DK207583A - Fremgangsmaade til fremstilling af alfa-substituerede oligopeptider - Google Patents
Fremgangsmaade til fremstilling af alfa-substituerede oligopeptider Download PDFInfo
- Publication number
- DK207583A DK207583A DK207583A DK207583A DK207583A DK 207583 A DK207583 A DK 207583A DK 207583 A DK207583 A DK 207583A DK 207583 A DK207583 A DK 207583A DK 207583 A DK207583 A DK 207583A
- Authority
- DK
- Denmark
- Prior art keywords
- substituted
- oigope
- alfa
- peptides
- procedure
- Prior art date
Links
- 102000004196 processed proteins & peptides Human genes 0.000 title 1
- 108090000765 processed proteins & peptides Proteins 0.000 title 1
- 102000015636 Oligopeptides Human genes 0.000 abstract 1
- 108010038807 Oligopeptides Proteins 0.000 abstract 1
- 230000009286 beneficial effect Effects 0.000 abstract 1
- 210000000170 cell membrane Anatomy 0.000 abstract 1
- 230000000973 chemotherapeutic effect Effects 0.000 abstract 1
- 230000000269 nucleophilic effect Effects 0.000 abstract 1
- 230000035699 permeability Effects 0.000 abstract 1
- 229940002612 prodrug Drugs 0.000 abstract 1
- 239000000651 prodrug Substances 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
- C07K5/0806—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US37953782A | 1982-05-18 | 1982-05-18 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK207583D0 DK207583D0 (da) | 1983-05-10 |
| DK207583A true DK207583A (da) | 1983-11-19 |
Family
ID=23497666
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK207583A DK207583A (da) | 1982-05-18 | 1983-05-10 | Fremgangsmaade til fremstilling af alfa-substituerede oligopeptider |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP0094815B1 (enExample) |
| JP (1) | JPS58219151A (enExample) |
| AT (1) | ATE39930T1 (enExample) |
| AU (2) | AU563196B2 (enExample) |
| CA (1) | CA1247088A (enExample) |
| DE (1) | DE3378914D1 (enExample) |
| DK (1) | DK207583A (enExample) |
| ES (1) | ES522476A0 (enExample) |
| GR (1) | GR81343B (enExample) |
| IE (1) | IE54927B1 (enExample) |
| PT (1) | PT76677B (enExample) |
| ZA (1) | ZA832844B (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4479898A (en) * | 1982-05-18 | 1984-10-30 | Smithkline Beckman Corporation | Oligopeptide prodrugs |
| US5126451A (en) * | 1988-02-11 | 1992-06-30 | Warner-Lambert Company | Renin inhibitors containing α-heteroatom amino acids |
| US5036054A (en) * | 1988-02-11 | 1991-07-30 | Warner-Lambert Company | Renin inhibitors containing alpha-heteroatom amino acids |
| JP2578044B2 (ja) * | 1992-03-14 | 1997-02-05 | 呉羽化学工業株式会社 | フェニルアラニン−グリシン誘導体、その製造方法、及びその誘導体を含有する抗腫瘍剤 |
| FR2736055B1 (fr) * | 1995-06-29 | 1997-09-12 | Laphal Sa Lab | Nouveaux thiophenoxy peptides, leur procede de preparation et les compositions pharmaceutiques en renfermant |
| IT1292438B1 (it) * | 1997-06-30 | 1999-02-08 | Zambon Spa | Derivati peptidomimetici inibitori suicidi della proliferazione del hiv |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH338197A (fr) * | 1954-08-18 | 1959-05-15 | Uclaf Societe Anonyme | Procédé d'obtention de peptides |
| CH616912A5 (en) * | 1974-06-17 | 1980-04-30 | Sandoz Ag | Process for the preparation of dipeptide derivatives. |
| PH14064A (en) * | 1977-05-06 | 1981-01-26 | Pfizer | Phenylgycine derivatives,pharmaceutical compositions and method of use |
| FR2434392A1 (fr) * | 1978-04-28 | 1980-03-21 | Toyo Jozo Kk | Nouveau compose disulfure utile dans la chromatographie de covalence |
| US4258193A (en) * | 1978-07-13 | 1981-03-24 | Toyo Jozo Kabushiki Kaisha | Disulfide derivatives having S--S exchange reactivity |
| IL58849A (en) * | 1978-12-11 | 1983-03-31 | Merck & Co Inc | Carboxyalkyl dipeptides and derivatives thereof,their preparation and pharmaceutical compositions containing them |
| US4284624A (en) * | 1980-05-02 | 1981-08-18 | E. R. Squibb & Sons, Inc. | Mixed disulfides |
| EP0046742B1 (en) * | 1980-08-25 | 1984-06-27 | KabiVitrum AB | Peptide substrates for determination of protease activity |
| JPS5754151A (en) * | 1980-09-18 | 1982-03-31 | Takeda Chem Ind Ltd | Physiologically active substance b-52653 and its preparation |
| CY1406A (en) * | 1980-12-18 | 1988-04-22 | Schering Corp | Substituted dipeptides, processes for their preparation and pharmaceutical compositions containing them and their use in the inhibition of enkephalinase |
| JPS57123155A (en) * | 1981-01-26 | 1982-07-31 | Takeda Chem Ind Ltd | Preparation of pyrrolidine derivative and its intermediate |
| DE3127930A1 (de) * | 1981-07-15 | 1983-01-27 | A. Nattermann & Cie GmbH, 5000 Köln | Neue optisch aktive dipeptide, verfahren zur herstellung und diese enthaltende pharmazeutische praeparate |
| DE3173632D1 (en) * | 1981-09-11 | 1986-03-13 | Amersham Int Plc | Derivatives of iodothyronine compounds and their use in an assay for the free iodothyronine compounds |
| JPS58105948A (ja) * | 1981-12-16 | 1983-06-24 | Fujirebio Inc | ジペプチド誘導体 |
| US4427582A (en) * | 1982-06-08 | 1984-01-24 | Smithkline Beckman Corporation | Antimicrobial disulfide prodrugs |
-
1983
- 1983-04-22 ZA ZA832844A patent/ZA832844B/xx unknown
- 1983-04-22 AU AU13883/83A patent/AU563196B2/en not_active Ceased
- 1983-04-27 CA CA000426790A patent/CA1247088A/en not_active Expired
- 1983-05-10 DK DK207583A patent/DK207583A/da not_active Application Discontinuation
- 1983-05-11 PT PT76677A patent/PT76677B/pt unknown
- 1983-05-16 EP EP83302736A patent/EP0094815B1/en not_active Expired
- 1983-05-16 DE DE8383302736T patent/DE3378914D1/de not_active Expired
- 1983-05-16 AT AT83302736T patent/ATE39930T1/de not_active IP Right Cessation
- 1983-05-17 ES ES522476A patent/ES522476A0/es active Granted
- 1983-05-17 GR GR71370A patent/GR81343B/el unknown
- 1983-05-17 IE IE1144/83A patent/IE54927B1/en unknown
- 1983-05-18 JP JP58088334A patent/JPS58219151A/ja active Pending
-
1987
- 1987-04-16 AU AU71759/87A patent/AU586743B2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| EP0094815A2 (en) | 1983-11-23 |
| CA1247088A (en) | 1988-12-20 |
| IE831144L (en) | 1983-11-18 |
| PT76677B (en) | 1986-01-14 |
| EP0094815B1 (en) | 1989-01-11 |
| AU563196B2 (en) | 1987-07-02 |
| ES8407010A1 (es) | 1984-08-16 |
| DE3378914D1 (en) | 1989-02-16 |
| EP0094815A3 (en) | 1986-03-12 |
| AU586743B2 (en) | 1989-07-20 |
| PT76677A (en) | 1983-06-01 |
| AU7175987A (en) | 1987-08-13 |
| DK207583D0 (da) | 1983-05-10 |
| ZA832844B (en) | 1984-03-28 |
| IE54927B1 (en) | 1990-03-28 |
| AU1388383A (en) | 1983-11-24 |
| GR81343B (enExample) | 1984-12-11 |
| JPS58219151A (ja) | 1983-12-20 |
| ATE39930T1 (de) | 1989-01-15 |
| ES522476A0 (es) | 1984-08-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |