EA200200160A1 - Аналоги псевдомицина с n-ацильной боковой цепью - Google Patents

Аналоги псевдомицина с n-ацильной боковой цепью

Info

Publication number
EA200200160A1
EA200200160A1 EA200200160A EA200200160A EA200200160A1 EA 200200160 A1 EA200200160 A1 EA 200200160A1 EA 200200160 A EA200200160 A EA 200200160A EA 200200160 A EA200200160 A EA 200200160A EA 200200160 A1 EA200200160 A1 EA 200200160A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pseudomycin
analogues
acyl
lateral chains
antifungal agents
Prior art date
Application number
EA200200160A
Other languages
English (en)
Inventor
Мэттью Дэвид Белво
Шу Хьюи Чен
Кристофер Уилльям Доеске
Сара Линн Хеллман
Джеймс Эндрю Джеймисон
Лоренс Эдвард Паттерсон
Майкл Джон Родригез
Ксиченг Дэвид Сун
Уилльям Уилсон Тернер
Венкатрагхаван Васудеван
Марк Джеймс Звейфел
Original Assignee
Эли Лилли Энд Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Эли Лилли Энд Компани filed Critical Эли Лилли Энд Компани
Publication of EA200200160A1 publication Critical patent/EA200200160A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Communicable Diseases (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Epoxy Compounds (AREA)

Abstract

Описаны полусинтетические соединения псевдомицина, имеющие структуру (I), которые могут быть пригодны в качестве противогрибковых агентов или промежуточных соединений для разработки противогрибковых агентов.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200200160A 1999-07-15 2000-06-08 Аналоги псевдомицина с n-ацильной боковой цепью EA200200160A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14398999P 1999-07-15 1999-07-15
PCT/US2000/015017 WO2001005814A1 (en) 1999-07-15 2000-06-08 Pseudomycin n-acyl side-chain analogs

Publications (1)

Publication Number Publication Date
EA200200160A1 true EA200200160A1 (ru) 2002-08-29

Family

ID=22506582

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200200160A EA200200160A1 (ru) 1999-07-15 2000-06-08 Аналоги псевдомицина с n-ацильной боковой цепью

Country Status (11)

Country Link
EP (1) EP1200460A1 (ru)
JP (1) JP2003505397A (ru)
CN (1) CN1360593A (ru)
AU (1) AU5724900A (ru)
BR (1) BR0012447A (ru)
CA (1) CA2379851A1 (ru)
EA (1) EA200200160A1 (ru)
HU (1) HUP0202347A2 (ru)
MX (1) MXPA02000321A (ru)
NO (1) NO20020193L (ru)
WO (1) WO2001005814A1 (ru)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102004051023A1 (de) * 2004-10-20 2006-05-04 Bayer Healthcare Ag Desoxo-Nonadepsipeptide
DE102004051025A1 (de) 2004-10-20 2006-04-27 Bayer Healthcare Ag Substituierte Nonadepsipeptide
DE102004053410A1 (de) 2004-11-05 2006-05-11 Bayer Healthcare Ag Cyclische Nonadepsipeptidamide
DE102006018080A1 (de) 2006-04-13 2007-10-18 Aicuris Gmbh & Co. Kg Lysobactinamide
SG175855A1 (en) * 2009-05-04 2011-12-29 Prometic Biosciences Inc Substituted aromatic compounds and pharmaceutical uses thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5576298A (en) * 1992-11-30 1996-11-19 Research And Development Institute, Inc. At Montana State University Peptides from pseudomonas syringae possessing broad-spectrum antibiotic activity

Also Published As

Publication number Publication date
HUP0202347A2 (en) 2002-10-28
CA2379851A1 (en) 2001-01-25
AU5724900A (en) 2001-02-05
MXPA02000321A (es) 2002-06-21
EP1200460A1 (en) 2002-05-02
CN1360593A (zh) 2002-07-24
NO20020193D0 (no) 2002-01-14
JP2003505397A (ja) 2003-02-12
NO20020193L (no) 2002-03-14
BR0012447A (pt) 2002-04-02
WO2001005814A1 (en) 2001-01-25

Similar Documents

Publication Publication Date Title
TR199902400T2 (xx) Fungusit etkinlik g�steren terkiplerin birle�imleri.
EA200100773A1 (ru) Замещенные 1-гетероциклические диариламины
PA8527001A1 (es) Poliarilcarboxamidas utiles como agentes reductores de lipidos
BR9804214A (pt) Compostos.
EA200000098A1 (ru) 4-АМИНОПИРРОЛ(3,2-d)ПИРИМИДИНЫ В КАЧЕСТВЕ АНТАГОНИСТОВ РЕЦЕПТОРА НЕЙРОПЕПТИДА Y
PT1140840E (pt) Difenilureias substituidas com (.)-carboxiarilo como inibidores de raf-quinase
TR200101906T2 (tr) Antiviral ajanlar olarak kuinolinkarboksamitler
EA200500017A1 (ru) Новые соединения
DK1131315T3 (da) Polyhydroxylerede heterocykliske derivater som antikoagulanter
EA200000251A1 (ru) Производные резорцинола
ES2172864T3 (es) 2-metoxibenzofenonas fungicidas.
ID29076A (id) Kombinasi senyawa aktif fungisida
EA200300593A1 (ru) Соединения пиперазинилпиразинов в качестве агонистов или антагонистов серотонин 5-ht2 рецептора
PT892780E (pt) Analogos de m-amidino fenilo como inibidores do factor xa
EA200100012A1 (ru) Мостиковые инденопирролокарбазолы
BRPI0516981A (pt) inibidores de mif
EA200200732A1 (ru) Замещенные производные фенилпиперазина, их получение и применение
TR200103119T2 (tr) Göz kurumasının tedavisi için madde.
EA200300450A1 (ru) Фармацевтические растворы соединений модафинила
EA200000975A1 (ru) 6-(2-гало-4-алкоксифенил)триазолпиримидины с фунгицидным действием
EA200100854A1 (ru) Кальций-литические соединения
BR9916507A (pt) Proteìnas
PT882726E (pt) Carbazol-carboxamidas como agonistas 5-ht1f
EA200100517A1 (ru) Антагонисты 5ht1 для антидепрессантной терапии
EA200100852A1 (ru) Производные резорцина