EA201290817A1 - Твердые фармацевтические композиции рамиприла и безилата амлодипина и их получение - Google Patents
Твердые фармацевтические композиции рамиприла и безилата амлодипина и их получениеInfo
- Publication number
- EA201290817A1 EA201290817A1 EA201290817A EA201290817A EA201290817A1 EA 201290817 A1 EA201290817 A1 EA 201290817A1 EA 201290817 A EA201290817 A EA 201290817A EA 201290817 A EA201290817 A EA 201290817A EA 201290817 A1 EA201290817 A1 EA 201290817A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- pharmaceutical compositions
- ramipril
- amylodypine
- dilated
- free
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
- A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
- A61J3/00—Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms
- A61J3/10—Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms into the form of compressed tablets
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4422—1,4-Dihydropyridines, e.g. nifedipine, nicardipine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B65—CONVEYING; PACKING; STORING; HANDLING THIN OR FILAMENTARY MATERIAL
- B65B—MACHINES, APPARATUS OR DEVICES FOR, OR METHODS OF, PACKAGING ARTICLES OR MATERIALS; UNPACKING
- B65B3/00—Packaging plastic material, semiliquids, liquids or mixed solids and liquids, in individual containers or receptacles, e.g. bags, sacks, boxes, cartons, cans, or jars
- B65B3/04—Methods of, or means for, filling the material into the containers or receptacles
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B65—CONVEYING; PACKING; STORING; HANDLING THIN OR FILAMENTARY MATERIAL
- B65D—CONTAINERS FOR STORAGE OR TRANSPORT OF ARTICLES OR MATERIALS, e.g. BAGS, BARRELS, BOTTLES, BOXES, CANS, CARTONS, CRATES, DRUMS, JARS, TANKS, HOPPERS, FORWARDING CONTAINERS; ACCESSORIES, CLOSURES, OR FITTINGS THEREFOR; PACKAGING ELEMENTS; PACKAGES
- B65D11/00—Containers having bodies formed by interconnecting or uniting two or more rigid, or substantially rigid, components made wholly or mainly of plastics material
- B65D11/20—Details of walls made of plastics material
Abstract
Настоящее изобретение относится к твердым стабильным фармацевтическим композициям фиксированных доз, содержащим рамиприл, безилат амлодипина и фармацевтически приемлемые эксципиенты, и к их получению.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN417DE2010 | 2010-02-24 | ||
PCT/IB2010/051616 WO2011104588A2 (en) | 2010-02-24 | 2010-04-14 | Solid pharmaceutical formulations of ramipril and amlodipine besylate, and their preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201290817A1 true EA201290817A1 (ru) | 2013-01-30 |
Family
ID=42786564
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201290817A EA201290817A1 (ru) | 2010-02-24 | 2010-04-14 | Твердые фармацевтические композиции рамиприла и безилата амлодипина и их получение |
Country Status (28)
Country | Link |
---|---|
US (1) | US20130146496A1 (ru) |
EP (1) | EP2538924B1 (ru) |
JP (1) | JP5719385B2 (ru) |
KR (1) | KR20120130761A (ru) |
CN (1) | CN102781430B (ru) |
AR (1) | AR080256A1 (ru) |
AU (1) | AU2010346977A1 (ru) |
BR (1) | BR112012021203A2 (ru) |
CA (1) | CA2790817A1 (ru) |
CL (1) | CL2012002341A1 (ru) |
CR (1) | CR20120432A (ru) |
EA (1) | EA201290817A1 (ru) |
EC (1) | ECSP12012121A (ru) |
ES (1) | ES2483154T3 (ru) |
GT (1) | GT201200248A (ru) |
MA (1) | MA34130B1 (ru) |
MX (1) | MX2012009689A (ru) |
NI (1) | NI201200136A (ru) |
PE (1) | PE20130004A1 (ru) |
PL (1) | PL2538924T3 (ru) |
SG (1) | SG183449A1 (ru) |
SI (1) | SI2538924T1 (ru) |
TN (1) | TN2012000363A1 (ru) |
TW (1) | TW201138767A (ru) |
UA (1) | UA105285C2 (ru) |
UY (1) | UY33243A (ru) |
WO (1) | WO2011104588A2 (ru) |
ZA (1) | ZA201205559B (ru) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UA113977C2 (xx) * | 2012-02-17 | 2017-04-10 | Фармацевтична композиція з покращеною стабільністю | |
PL227900B1 (pl) | 2012-11-15 | 2018-01-31 | Adamed Spolka Z Ograniczona Odpowiedzialnoscia | Kompozycja farmaceutyczna zawierająca inhibitor ACE i bloker kanałów wapniowych, sposób jej wytwarzania i jednostka dawkowania zawierająca tę kompozycję |
CN104546773B (zh) * | 2015-01-30 | 2018-12-11 | 华润赛科药业有限责任公司 | 一种高稳定性苯磺酸氨氯地平片及其制备方法 |
WO2016207824A2 (en) * | 2015-06-23 | 2016-12-29 | Dr. Reddy's Laboratories Ltd | A stable pharmaceutical composition comprising ramipril and/or amlodipine |
EP3501502A1 (en) * | 2017-12-20 | 2019-06-26 | Midas Pharma GmbH | Fixed dosed pharmaceutical compositions comprising amlodipine, ramipril and atorvastatin |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3633496A1 (de) | 1986-10-02 | 1988-04-14 | Hoechst Ag | Kombination von angiotensin-converting-enzyme-hemmern mit calciumantagonisten sowie deren verwendung in arzneimitteln |
PT804229E (pt) | 1995-03-16 | 2003-06-30 | Pfizer | Utilizacao de amlodipina de um dos seus sais ou defelodipina em combinacao com um inibidor da en zima de conversao da angiotensina (ace) para no fabrico de um medicamento destinado ao tratamento da insuficiencia cardiaca congestiva nao isquemica |
WO2001015674A2 (en) | 1999-08-30 | 2001-03-08 | Aventis Pharma Deutschland Gmbh | Use of inhibitors of the renin-angiotensin system in the prevention of cardiovascular events |
WO2005079772A2 (en) | 2004-02-18 | 2005-09-01 | Sepracor Inc. | Combination of (s)-amlodipine and an ace inhibitor, and methods for reducing hypertension |
HUP0401170A2 (en) * | 2004-06-10 | 2006-09-28 | Richter Gedeon Vegyeszet | Pharmaceutical composition comprising amlodipine besilate and lisinopril dihydrate and process for |
EP1817007A2 (en) * | 2004-11-05 | 2007-08-15 | King Pharmaceuticals Research and Development Inc. | Stabilized individually coated ramipril particles, compositions and methods |
CN101272791A (zh) * | 2005-09-28 | 2008-09-24 | 特瓦制药工业有限公司 | 苯磺酸氨氯地平和盐酸贝那普利的稳定的组合 |
AU2005336956A1 (en) * | 2005-09-28 | 2007-04-12 | Teva Pharmaceutical Industries Ltd. | Stable combinations of amlodipine besylate and benazepril hydrochloride |
TWI399223B (zh) * | 2006-09-15 | 2013-06-21 | Daiichi Sankyo Co Ltd | 奧美沙坦酯及氨氯地平之固體劑型 |
US20080096863A1 (en) * | 2006-10-19 | 2008-04-24 | Torrent Pharmaceuticals Limited | Stable pharmaceutical compositions of calcium channel blocker and an ACE inhibitor |
-
2010
- 2010-04-14 UA UAA201210997A patent/UA105285C2/ru unknown
- 2010-04-14 WO PCT/IB2010/051616 patent/WO2011104588A2/en active Application Filing
- 2010-04-14 AU AU2010346977A patent/AU2010346977A1/en not_active Abandoned
- 2010-04-14 MA MA35197A patent/MA34130B1/fr unknown
- 2010-04-14 EP EP10717277.7A patent/EP2538924B1/en active Active
- 2010-04-14 SG SG2012062238A patent/SG183449A1/en unknown
- 2010-04-14 PL PL10717277T patent/PL2538924T3/pl unknown
- 2010-04-14 MX MX2012009689A patent/MX2012009689A/es unknown
- 2010-04-14 BR BR112012021203A patent/BR112012021203A2/pt not_active IP Right Cessation
- 2010-04-14 EA EA201290817A patent/EA201290817A1/ru unknown
- 2010-04-14 SI SI201030701T patent/SI2538924T1/sl unknown
- 2010-04-14 JP JP2012554429A patent/JP5719385B2/ja not_active Expired - Fee Related
- 2010-04-14 ES ES10717277.7T patent/ES2483154T3/es active Active
- 2010-04-14 CN CN201080064730.8A patent/CN102781430B/zh not_active Expired - Fee Related
- 2010-04-14 KR KR1020127022080A patent/KR20120130761A/ko not_active Application Discontinuation
- 2010-04-14 PE PE2012001353A patent/PE20130004A1/es not_active Application Discontinuation
- 2010-04-14 CA CA2790817A patent/CA2790817A1/en not_active Abandoned
-
2011
- 2011-02-23 TW TW100105890A patent/TW201138767A/zh unknown
- 2011-02-23 AR ARP110100551A patent/AR080256A1/es unknown
- 2011-02-24 UY UY0001033243A patent/UY33243A/es not_active Application Discontinuation
-
2012
- 2012-07-17 TN TNP2012000363A patent/TN2012000363A1/en unknown
- 2012-07-24 ZA ZA2012/05559A patent/ZA201205559B/en unknown
- 2012-08-20 CR CR20120432A patent/CR20120432A/es unknown
- 2012-08-20 NI NI201200136A patent/NI201200136A/es unknown
- 2012-08-23 EC ECSP12012121 patent/ECSP12012121A/es unknown
- 2012-08-23 GT GT201200248A patent/GT201200248A/es unknown
- 2012-08-23 US US13/592,958 patent/US20130146496A1/en not_active Abandoned
- 2012-08-23 CL CL2012002341A patent/CL2012002341A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
NI201200136A (es) | 2012-10-29 |
GT201200248A (es) | 2014-05-14 |
MA34130B1 (fr) | 2013-04-03 |
ZA201205559B (en) | 2013-09-25 |
TW201138767A (en) | 2011-11-16 |
AU2010346977A1 (en) | 2012-09-13 |
AR080256A1 (es) | 2012-03-21 |
MX2012009689A (es) | 2012-09-12 |
CN102781430B (zh) | 2015-09-09 |
PL2538924T3 (pl) | 2014-10-31 |
UY33243A (es) | 2011-09-30 |
SG183449A1 (en) | 2012-09-27 |
KR20120130761A (ko) | 2012-12-03 |
JP2013520485A (ja) | 2013-06-06 |
US20130146496A1 (en) | 2013-06-13 |
WO2011104588A3 (en) | 2012-04-19 |
PE20130004A1 (es) | 2013-02-01 |
EP2538924B1 (en) | 2014-05-21 |
CA2790817A1 (en) | 2011-09-01 |
EP2538924A2 (en) | 2013-01-02 |
BR112012021203A2 (pt) | 2016-05-17 |
WO2011104588A2 (en) | 2011-09-01 |
ES2483154T3 (es) | 2014-08-05 |
CR20120432A (es) | 2012-11-29 |
UA105285C2 (ru) | 2014-04-25 |
CL2012002341A1 (es) | 2012-11-30 |
TN2012000363A1 (en) | 2014-01-30 |
JP5719385B2 (ja) | 2015-05-20 |
CN102781430A (zh) | 2012-11-14 |
ECSP12012121A (es) | 2012-09-28 |
SI2538924T1 (sl) | 2014-09-30 |
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