DK71786A - 1,8-naphthyridinderivater med antibakteriel aktivitet - Google Patents

1,8-naphthyridinderivater med antibakteriel aktivitet Download PDF

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Publication number
DK71786A
DK71786A DK71786A DK71786A DK71786A DK 71786 A DK71786 A DK 71786A DK 71786 A DK71786 A DK 71786A DK 71786 A DK71786 A DK 71786A DK 71786 A DK71786 A DK 71786A
Authority
DK
Denmark
Prior art keywords
antibacterial activity
naphthyridine derivatives
naphthyridine
derivatives
antibacterial
Prior art date
Application number
DK71786A
Other languages
Danish (da)
English (en)
Other versions
DK71786D0 (da
Inventor
Jun-Ichi Matsumoto
Junji Nakano
Katsumi Chiba
Shinichi Nakamura
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP60028998A external-priority patent/JPH0635458B2/ja
Priority claimed from JP60084985A external-priority patent/JPS61243081A/ja
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Publication of DK71786D0 publication Critical patent/DK71786D0/da
Publication of DK71786A publication Critical patent/DK71786A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK71786A 1985-02-15 1986-02-14 1,8-naphthyridinderivater med antibakteriel aktivitet DK71786A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP60028998A JPH0635458B2 (ja) 1985-02-15 1985-02-15 ピリドンカルボン酸誘導体、そのエステルおよびその塩
JP60084985A JPS61243081A (ja) 1985-04-19 1985-04-19 ピリドンカルボン酸誘導体、そのエステルおよびその塩

Publications (2)

Publication Number Publication Date
DK71786D0 DK71786D0 (da) 1986-02-14
DK71786A true DK71786A (da) 1986-08-16

Family

ID=26367144

Family Applications (1)

Application Number Title Priority Date Filing Date
DK71786A DK71786A (da) 1985-02-15 1986-02-14 1,8-naphthyridinderivater med antibakteriel aktivitet

Country Status (10)

Country Link
US (1) US4738968A (fi)
EP (1) EP0191451B1 (fi)
KR (1) KR860006462A (fi)
AU (1) AU578793B2 (fi)
DE (1) DE3664774D1 (fi)
DK (1) DK71786A (fi)
ES (1) ES8706144A1 (fi)
FI (1) FI860556A (fi)
HU (1) HUT41784A (fi)
PH (1) PH23723A (fi)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4822801A (en) * 1984-07-20 1989-04-18 Warner-Lambert Company 4-oxo-1,4-dihydroquinoline-3-carboxylic acid derivative as antibacterial agents
US4692454A (en) * 1986-02-03 1987-09-08 Warner-Lambert Company Opthalmic use of quinolone antibiotics
DE3705621C2 (de) * 1986-02-25 1997-01-09 Otsuka Pharma Co Ltd Heterocyclisch substituierte Chinoloncarbonsäurederivate
KR910003630B1 (ko) * 1988-06-17 1991-06-07 한국과학기술원 벤조일 아세틱 에스테르 유도체 및 그 제조방법
CA1332605C (en) * 1988-10-03 1994-10-18 Yasuhiro Nishitani Pyridonecarboxylic acids
DE3918544A1 (de) * 1989-06-07 1990-12-13 Bayer Ag Verfahren zur herstellung von 7-(3-amino- sowie 3-amino-methyl-1-pyrrolidinyl)-3-chinolon- carbonsaeuren sowie -naphthyridoncarbonsaeuren
KR100364226B1 (ko) * 1998-03-18 2003-01-24 주식회사 엘지생명과학 7-할로-1-시클로프로필-6-플루오로-4-옥소-1,4-디히드로-[1.8]나프티리딘-3-카복실레이트의 제조방법
DE19926400A1 (de) * 1999-06-10 2000-12-14 Bayer Ag Verbessertes Verfahren zur Herstellung von 2,6-Dichlor-5-fluor-nicotinsäure und grobteilige und besonders reine 2,6-Dichlor-5-fluor-nicotinsäure
AU2004272414B2 (en) * 2003-09-10 2009-05-28 Kyorin Pharmaceutical Co., Ltd. 7-(4-substituted 3- cyclopropylaminomethyl-1- pyrrolidinyl) quinolonecarboxylic acid derivative
EP1947083B1 (en) * 2005-08-23 2010-11-10 Kaneka Corporation Process for production of aralkyloxypyrrolidine derivative
WO2008143343A1 (ja) * 2007-05-24 2008-11-27 Kyorin Pharmaceutical Co., Ltd. 14位置換基に複素芳香環カルボン酸構造を有するムチリン誘導体
US7902227B2 (en) * 2007-07-27 2011-03-08 Janssen Pharmaceutica Nv. C-7 isoxazolinyl quinolone / naphthyridine derivatives useful as antibacterial agents
KR20120112769A (ko) * 2010-01-08 2012-10-11 교린 세이야꾸 가부시키 가이샤 3,4-2치환 피롤리딘 유도체의 제조 방법 및 제조 중간체

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3963736A (en) * 1970-01-28 1976-06-15 Sumitomo Chemical Company, Limited Preparation of 1-(lower alkyl)-1,4-dihydro-7-methyl-4-oxo-1,8-naphthyridine-3-carboxylic acids
US4382937A (en) * 1981-02-27 1983-05-10 Dainippon Pharmaceutical Co., Ltd. Naphthyridine derivatives and their use as anti-bacterials
US4665079A (en) * 1984-02-17 1987-05-12 Warner-Lambert Company Antibacterial agents
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
EP0160578B1 (en) * 1984-02-17 1989-11-23 Daiichi Seiyaku Co., Ltd. 1,8-naphthyridine derivatives

Also Published As

Publication number Publication date
ES8706144A1 (es) 1987-06-01
AU578793B2 (en) 1988-11-03
ES552032A0 (es) 1987-06-01
FI860556A0 (fi) 1986-02-07
EP0191451B1 (en) 1989-08-02
PH23723A (en) 1989-11-03
US4738968A (en) 1988-04-19
AU5321686A (en) 1986-08-21
HUT41784A (en) 1987-05-28
DE3664774D1 (en) 1989-09-07
DK71786D0 (da) 1986-02-14
EP0191451A1 (en) 1986-08-20
KR860006462A (ko) 1986-09-11
FI860556A (fi) 1986-08-16

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment