DK424189A - Hemiphosphat-hemihydrat af 2-(1-pentyl-3-guanidino-4-imidazolyl)thiazol - Google Patents

Hemiphosphat-hemihydrat af 2-(1-pentyl-3-guanidino-4-imidazolyl)thiazol

Info

Publication number
DK424189A
DK424189A DK424189A DK424189A DK424189A DK 424189 A DK424189 A DK 424189A DK 424189 A DK424189 A DK 424189A DK 424189 A DK424189 A DK 424189A DK 424189 A DK424189 A DK 424189A
Authority
DK
Denmark
Prior art keywords
guanidino
thiazole
imidazolyl
pentyl
hemiphosphate
Prior art date
Application number
DK424189A
Other languages
Danish (da)
English (en)
Other versions
DK424189D0 (da
Inventor
Troy Anthony Appleton
Ward Marvin Smith
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK424189D0 publication Critical patent/DK424189D0/da
Publication of DK424189A publication Critical patent/DK424189A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Cephalosporin Compounds (AREA)
DK424189A 1988-08-30 1989-08-29 Hemiphosphat-hemihydrat af 2-(1-pentyl-3-guanidino-4-imidazolyl)thiazol DK424189A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US1988/003019 WO1990002127A1 (en) 1988-08-30 1988-08-30 Hemiphosphate hemihydrate of 2-(1-pentyl-3-guanidino-4-imidazolyl)thiazole

Publications (2)

Publication Number Publication Date
DK424189D0 DK424189D0 (da) 1989-08-29
DK424189A true DK424189A (da) 1990-03-01

Family

ID=22208884

Family Applications (1)

Application Number Title Priority Date Filing Date
DK424189A DK424189A (da) 1988-08-30 1989-08-29 Hemiphosphat-hemihydrat af 2-(1-pentyl-3-guanidino-4-imidazolyl)thiazol

Country Status (11)

Country Link
EP (1) EP0357315B1 (cs)
JP (1) JPH02108690A (cs)
AT (1) ATE96794T1 (cs)
CA (1) CA1320207C (cs)
DE (1) DE68910444T2 (cs)
DK (1) DK424189A (cs)
ES (1) ES2059773T3 (cs)
FI (1) FI94248C (cs)
IE (1) IE61736B1 (cs)
PT (1) PT91562B (cs)
WO (1) WO1990002127A1 (cs)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4621424A (en) * 1982-09-17 1986-11-11 The Gillette Company Razor blade assembly
US4560690A (en) * 1984-04-30 1985-12-24 Pfizer Inc. 2-(N-substituted guanidino)-4-hetero-arylthiazole antiulcer agents
US4632993A (en) * 1984-10-11 1986-12-30 Pfizer Inc. Process for making 2-guanidino-4-(2-methyl-4-imidazolyl) thiazole dihydrobromide
DE3750023T2 (de) * 1986-10-29 1994-09-29 Pfizer, Inc., New York, N.Y. Verfahren zur Herstellung von 2-(1-Pentyl-3-guanidino)-4-(2-methyl-4-imidazolyl)Thiazol und dessen kristallinisches Dihydrochlorid-Trihydrat.

Also Published As

Publication number Publication date
IE892765L (en) 1990-02-28
WO1990002127A1 (en) 1990-03-08
ATE96794T1 (de) 1993-11-15
EP0357315B1 (en) 1993-11-03
PT91562A (pt) 1990-03-30
PT91562B (pt) 1995-05-31
EP0357315A3 (en) 1990-08-16
IE61736B1 (en) 1994-11-30
FI94248B (fi) 1995-04-28
CA1320207C (en) 1993-07-13
FI94248C (fi) 1995-08-10
DE68910444D1 (de) 1993-12-09
FI910956A0 (fi) 1991-02-27
JPH02108690A (ja) 1990-04-20
JPH0456038B2 (cs) 1992-09-07
DE68910444T2 (de) 1994-03-03
DK424189D0 (da) 1989-08-29
EP0357315A2 (en) 1990-03-07
ES2059773T3 (es) 1994-11-16

Similar Documents

Publication Publication Date Title
FI904414A7 (fi) Tiatsolidiinidioni-hypoglykeemisesti vaikuttavat aineet
FI912142L (fi) Menetelmä uusien, terapeuttisesti käyttökelpoisten 5-(2-((2-aryyli-2-hydroksietyyli)amino)propyyli)-1,3-bentsodioksolijohdannaisten valmistamiseksi
DK405489A (da) Heterocykliske forbindelser
DK13082A (da) Analogifremgangsmaade til fremstilling af n-(2-pyridyl)-2-methyl-4-hydroxy-2h-1,2-benzothiazin-3-carboxamid-1,1-dioxid-derivater
LV10443A (lv) Heterocikliskie savienojumi
BR9006799A (pt) Compostos heterociclicos
FI812470L (fi) 7-beta-/alfa-syn-metoxi-imino-alfa-(2-aminotiatsol-4-yl)acetamido)-3-((1,2,3-tiadiatsol-5-yltio)metyl)-3-cefem-4-karboxylsyra och dess c1-6-alkylderivat
DK424189A (da) Hemiphosphat-hemihydrat af 2-(1-pentyl-3-guanidino-4-imidazolyl)thiazol
DK155488A (da) Fremgangsmaade til fremstilling af nitroethenderivater
DE3575925D1 (de) Kristalline form von benzothiazindioxydsalz.
DE69014705D1 (de) Thiazol-Derivate.
DK350989A (da) Tiazolderivater
DK507289A (da) Heterocykliske forbindelser
DE69008019D1 (de) Benzothiazol-Derivate.
FI820923A7 (fi) Menetelmä 2-amino-5-(o-sulfamidofenyyli)-1,3,4- tiadiatsolijohdannaisten valmistamiseksi.
FI892034L (fi) Kristallint 2-(1-pentyl-3-guanidino)-4-(2-metyl-4-imidazolyl) tiazoldihydrokloridtrihydrat.
DK565289D0 (da) Heterocykliske forbindelser
FI892035A0 (fi) Foerfaranden foer 2-(1-pentyl-3-guanidino)-4-(2-metyl-4-imidazolyl) tiazol och analoger.
FI883939A7 (fi) Menetelmä (substituoitu tio) alkyyli-isotiosyanaattien valmistamiseksi.
NZ201143A (en) 2-phenethyl-3-aryl(2,3,5,6-tetrahydroimidazo-(2,1-b)-thiazol or 2,3,6,7-tetrahydro-5h-thiazolo (3,2-a) pyrimid)-3-ols
JPS5283837A (en) Aminothiazole derivatives
IT1140281B (it) Procedimento per la preparazione di 4-idrossi-2-metil-n-(2-piridil)-2h-1,2-benzotiazin-3-carbossamide 1,1-diossido
IS3491A7 (is) Ný efnasambönd samtengdra heteróhringa
FI990541A7 (fi) Rikkiä sisältävät heterosykliset yhdisteet
FI882331A0 (fi) Menetelmä terapeuttisesti käyttökelpoisten heterosyklisten sulfonamidien valmistamiseksi

Legal Events

Date Code Title Description
AHB Application shelved due to non-payment