwendungen und verabreichungsysteme von dehydroepiandrosteron |
ES2098193B1 (es) | 1995-07-21 | 1997-12-01 | Gomez Jesus Calderon | Nueva formulacion farmaceutica de dehidroepiandrosterona para aplicacion topica percutanea. |
WO1999021562A1 (en) | 1997-10-28 | 1999-05-06 | Asivi, Llc | Treatment of female sexual dysfunction |
US20020099003A1 (en) | 1997-10-28 | 2002-07-25 | Wilson Leland F. | Treatment of female sexual dysfunction with vasoactive agents, particularly vasoactive intestinal polypeptide and agonists thereof |
WO2002076426A2 (en) | 2001-03-27 | 2002-10-03 | Galen (Chemicals) Limited | Intravaginal drug delivery devices for the administration of an antimicrobial agent |
EP1350541A1 (de) | 2002-04-04 | 2003-10-08 | Jenapharm GmbH & Co. KG | Verwendung von einem Dehydroepiandrosteron und einem Estradiol Derivat zur Herstellung einer pharmazeutischen Zubereitung zur Behandlung klimakterischer Beschwerden in der Postmenopause |
US8501718B2 (en) | 2005-11-08 | 2013-08-06 | American Infertility Of New York | Androgen treatment in females |
US8501719B2 (en) | 2005-11-08 | 2013-08-06 | American Infertility Of New York | Androgen treatment in females |
US9375436B2 (en) | 2004-10-26 | 2016-06-28 | Norbert Gleicher | Androgen treatment in females |
US7615544B2 (en) | 2004-10-26 | 2009-11-10 | American Infertility Of New York | Method of improving cumulative embryo score and quantity of fertilized oocytes, increasing euploidy rate and of normalizing ovarian function using an androgen such as dehydroepiandrosterone |
US8067400B2 (en) | 2004-10-26 | 2011-11-29 | American Infertility Of New York | Androgen treatment in females |
US20060089308A1 (en) | 2004-10-26 | 2006-04-27 | American Infertility Of New York | Method of improving ovulation induction using an androgen such as dehydroepiandrosterone |
EP1890704A1 (en) * | 2005-12-16 | 2008-02-27 | Lyle Corporate Development, Inc. | Regeneration of vaginal tissue with non-systemic vaginal administration of estrogen |
SG195525A1 (en) * | 2007-06-26 | 2013-12-30 | Warner Chilcott Co Llc | Intravaginal drug delivery devices for the delivery of macromolecules and water-soluble drugs |
US8268806B2 (en) * | 2007-08-10 | 2012-09-18 | Endorecherche, Inc. | Pharmaceutical compositions |
-
2011
- 2011-12-29 WO PCT/IB2011/056023 patent/WO2013098592A1/es active Application Filing
- 2011-12-29 JP JP2014549544A patent/JP5887424B2/ja not_active Expired - Fee Related
- 2011-12-29 KR KR1020147020208A patent/KR101622861B1/ko active IP Right Grant
- 2011-12-29 US US14/367,826 patent/US9066956B2/en not_active Expired - Fee Related
- 2011-12-29 BR BR112014014308A patent/BR112014014308A2/pt not_active Application Discontinuation
- 2011-12-29 CN CN201180076298.9A patent/CN104271084B/zh not_active Expired - Fee Related
- 2011-12-29 EP EP11879080.7A patent/EP2799042A4/en not_active Withdrawn
- 2011-12-29 MX MX2014007957A patent/MX350336B/es active IP Right Grant
- 2011-12-29 CA CA2860133A patent/CA2860133C/en not_active Expired - Fee Related
- 2011-12-29 EA EA201491165A patent/EA027633B1/ru not_active IP Right Cessation
-
2014
- 2014-06-11 CR CR20140270A patent/CR20140270A/es unknown
- 2014-06-20 NI NI201400067A patent/NI201400067A/es unknown
Also Published As
Publication number | Publication date |
---|---|
NI201400067A (es) | 2016-02-15 |
CR20140270A (es) | 2014-10-31 |
BR112014014308A2 (pt) | 2017-06-13 |
US9066956B2 (en) | 2015-06-30 |
KR20140109987A (ko) | 2014-09-16 |
EP2799042A1 (en) | 2014-11-05 |
MX350336B (es) | 2017-09-04 |
US20150004214A1 (en) | 2015-01-01 |
CN104271084A (zh) | 2015-01-07 |
CA2860133C (en) | 2016-10-11 |
MX2014007957A (es) | 2015-11-06 |
JP2015506933A (ja) | 2015-03-05 |
WO2013098592A1 (es) | 2013-07-04 |
KR101622861B1 (ko) | 2016-05-19 |
EA027633B1 (ru) | 2017-08-31 |
EP2799042A4 (en) | 2015-02-11 |
CN104271084B (zh) | 2017-03-01 |
CA2860133A1 (en) | 2013-07-04 |
JP5887424B2 (ja) | 2016-03-16 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA201491165A1 (ru) | Вагинальное кольцо, содержащее dhea или сульфат dhea и возможно агент, модулирующий высвобождение активного ингредиента, полезное для увеличения овариального резерва у женщин и для облегчения симптомов, связанных с менопаузой | |
PE20130524A1 (es) | Forma farmaceutica parenteral, que libera inhibidores de aromatasa y gestagenos para el tratamiento de endometrosis | |
PE20080273A1 (es) | Composicion farmaceutica que contiene un progestageno, un estrogeno y un acido tetrahidrofolico | |
HRP20240121T1 (hr) | Kontracepcija na bazi drospirenona za pacijenticu s viškom tjelesne težine | |
BR112013024558A2 (pt) | pessários de uso único | |
HRP20192026T4 (hr) | Formulacija tableta od neratinib maleata | |
HRP20220902T3 (hr) | Pripravci i njihova upotreba u liječenju multiple skleroze | |
NZ596844A (en) | Monolithic intravaginal rings comprising progesterone and methods of making and uses thereof | |
AR081670A1 (es) | Composicion farmaceutica que comprende drospirenona y kit anticonceptivo | |
JP2011527709A5 (ru) | ||
CL2011002847A1 (es) | Uso de (r)-7-cloro-n-(quinuclidin-3-il)benzo[b]tiofeno-2-carboxamida o una sal farmaceuticamente aceptable del mismo y un inhibidor de acetilcolinesterasa para preparar un medicamento util para mejorar la cognicion. | |
Sato et al. | Interactions of vasopressin, prostaglandins, and cAMP in rat renal papillary collecting tubule cells in culture | |
AR095691A1 (es) | FORMULACIÓN DE L-5-METILTETRAHIDROFOLATO DE CALCIO AMORFO (L-5-MTHF-Ca), PROCEDIMIENTO, USO | |
JP2018527305A5 (ru) | ||
HRP20230762T1 (hr) | Nalmefen za smanjenje konzumacije alkohola u specifičnim ciljnim populacijama | |
PL1879572T3 (pl) | Zastosowanie antagonistów oksytocyny i/lub wazopresyny we wspomaganym rozrodzie | |
AR088704A1 (es) | Anillo vaginal que comprende dhea o dhea sulfato y opcionalmente un agente modulador de la liberacion del principio activo, util para aumentar la reserva ovarica en mujeres y para aliviar sintomas asociados a la menopausia | |
ECSP14008170A (es) | Anillo vaginal que comprende dhea o dhea sulfato y opcionalmente un agente modulador de la liberación del principio activo, útil para aumentar la reserva ovárica en mujeres y para aliviar síntomas asociados a la menopausia | |
PE20090805A1 (es) | COMBINACION DE DROSPIRENONA Y 17ß-ESTRADIOL COMO CONTRACEPTIVO ORAL | |
PH12015502326A1 (en) | Progesterone receptor antagonist dosage form | |
DOP2014000143A (es) | Anillo vaginal que comprende dhea o dhea sulfato y opcionalmente un agente modulador de la liberación del principio activo, útil para aumentar la reserva ovárica en mujeres y para aliviar síntomas asociados a la menopausia | |
CO7151514A2 (es) | Anillo vaginal que comprende dhea o dhea sulfato y opcionalmente un agente modulador de la liberación del principio activo, útil para aumentar la reserva ovárica en mujeres y para aliviar síntomas asociados a la menopausia. | |
GT201400124A (es) | Anillo vaginal que comprende dhea o dhea sulfato y opcionalmente un agente modulador de la liberación del principio activo, útil para aumentar la reserva ovárica en mujeres y para aliviar síntomas asociados a la menopausia | |
PE20142116A1 (es) | Anillo vaginal que comprende dhea o dhea sulfato y opcionalmente un agente modulador de la liberacion del principio activo, util para aumentar la reserva ovarica en mujeres y para aliviar sintomas asociados a la menopausia | |
DOP2007000122A (es) | Forma farmacologica peroral para anticoncepcion |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM |
|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): RU |