EA200300741A1 - METHOD OF OBTAINING MALEAT AMLODIPINA - Google Patents
METHOD OF OBTAINING MALEAT AMLODIPINAInfo
- Publication number
- EA200300741A1 EA200300741A1 EA200300741A EA200300741A EA200300741A1 EA 200300741 A1 EA200300741 A1 EA 200300741A1 EA 200300741 A EA200300741 A EA 200300741A EA 200300741 A EA200300741 A EA 200300741A EA 200300741 A1 EA200300741 A1 EA 200300741A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- obtaining
- amlodipine
- amlodipina
- maleat
- product
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
- C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Способ получения малеата амлодипина, включающий взаимодействие амлодипина или его соли - продукта присоединения кислоты с малеиновой кислотой в кислой среде, с получением при этом продукта малеата амлодипина. Способ позволяет получить малеат амлодипина, по существу не содержащий аспартат амлодипина.Международная заявка была опубликована вместе с отчетом о международном поиске.The method of obtaining amlodipine maleate, including the interaction of amlodipine or its salt - the product of the addition of acid with maleic acid in an acidic medium, with the receipt of the product of amlodipine maleate. The method allows to obtain amlodipine maleate, essentially not containing aslodate amlodipine. The international application was published together with an international search report.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US25861200P | 2000-12-29 | 2000-12-29 | |
US80934301A | 2001-03-16 | 2001-03-16 | |
PCT/NL2001/000607 WO2002053542A1 (en) | 2000-12-29 | 2001-08-15 | Process for making amlodipine maleate |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200300741A1 true EA200300741A1 (en) | 2003-10-30 |
EA008141B1 EA008141B1 (en) | 2007-04-27 |
Family
ID=41639550
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200300741A EA008141B1 (en) | 2000-12-29 | 2001-08-15 | Process for making amlodipine maleate |
Country Status (4)
Country | Link |
---|---|
KR (1) | KR20030066782A (en) |
EA (1) | EA008141B1 (en) |
GE (1) | GEP20063946B (en) |
OA (1) | OA13133A (en) |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK161312C (en) * | 1982-03-11 | 1991-12-09 | Pfizer | CHANGES FOR THE PREPARATION FOR THE PREPARATION OF 2-Amino-CO-Methyl-4-Methyl-4-Methyl-4-Methyl-4-Methyl-4-Methyl-4-Methyl-2-D-Hydroxy |
PL189666B1 (en) * | 1998-04-09 | 2005-09-30 | Adamed Sp Z Oo | Method of obtaining amlopidine benzenosulphonate |
-
2001
- 2001-08-15 EA EA200300741A patent/EA008141B1/en unknown
- 2001-08-15 KR KR10-2003-7008835A patent/KR20030066782A/en not_active Application Discontinuation
- 2001-08-15 OA OA1200300166A patent/OA13133A/en unknown
- 2001-08-15 GE GE5245A patent/GEP20063946B/en unknown
Also Published As
Publication number | Publication date |
---|---|
OA13133A (en) | 2006-12-13 |
EA008141B1 (en) | 2007-04-27 |
GEP20063946B (en) | 2006-10-25 |
KR20030066782A (en) | 2003-08-09 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EA200300118A1 (en) | TETRAHYDROPYRIDINO- OR PIPERIDINO-HETEROCYCLIC DERIVATIVES | |
WO2002042418A3 (en) | 3-hydroxypropionic acid and other organic compounds | |
TR199901238T2 (en) | 3-thiocarbamoylpyrazole derivatives as parasitic. | |
BR0111981A (en) | substituted pyridine herbicides | |
CR7728A (en) | NEW ESPIROCONDENSED KINAZOLINS AND ITS USE AS PHOSPHODESTERASE INHIBITORS | |
ATE370936T1 (en) | SUBSTITUTED PYRAZINE OR PYRIDINE DERIVATIVES AS GLUCOCINASE ACTIVATORS | |
DE69531331D1 (en) | Phenylpiperidine derivatives as neurokinin antagonists | |
BRPI0414599A (en) | substituted pyrrol indoles | |
DE60134682D1 (en) | Optical amplifier with rod-shaped amplification medium pumped from the end side | |
ITTO20000111V0 (en) | FOLDABLE STRUCTURE, AS AN EXHIBITION STRUCTURE. | |
ATE247726T1 (en) | TARGETED ELECTROCHEMICAL REDUCTION OF HALOGENATED 4-AMINO-PICOLINIC ACIDS | |
WO2001064834A8 (en) | Novel nucleic acids and polypeptides | |
EA200401559A1 (en) | TECHNOLOGY OF PRESSING WOOD-FIBER PLATES OF MEDIUM DENSITY | |
ATE309220T1 (en) | SUBSTITUTED 1,2,3,4-TETRAHYDROCINOLINE-2-CARBOXYLIC ACID DERIVATIVES | |
FI962639A0 (en) | Diaryl-5,6-fused heterocyclic acids as leukotriene antagonists | |
ATE309356T1 (en) | DESIGNED FLUORESCENT PROTEINS WITH LONG WAVELENGTHS | |
WO2004009564A3 (en) | Co-surfactants based on aldehydes | |
EA200100852A1 (en) | DERIVATIVES OF RESORT | |
YU12397A (en) | NOVEL PYRIMIDO [1,2-a] INDOLES | |
DE60207399D1 (en) | ALKOXYCARBONYLAMINOBENOIC ACID OR ALKOXYCARBONYLAMINOTETROZOLYLPHENYL DERIVATIVES AS IP ANTAGONISTS | |
NO20011287L (en) | Wood stove with swivel plate, as well as method | |
EA200300741A1 (en) | METHOD OF OBTAINING MALEAT AMLODIPINA | |
EA200200887A1 (en) | METHOD OF MANUFACTURING ELECTRODE AND ELECTRODE | |
CR7011A (en) | PROCESS TO MAKE AMLODIPINE MALEATE | |
DE60323748D1 (en) | 1,3-DIAZA-DIBENZOAZULENE AS INHIBITORS OF THE PRODUCTION FOR THEIR PRODUCTION |