DOP2012000056A - Agente terapeutico para trastornos de ansiedad - Google Patents
Agente terapeutico para trastornos de ansiedadInfo
- Publication number
- DOP2012000056A DOP2012000056A DO2012000056A DO2012000056A DOP2012000056A DO P2012000056 A DOP2012000056 A DO P2012000056A DO 2012000056 A DO2012000056 A DO 2012000056A DO 2012000056 A DO2012000056 A DO 2012000056A DO P2012000056 A DOP2012000056 A DO P2012000056A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- therapeutic agent
- anxiety disorders
- agent
- sìmìlar
- prophylaxis
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
- C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
- C07D491/052—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being six-membered
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Se proporciona un agente para el tratamiento y/o profilaxis de un trastorno de ansiedad que comprende, como un ingrediente activo, un derivado de tiazol representado por la fórmula (I) en donde R representa arilo o similar, y R2 representa piridilo o similar, o una de sus sales farmacéutìcamente aceptables, y sìmìlar.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2009202894 | 2009-09-02 |
Publications (1)
Publication Number | Publication Date |
---|---|
DOP2012000056A true DOP2012000056A (es) | 2012-06-30 |
Family
ID=43649340
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DO2012000056A DOP2012000056A (es) | 2009-09-02 | 2012-03-01 | Agente terapeutico para trastornos de ansiedad |
Country Status (31)
Country | Link |
---|---|
US (1) | US20120172362A1 (es) |
EP (1) | EP2474544B1 (es) |
JP (1) | JP5663485B2 (es) |
KR (2) | KR20120047311A (es) |
CN (1) | CN102482271A (es) |
AU (1) | AU2010290424C1 (es) |
BR (1) | BR112012004850A2 (es) |
CA (1) | CA2772922C (es) |
CL (1) | CL2012000533A1 (es) |
CY (1) | CY1119483T1 (es) |
DK (1) | DK2474544T3 (es) |
DO (1) | DOP2012000056A (es) |
EA (1) | EA023728B1 (es) |
ES (1) | ES2643840T3 (es) |
GE (1) | GEP20156225B (es) |
HR (1) | HRP20171418T1 (es) |
HU (1) | HUE036543T2 (es) |
IL (1) | IL218320A (es) |
LT (1) | LT2474544T (es) |
MA (1) | MA33619B1 (es) |
ME (1) | ME02877B (es) |
MX (1) | MX2012002529A (es) |
NZ (1) | NZ598754A (es) |
PL (1) | PL2474544T3 (es) |
PT (1) | PT2474544T (es) |
RS (1) | RS56401B1 (es) |
SI (1) | SI2474544T1 (es) |
TN (1) | TN2012000093A1 (es) |
UA (1) | UA113383C2 (es) |
WO (1) | WO2011027806A1 (es) |
ZA (1) | ZA201202347B (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7718808B2 (en) * | 2003-12-26 | 2010-05-18 | Kyowa Hakko Kirin Co., Ltd. | Thiazole derivatives |
MA41090A (fr) * | 2014-12-03 | 2017-10-10 | H Lundbeck As | Antagoniste de a2a faiblement dosé pour le traitement du tdah et de la maladie de parkinson |
JOP20200093A1 (ar) | 2015-01-09 | 2017-06-16 | Kyowa Kirin Co Ltd | طريقة لإنتاج مشتق ثيازول |
JO3544B1 (ar) * | 2015-03-19 | 2020-07-05 | Kyowa Kirin Co Ltd | عامل علاجي للاختلال الوظيفي في الفص الجبهي |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5543415A (en) | 1992-07-08 | 1996-08-06 | Kyowa Hakko Kogyo Co., Ltd. | Antidepressants |
EP1666041A3 (en) | 1997-09-05 | 2008-04-02 | Kyowa Hakko Kogyo Co., Ltd. | Xanthine derivatives for treating neurodegenerative disorders |
US20040152659A1 (en) * | 1999-05-12 | 2004-08-05 | Fujisawa Pharmaceutical Co. Ltd. | Method for the treatment of parkinson's disease comprising administering an A1A2a receptor dual antagonist |
WO2000069464A1 (fr) * | 1999-05-12 | 2000-11-23 | Fujisawa Pharmaceutical Co., Ltd. | Nouvelle utilisation |
WO2003022283A1 (en) * | 2001-09-13 | 2003-03-20 | Schering Corporation | Combination of an adenosine a2a receptor antagonist and an antidepressant or anxiolytic |
US6620811B2 (en) | 2001-11-19 | 2003-09-16 | Hoffmann-La Roche Inc. | Isonicotin- and nicotinamide derivatives of benzothiazoles |
CN1787821A (zh) * | 2003-06-10 | 2006-06-14 | 协和发酵工业株式会社 | 一种治疗焦虑症的方法 |
US7718808B2 (en) * | 2003-12-26 | 2010-05-18 | Kyowa Hakko Kirin Co., Ltd. | Thiazole derivatives |
US20100280023A1 (en) * | 2005-06-23 | 2010-11-04 | Kyowa Hakko Kogyo Co., Ltd. | Thiazole derivatives |
JP5121453B2 (ja) * | 2005-08-02 | 2013-01-16 | 協和発酵キリン株式会社 | 睡眠障害の治療および/または予防剤 |
UA110097C2 (uk) * | 2009-09-02 | 2015-11-25 | Терапевтичний агент для лікування розладів настрою |
-
2010
- 2010-02-09 UA UAA201203922A patent/UA113383C2/uk unknown
- 2010-09-02 JP JP2011529927A patent/JP5663485B2/ja not_active Expired - Fee Related
- 2010-09-02 NZ NZ598754A patent/NZ598754A/en not_active IP Right Cessation
- 2010-09-02 RS RS20170966A patent/RS56401B1/sr unknown
- 2010-09-02 AU AU2010290424A patent/AU2010290424C1/en not_active Ceased
- 2010-09-02 MX MX2012002529A patent/MX2012002529A/es active IP Right Grant
- 2010-09-02 WO PCT/JP2010/064989 patent/WO2011027806A1/ja active Application Filing
- 2010-09-02 EA EA201270360A patent/EA023728B1/ru not_active IP Right Cessation
- 2010-09-02 ES ES10813754.8T patent/ES2643840T3/es active Active
- 2010-09-02 PT PT108137548T patent/PT2474544T/pt unknown
- 2010-09-02 SI SI201031544T patent/SI2474544T1/sl unknown
- 2010-09-02 BR BR112012004850-3A patent/BR112012004850A2/pt not_active Application Discontinuation
- 2010-09-02 EP EP10813754.8A patent/EP2474544B1/en active Active
- 2010-09-02 ME MEP-2017-233A patent/ME02877B/me unknown
- 2010-09-02 CA CA2772922A patent/CA2772922C/en not_active Expired - Fee Related
- 2010-09-02 CN CN2010800392099A patent/CN102482271A/zh active Pending
- 2010-09-02 LT LTEP10813754.8T patent/LT2474544T/lt unknown
- 2010-09-02 US US13/393,068 patent/US20120172362A1/en not_active Abandoned
- 2010-09-02 PL PL10813754T patent/PL2474544T3/pl unknown
- 2010-09-02 HU HUE10813754A patent/HUE036543T2/hu unknown
- 2010-09-02 DK DK10813754.8T patent/DK2474544T3/en active
- 2010-09-02 GE GEAP201012648A patent/GEP20156225B/en unknown
- 2010-09-02 KR KR1020127008310A patent/KR20120047311A/ko active Application Filing
- 2010-09-02 KR KR1020177010507A patent/KR20170044768A/ko not_active Application Discontinuation
-
2012
- 2012-02-26 IL IL218320A patent/IL218320A/en active IP Right Grant
- 2012-02-27 TN TNP2012000093A patent/TN2012000093A1/en unknown
- 2012-02-29 CL CL2012000533A patent/CL2012000533A1/es unknown
- 2012-03-01 DO DO2012000056A patent/DOP2012000056A/es unknown
- 2012-03-30 ZA ZA2012/02347A patent/ZA201202347B/en unknown
- 2012-03-30 MA MA34734A patent/MA33619B1/fr unknown
-
2017
- 2017-09-19 HR HRP20171418TT patent/HRP20171418T1/hr unknown
- 2017-10-04 CY CY20171101029T patent/CY1119483T1/el unknown
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