DK42490A - Melatoninanaloger - Google Patents

Melatoninanaloger Download PDF

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Publication number
DK42490A
DK42490A DK042490A DK42490A DK42490A DK 42490 A DK42490 A DK 42490A DK 042490 A DK042490 A DK 042490A DK 42490 A DK42490 A DK 42490A DK 42490 A DK42490 A DK 42490A
Authority
DK
Denmark
Prior art keywords
melatonin analogs
melatonin
analogs
Prior art date
Application number
DK042490A
Other languages
English (en)
Other versions
DK42490D0 (da
Inventor
Margarita L Dubocovich
James V Peck
Atef A Helmy
Vithal J Rajadhyaksha
Original Assignee
Nelson Res & Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nelson Res & Dev filed Critical Nelson Res & Dev
Publication of DK42490D0 publication Critical patent/DK42490D0/da
Publication of DK42490A publication Critical patent/DK42490A/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16Tryptamines
DK042490A 1987-08-17 1990-02-16 Melatoninanaloger DK42490A (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8629087A 1987-08-17 1987-08-17
US8606287A 1987-08-17 1987-08-17
PCT/US1988/001859 WO1989001472A1 (en) 1987-08-17 1988-05-20 Melatonin analogues

Publications (2)

Publication Number Publication Date
DK42490D0 DK42490D0 (da) 1990-02-16
DK42490A true DK42490A (da) 1990-04-17

Family

ID=26774333

Family Applications (1)

Application Number Title Priority Date Filing Date
DK042490A DK42490A (da) 1987-08-17 1990-02-16 Melatoninanaloger

Country Status (7)

Country Link
EP (1) EP0375726A4 (da)
KR (1) KR910006124B1 (da)
AU (1) AU616907B2 (da)
DK (1) DK42490A (da)
FI (1) FI900801A0 (da)
NO (1) NO173732C (da)
WO (1) WO1989001472A1 (da)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3402425A (en) * 1964-10-15 1968-09-24 Slagteriernes Forskningsinst Method of wholly or partially cutting out the backbone of open carcasses, such as pigs' carcasses, and apparatus for carrying out this method

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU644367B2 (en) * 1989-05-17 1993-12-09 Applied Medical Research Ltd Use of melatonin derivatives for effecting contraception
US5071875A (en) * 1989-09-25 1991-12-10 Northwestern University Substituted 2-amidotetralins as melatonin agonists and antagonists
IT1251544B (it) * 1991-05-13 1995-05-17 Gabriele Biella Composizioni farmaceutiche attive nella terapia dei disturbi del sonno comprendenti melatonina o un suo derivato in associazione con un derivato benzodiazepinico
FR2680366B1 (fr) * 1991-08-13 1995-01-20 Adir Nouveaux derives d'arylethylamines, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent.
EP0608362A1 (en) * 1991-10-18 1994-08-03 Alza Corporation Device for the transdermal administration of melatonin
US5206377A (en) * 1991-12-05 1993-04-27 Whitby Research, Inc. Compounds useful as antiproliferative agents
IT1255199B (it) * 1992-07-01 1995-10-20 Franco Fraschini Farmaco sintetizzato analogo della melatonina particolarmente efficacenelle patologie che interferiscono con i ritmi circadiani
US5300481A (en) * 1993-05-05 1994-04-05 The Regents Of The University Of California Methods for controlling flowering in plants
US5654325A (en) * 1993-11-18 1997-08-05 Eli Lilly And Company Melatonin derivatives for use in treating sleep disorders
US6180657B1 (en) 1993-11-18 2001-01-30 Eli Lilly And Company Melatonin derivatives for use in treating desynchronization disorders
FR2713636B1 (fr) * 1993-12-07 1996-01-05 Adir Nouveaux dérivés naphtaléniques, leur procédé de préparation, et les compositions pharmaceutiques qui les contiennent.
US5403851A (en) * 1994-04-05 1995-04-04 Interneuron Pharmaceuticals, Inc. Substituted tryptamines, phenalkylamines and related compounds
FR2724170B1 (fr) * 1994-09-02 1997-05-30 Cemaf Nouveaux derives de spiro(indole-pyrrolidine) agonistes de la melatonine, leur procede de preparation et leur utilisation a titre de medicament
FR2718445B1 (fr) * 1994-04-07 1996-06-28 Cemaf Nouveaux dérivés de spiro [indole-pyrrolidine] agonistes de la mélatonine, leur procédé de préparation et leur utilisation à titre de médicament.
EP0754183A1 (fr) * 1994-04-07 1997-01-22 Cemaf Nouveaux derives de spiro[indole-pyrrolidine] agonistes melatoninergiques, leur procede de preparation et leur utilisation a titre de medicament
ES2172415B2 (es) * 2000-07-28 2003-11-16 Univ Madrid Complutense Tratamiento del glaucoma y la hipertension ocular por medio de un analogo de la melatonina.
JP2004518612A (ja) * 2000-07-28 2004-06-24 インスパイアー ファーマシューティカルズ,インコーポレイティド インドール誘導体を用いて眼圧を下降させる方法
JP4175113B2 (ja) 2001-03-14 2008-11-05 小野薬品工業株式会社 Ep1アンタゴニストを有効成分として含有するうつ病の治療剤
FR2874611B1 (fr) * 2004-08-31 2006-11-17 Servier Lab Nouveaux derives d'imidazopyridine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
TW201018695A (en) 2008-07-30 2010-05-16 Ferrer Int 1,6-dihydro-2H-3-oxa-6-aza-as-indacene compounds
KR101534523B1 (ko) * 2013-04-30 2015-07-09 경희대학교 산학협력단 1,2,3,4-테트라히드로-6-메톡시-1-옥소-베타-카르볼린을 포함하는 피부 미백용 화장료 조성물
FR3065225B1 (fr) 2017-04-12 2024-04-05 Patrick Choay Sas Adjuvants depourvus de cytokines pour milieux de culture cellulaire, notamment pour fecondation in vitro, ou pour la culture de follicules, cellules germinales males ou embryons

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3370063A (en) * 1964-10-05 1968-02-20 Mcneilab Inc Substituted dimethoxy indoles and method of making the same
US3915990A (en) * 1973-03-13 1975-10-28 Nelson Res & Dev Tryptamines
US4087444A (en) * 1976-09-08 1978-05-02 Eli Lilly And Company Amides as ovulation inhibitors

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3402425A (en) * 1964-10-15 1968-09-24 Slagteriernes Forskningsinst Method of wholly or partially cutting out the backbone of open carcasses, such as pigs' carcasses, and apparatus for carrying out this method

Also Published As

Publication number Publication date
EP0375726A4 (en) 1991-01-30
KR910006124B1 (ko) 1991-08-13
NO173732C (no) 1994-01-26
EP0375726A1 (en) 1990-07-04
NO173732B (no) 1993-10-18
AU616907B2 (en) 1991-11-14
NO900790D0 (no) 1990-02-19
DK42490D0 (da) 1990-02-16
FI900801A0 (fi) 1990-02-16
KR890701558A (ko) 1989-12-20
AU2309788A (en) 1989-03-09
NO900790L (no) 1990-03-26
WO1989001472A1 (en) 1989-02-23

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Legal Events

Date Code Title Description
AHS Application shelved for other reasons than non-payment