EA200701595A1 - Устойчивые к спиртам лекарственные формы - Google Patents

Устойчивые к спиртам лекарственные формы

Info

Publication number
EA200701595A1
EA200701595A1 EA200701595A EA200701595A EA200701595A1 EA 200701595 A1 EA200701595 A1 EA 200701595A1 EA 200701595 A EA200701595 A EA 200701595A EA 200701595 A EA200701595 A EA 200701595A EA 200701595 A1 EA200701595 A1 EA 200701595A1
Authority
EA
Eurasian Patent Office
Prior art keywords
sustainable
medicine forms
alcohols
alcohols medicine
forms
Prior art date
Application number
EA200701595A
Other languages
English (en)
Other versions
EA015615B1 (ru
Inventor
Ричард О. Мэннион
Уильям Х. Маккенна
Эдвард П. О'Доннелл
Хелен Кэтлин Данагер
Джеффри Джерард Хэйз
Хассан Мохаммад
Дерек Аллен Пратер
Харджит Тамбер
Мелколм Уолден
Стив Уайтлок
Вольфганг Флайшер
Удо Хан
Кристоф Спитцлай
Кристиан Лойнер
Original Assignee
Еуро-Селтик С. А.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36297284&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA200701595(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB0501638.1A external-priority patent/GB0501638D0/en
Priority claimed from PCT/GB2005/050014 external-priority patent/WO2005079760A1/en
Application filed by Еуро-Селтик С. А. filed Critical Еуро-Селтик С. А.
Publication of EA200701595A1 publication Critical patent/EA200701595A1/ru
Publication of EA015615B1 publication Critical patent/EA015615B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/36—Opioid-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)

Abstract

Составы с контролируемым высвобождением опиоида, устойчивые к экстракции опиоида спиртом.
EA200701595A 2005-01-28 2006-01-27 Устойчивые к спиртам лекарственные формы EA015615B1 (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GBGB0501638.1A GB0501638D0 (en) 2005-01-28 2005-01-28 Particulates
PCT/GB2005/050014 WO2005079760A1 (en) 2004-02-12 2005-02-11 Particulates
US67050605P 2005-04-12 2005-04-12
US73033905P 2005-10-26 2005-10-26
PCT/EP2006/000727 WO2006079550A2 (en) 2005-01-28 2006-01-27 Alcohol resistant dosage forms

Publications (2)

Publication Number Publication Date
EA200701595A1 true EA200701595A1 (ru) 2008-02-28
EA015615B1 EA015615B1 (ru) 2011-10-31

Family

ID=36297284

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200701595A EA015615B1 (ru) 2005-01-28 2006-01-27 Устойчивые к спиртам лекарственные формы

Country Status (14)

Country Link
US (1) US20070259045A1 (ru)
EP (4) EP3228308A1 (ru)
JP (1) JP5704789B2 (ru)
KR (2) KR20090029856A (ru)
CN (1) CN101132772B (ru)
AP (1) AP2274A (ru)
AU (1) AU2006208627B8 (ru)
BR (1) BRPI0606339A2 (ru)
CA (1) CA2594373A1 (ru)
EA (1) EA015615B1 (ru)
GE (1) GEP20105052B (ru)
IL (1) IL184858A (ru)
MX (1) MX2007009162A (ru)
WO (1) WO2006079550A2 (ru)

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EP3228308A1 (en) 2017-10-11
IL184858A (en) 2016-03-31
EP1771160A2 (en) 2007-04-11
IL184858A0 (en) 2007-12-03
MX2007009162A (es) 2007-10-23
US20070259045A1 (en) 2007-11-08
WO2006079550A2 (en) 2006-08-03
BRPI0606339A2 (pt) 2009-06-16
AP2007004099A0 (en) 2007-08-31
CN101132772A (zh) 2008-02-27
CN101132772B (zh) 2012-05-09
JP5704789B2 (ja) 2015-04-22
EA015615B1 (ru) 2011-10-31
EP2319499A1 (en) 2011-05-11
AU2006208627B2 (en) 2009-08-06
KR20070104443A (ko) 2007-10-25
WO2006079550A3 (en) 2006-12-14
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AP2274A (en) 2011-08-19
KR20090029856A (ko) 2009-03-23
AU2006208627A1 (en) 2006-08-03
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AU2006208627B8 (en) 2009-08-13
JP2008528534A (ja) 2008-07-31

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