DK72282A - Fremgangsmaade til fremstilling af bis-estere af 1,1-alkandioler med 2beta-acetoxymethyl-2alfa-methyl-(5r)penam-3alfa-carboxylsyre-1,1-dioxid og en 6-acylaminopenicillansyre eller farmaceutisk acceptable salte deraf - Google Patents
Fremgangsmaade til fremstilling af bis-estere af 1,1-alkandioler med 2beta-acetoxymethyl-2alfa-methyl-(5r)penam-3alfa-carboxylsyre-1,1-dioxid og en 6-acylaminopenicillansyre eller farmaceutisk acceptable salte deraf Download PDFInfo
- Publication number
- DK72282A DK72282A DK72282A DK72282A DK72282A DK 72282 A DK72282 A DK 72282A DK 72282 A DK72282 A DK 72282A DK 72282 A DK72282 A DK 72282A DK 72282 A DK72282 A DK 72282A
- Authority
- DK
- Denmark
- Prior art keywords
- methyl
- penam
- acetoxymethyl
- dioxide
- esters
- Prior art date
Links
- 125000004494 ethyl ester group Chemical group 0.000 abstract 3
- 239000003242 anti bacterial agent Substances 0.000 abstract 2
- 150000002148 esters Chemical class 0.000 abstract 2
- 239000000543 intermediate Substances 0.000 abstract 1
- -1 mono-substituted methyl Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/236,407 US4364957A (en) | 1979-09-26 | 1981-02-20 | Bis-esters of alkanediols as antibacterial agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK72282A true DK72282A (da) | 1982-08-21 |
Family
ID=22889370
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK72282A DK72282A (da) | 1981-02-20 | 1982-02-19 | Fremgangsmaade til fremstilling af bis-estere af 1,1-alkandioler med 2beta-acetoxymethyl-2alfa-methyl-(5r)penam-3alfa-carboxylsyre-1,1-dioxid og en 6-acylaminopenicillansyre eller farmaceutisk acceptable salte deraf |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US4364957A (OSRAM) |
| EP (1) | EP0059046B1 (OSRAM) |
| JP (1) | JPS57154192A (OSRAM) |
| AT (1) | ATE15044T1 (OSRAM) |
| AU (1) | AU527894B2 (OSRAM) |
| CA (1) | CA1176242A (OSRAM) |
| DE (1) | DE3265503D1 (OSRAM) |
| DK (1) | DK72282A (OSRAM) |
| ES (1) | ES8304992A1 (OSRAM) |
| GR (1) | GR75173B (OSRAM) |
| IE (1) | IE52902B1 (OSRAM) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4478748A (en) * | 1981-02-20 | 1984-10-23 | Pfizer Inc. | Bis-esters of alkanediols |
| US4530792A (en) * | 1982-11-01 | 1985-07-23 | Pfizer Inc. | Process and intermediates for preparation of 1,1-dioxopenicillanoyloxymethyl 6-beta-aminopenicillanate |
| US4462934A (en) | 1983-03-31 | 1984-07-31 | Pfizer Inc. | Bis-esters of dicarboxylic acids with amoxicillin and certain hydroxymethylpenicillanate 1,1-dioxides |
| JPS60214792A (ja) * | 1984-04-06 | 1985-10-28 | Taiho Yakuhin Kogyo Kk | ペナム酸エステル誘導体 |
| CN104650119B (zh) * | 2015-02-10 | 2017-04-05 | 中国科学院长春应用化学研究所 | 一种β‑内酰胺化合物的制备方法 |
| IT202000031070A1 (it) | 2020-12-16 | 2022-06-16 | Paolo Bonomi | Procedimento di sintesi di derivati ammidici dell’acido 8-idrossi penicillanico |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4234579A (en) * | 1977-06-07 | 1980-11-18 | Pfizer Inc. | Penicillanic acid 1,1-dioxides as β-lactamase inhibitors |
| KR830001903B1 (ko) | 1979-02-13 | 1983-09-19 | 레오 파마슈티칼 프로덕츠 리미티드 | 페니실란산유도체의 제조방법 |
| US4325960A (en) * | 1979-02-13 | 1982-04-20 | Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Fabrik Produktionsaktieselskab) | 6-Amidinopenicillanic acid derivatives including the radical of a β-lactamase inhibitor |
| IE49880B1 (en) * | 1979-02-13 | 1986-01-08 | Leo Pharm Prod Ltd | Penicillin derivatives |
| US4244951A (en) * | 1979-05-16 | 1981-01-13 | Pfizer Inc. | Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide |
| US4256733A (en) * | 1979-09-26 | 1981-03-17 | Pfizer Inc. | Acetoxymethyl penam compounds as β-lactamase inhibitors |
-
1981
- 1981-02-20 US US06/236,407 patent/US4364957A/en not_active Expired - Lifetime
-
1982
- 1982-02-05 GR GR67227A patent/GR75173B/el unknown
- 1982-02-12 DE DE8282300704T patent/DE3265503D1/de not_active Expired
- 1982-02-12 EP EP82300704A patent/EP0059046B1/en not_active Expired
- 1982-02-12 AT AT82300704T patent/ATE15044T1/de not_active IP Right Cessation
- 1982-02-18 IE IE342/82A patent/IE52902B1/en unknown
- 1982-02-19 CA CA000396680A patent/CA1176242A/en not_active Expired
- 1982-02-19 DK DK72282A patent/DK72282A/da not_active Application Discontinuation
- 1982-02-19 AU AU80623/82A patent/AU527894B2/en not_active Ceased
- 1982-02-19 JP JP57025821A patent/JPS57154192A/ja active Granted
- 1982-02-19 ES ES509782A patent/ES8304992A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| AU8062382A (en) | 1982-11-04 |
| GR75173B (OSRAM) | 1984-07-13 |
| US4364957A (en) | 1982-12-21 |
| JPS6330312B2 (OSRAM) | 1988-06-17 |
| ES509782A0 (es) | 1983-03-16 |
| EP0059046A1 (en) | 1982-09-01 |
| DE3265503D1 (en) | 1985-09-26 |
| ATE15044T1 (de) | 1985-09-15 |
| EP0059046B1 (en) | 1985-08-21 |
| IE820342L (en) | 1982-08-20 |
| JPS57154192A (en) | 1982-09-22 |
| ES8304992A1 (es) | 1983-03-16 |
| AU527894B2 (en) | 1983-03-31 |
| IE52902B1 (en) | 1988-04-13 |
| CA1176242A (en) | 1984-10-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |