DK207186A - PYRIDINYL PIPERAZINE DERIVATIVES WITH CONDENSED RING SYSTEM - Google Patents

PYRIDINYL PIPERAZINE DERIVATIVES WITH CONDENSED RING SYSTEM

Info

Publication number
DK207186A
DK207186A DK207186A DK207186A DK207186A DK 207186 A DK207186 A DK 207186A DK 207186 A DK207186 A DK 207186A DK 207186 A DK207186 A DK 207186A DK 207186 A DK207186 A DK 207186A
Authority
DK
Denmark
Prior art keywords
ring system
condensed ring
piperazine derivatives
pyridinyl
pyridinyl piperazine
Prior art date
Application number
DK207186A
Other languages
Danish (da)
Other versions
DK165745B (en
DK207186D0 (en
DK165745C (en
Inventor
James Stewart New
Joseph P Yevich
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of DK207186D0 publication Critical patent/DK207186D0/en
Publication of DK207186A publication Critical patent/DK207186A/en
Publication of DK165745B publication Critical patent/DK165745B/en
Application granted granted Critical
Publication of DK165745C publication Critical patent/DK165745C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK207186A 1985-05-06 1986-05-05 PYRIDINYLPIPERAZINE DERIVATIVES WITH CONDENSED RING SYSTEM, PROCEDURES FOR PREPARING THEM AND PHARMACEUTICAL PREPARATIONS CONTAINING THE COMPOUNDS. DK165745C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US73120185A 1985-05-06 1985-05-06
US73120185 1985-05-06

Publications (4)

Publication Number Publication Date
DK207186D0 DK207186D0 (en) 1986-05-05
DK207186A true DK207186A (en) 1986-11-07
DK165745B DK165745B (en) 1993-01-11
DK165745C DK165745C (en) 1993-06-14

Family

ID=24938510

Family Applications (1)

Application Number Title Priority Date Filing Date
DK207186A DK165745C (en) 1985-05-06 1986-05-05 PYRIDINYLPIPERAZINE DERIVATIVES WITH CONDENSED RING SYSTEM, PROCEDURES FOR PREPARING THEM AND PHARMACEUTICAL PREPARATIONS CONTAINING THE COMPOUNDS.

Country Status (25)

Country Link
JP (1) JPH0753728B2 (en)
KR (1) KR940000829B1 (en)
CN (1) CN1017901B (en)
AT (1) AT398572B (en)
AU (1) AU593244B2 (en)
BE (1) BE904724A (en)
CA (1) CA1278792C (en)
CH (1) CH672787A5 (en)
DE (1) DE3615180C2 (en)
DK (1) DK165745C (en)
EG (1) EG18206A (en)
ES (6) ES8801250A1 (en)
FI (1) FI85484C (en)
FR (1) FR2581385B1 (en)
GB (1) GB2174703B (en)
GR (1) GR861149B (en)
HU (1) HU195509B (en)
IE (1) IE59201B1 (en)
IT (1) IT1208607B (en)
LU (1) LU86421A1 (en)
MY (1) MY100777A (en)
NL (1) NL8601146A (en)
PT (1) PT82523B (en)
SE (1) SE465270B (en)
ZA (1) ZA862046B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5801186A (en) 1987-11-20 1998-09-01 Hoechst Marion Roussel, Inc. 3- 4-(1-substituted-4-piperazinyl)butyl!-4-thiazolidinone and related compounds
US4880930A (en) * 1987-11-30 1989-11-14 New James S Psychotropic acyclic amide derivatives
US4780466A (en) * 1988-03-17 1988-10-25 Hoechst-Roussel Pharmaceuticals, Inc. Arylpiperazinylalkoxy derivatives of cyclic imides
IE903410A1 (en) * 1989-10-09 1991-04-10 Novo Nordisk As Indole derivatives, their preparation and use
US5272148A (en) * 1992-09-09 1993-12-21 Hoechst-Roussel Pharmaceuticals Incorporated Heteroarenylpiperazines
FR2738822B1 (en) * 1995-09-15 1997-10-31 Synthelabo DERIVATIVES OF 4- (OMEGA- (4- (THIENO (3,2-C) PYRIDIN-4-YL) PIPERAZIN- 1-YL) ALKYL) QUINOLEIN-2 (1H) -ONE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR2738823B1 (en) * 1995-09-15 1997-10-31 Synthelabo DERIVATIVES OF 3- (OMEGA- (4- (THIENO (3,2-C) PYRIDIN-4-YL) PIPERAZIN- 1-YL) ALKYL) -3,4-DIHYDROQUINOLEIN-2 (1H) -ONE, THEIR PREPARATION AND THEIR APPLICATION IN THERAPEUTICS
BR9610579A (en) * 1995-09-15 1999-07-06 Sanofi Synthelabo Quinoline-2 (1H) -one derivatives as serotonin antagonists
FR2738824B1 (en) * 1995-09-15 1997-10-31 Synthelabo DERIVATIVES OF 3- (OMEGA (4- (THIENO (3,2-C) PYRIDIN-4-YL) PIPERAZIN-1 -YL) ALKYL) -3,4-DIHYDROQUINAZOLIN-2 (1H) -ONE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR2761071B1 (en) * 1997-03-20 1999-12-03 Synthelabo DERIVATIVES OF QUINOLEIN-2 (1H) -ONE AND DIHYDROQUINOLEIN-2 (1H) - ONE, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR2797874B1 (en) * 1999-08-27 2002-03-29 Adir NOVEL PYRIDINE DERIVATIVES, THEIR PREPARATION PROCESS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4367335A (en) * 1981-08-03 1983-01-04 Mead Johnson & Company Thiazolidinylalkylene piperazine derivatives
US4452799A (en) * 1981-12-23 1984-06-05 Mead Johnson & Company Benzisothiazole and benzisoxazole piperazine derivatives
US4361565A (en) * 1981-12-28 1982-11-30 Mead Johnson & Company 2-[4-[(4,4-Dialkyl-2,6-piperidinedion-1-yl)butyl]-1-piperazinyl]pyridines

Also Published As

Publication number Publication date
HU195509B (en) 1988-05-30
ES9000005A1 (en) 1989-11-01
ZA862046B (en) 1986-11-26
ES8900253A1 (en) 1989-05-16
GB2174703B (en) 1988-10-26
CA1278792C (en) 1991-01-08
FR2581385B1 (en) 1991-10-04
LU86421A1 (en) 1986-12-05
GB8610810D0 (en) 1986-06-11
BE904724A (en) 1986-11-05
DE3615180C2 (en) 1996-03-07
ES8802614A1 (en) 1988-09-01
JPS61268681A (en) 1986-11-28
PT82523B (en) 1988-10-14
CN1017901B (en) 1992-08-19
SE465270B (en) 1991-08-19
FI861820A0 (en) 1986-04-30
SE8602061D0 (en) 1986-05-05
ES8801250A1 (en) 1987-12-16
IT1208607B (en) 1989-07-10
ES557757A0 (en) 1988-04-01
CH672787A5 (en) 1989-12-29
FR2581385A1 (en) 1986-11-07
GR861149B (en) 1986-09-09
ES557839A0 (en) 1989-01-16
IE861193L (en) 1986-11-06
FI85484C (en) 1992-04-27
PT82523A (en) 1986-06-01
ES557855A0 (en) 1989-05-16
KR940000829B1 (en) 1994-02-02
DE3615180A1 (en) 1986-11-06
ES8802149A1 (en) 1988-04-01
ES8900138A1 (en) 1989-01-16
SE8602061L (en) 1986-11-07
JPH0753728B2 (en) 1995-06-07
MY100777A (en) 1991-02-14
NL8601146A (en) 1986-12-01
ATA121486A (en) 1994-05-15
ES554659A0 (en) 1987-12-16
IE59201B1 (en) 1994-01-26
DK165745B (en) 1993-01-11
FI85484B (en) 1992-01-15
DK207186D0 (en) 1986-05-05
DK165745C (en) 1993-06-14
CN86103071A (en) 1987-03-18
GB2174703A (en) 1986-11-12
EG18206A (en) 1992-09-30
AU593244B2 (en) 1990-02-08
AT398572B (en) 1994-12-27
KR860009008A (en) 1986-12-19
HUT43848A (en) 1987-12-28
ES557809A0 (en) 1988-09-01
IT8620313A0 (en) 1986-05-06
FI861820A (en) 1986-11-07
AU5679586A (en) 1986-11-13

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Legal Events

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PUP Patent expired