DK156771C - Bis-dioxopiperazin-derivater med antitumor-aktivitet og laegemiddelformuleringer indeholdende saadanne forbindelser - Google Patents
Bis-dioxopiperazin-derivater med antitumor-aktivitet og laegemiddelformuleringer indeholdende saadanne forbindelserInfo
- Publication number
- DK156771C DK156771C DK060187A DK60187A DK156771C DK 156771 C DK156771 C DK 156771C DK 060187 A DK060187 A DK 060187A DK 60187 A DK60187 A DK 60187A DK 156771 C DK156771 C DK 156771C
- Authority
- DK
- Denmark
- Prior art keywords
- bis
- compounds
- pharmaceutical formulations
- formulations containing
- antitumor activity
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
- C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP13973185 | 1985-06-26 | ||
JP13973185 | 1985-06-26 | ||
PCT/JP1986/000324 WO1987000170A1 (en) | 1985-06-26 | 1986-06-25 | Bis-dioxopiperazine derivatives and drug composition containing same |
JP8600324 | 1986-06-25 |
Publications (4)
Publication Number | Publication Date |
---|---|
DK60187D0 DK60187D0 (da) | 1987-02-05 |
DK60187A DK60187A (da) | 1987-03-20 |
DK156771B DK156771B (da) | 1989-10-02 |
DK156771C true DK156771C (da) | 1990-03-19 |
Family
ID=15252071
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK060187A DK156771C (da) | 1985-06-26 | 1987-02-05 | Bis-dioxopiperazin-derivater med antitumor-aktivitet og laegemiddelformuleringer indeholdende saadanne forbindelser |
Country Status (7)
Country | Link |
---|---|
US (1) | US4877803A (da) |
EP (1) | EP0230474B1 (da) |
JP (1) | JPH0676392B2 (da) |
AU (1) | AU584448B2 (da) |
DE (1) | DE3673801D1 (da) |
DK (1) | DK156771C (da) |
WO (1) | WO1987000170A1 (da) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH0674251B2 (ja) * | 1986-02-07 | 1994-09-21 | 全薬工業株式▲会▼社 | ビス−ジオキソピペラジン誘導体 |
FR2601364B1 (fr) * | 1986-07-09 | 1988-10-21 | Adir | Nouveaux derives de la piperazine dione-2,6, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent. |
EP0491053B1 (en) * | 1990-07-04 | 1996-02-07 | Zenyaku Kogyo Kabushikikaisha | Water-soluble bis-dioxopiperazine derivatives with antitumoral properties |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS59190976A (ja) * | 1983-04-12 | 1984-10-29 | Zenyaku Kogyo Kk | ビス−ジオキソピペラジン誘導体、その製造方法及びそれからなる抗腫瘍剤 |
US4737497A (en) * | 1983-04-12 | 1988-04-12 | Zenyaki Kogyo Kabushiki Kaisha | Bis-dioxopiperazine derivatives, antitumor agents comprising them and compositions containing them |
-
1986
- 1986-06-23 JP JP61146591A patent/JPH0676392B2/ja not_active Expired - Lifetime
- 1986-06-25 EP EP86904348A patent/EP0230474B1/en not_active Expired - Lifetime
- 1986-06-25 AU AU61219/86A patent/AU584448B2/en not_active Ceased
- 1986-06-25 US US07/031,011 patent/US4877803A/en not_active Expired - Fee Related
- 1986-06-25 DE DE8686904348T patent/DE3673801D1/de not_active Expired - Fee Related
- 1986-06-25 WO PCT/JP1986/000324 patent/WO1987000170A1/ja active IP Right Grant
-
1987
- 1987-02-05 DK DK060187A patent/DK156771C/da not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
EP0230474A1 (en) | 1987-08-05 |
DK60187D0 (da) | 1987-02-05 |
EP0230474B1 (en) | 1990-08-29 |
US4877803A (en) | 1989-10-31 |
WO1987000170A1 (en) | 1987-01-15 |
DE3673801D1 (de) | 1990-10-04 |
EP0230474A4 (en) | 1987-10-01 |
AU584448B2 (en) | 1989-05-25 |
DK60187A (da) | 1987-03-20 |
AU6121986A (en) | 1987-01-30 |
JPS6289668A (ja) | 1987-04-24 |
JPH0676392B2 (ja) | 1994-09-28 |
DK156771B (da) | 1989-10-02 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NZ216793A (en) | Phenethanolaminotetraline derivatives and pharmaceutical compositions | |
PH24833A (en) | Ascorbic acid derivatives and pharmaceutical composition thereof | |
DK127787A (da) | Interleukin-1alfa-derivater og medikamenter indeholdende saadanne derivater | |
DK163923C (da) | 2-phenyl-3-aminomethyl-imidazooe1,2-aaapyridinderivater og farmaceutisk praeparat indeholdende saadanne forbindelser | |
NZ216951A (en) | Pyrimidine derivatives and pharmaceutical compositions | |
DK475684A (da) | Phenothiazinderivater og farmaceutiske praeparater indeholdende phenothiazinderivaterne | |
DK272486D0 (da) | Tienopyridoner og farmaceutiske praeparater indeholdende dem | |
DK497685A (da) | Ketongruppeholdige oxindol-3-carboxamid-derivater og laegemiddel indeholdende saadanne derivater | |
DK64795A (da) | Cephemderivat og fremgangsmåde til fremstilling deraf | |
NZ217220A (en) | Guanine derivatives and pharmaceutical compositions | |
NZ215871A (en) | Fluorinated phenylalkyl-triazole derivatives and pharmaceutical compositions | |
DK272386A (da) | Quinoloner og farmaceutiske praeparater indeholdende dem | |
NZ217078A (en) | N-piperidyl-benzamide derivatives and pharmaceutical compositions | |
NZ216894A (en) | Penicillin derivatives and pharmaceutical compositions | |
IL86711A0 (en) | 5-pyrimidinecarboxamide derivatives and pharmaceutical compositions containing them | |
NZ218498A (en) | Fluoroalkylamine derivatives and pharmaceutical compositions | |
NZ216720A (en) | Diazinylpiperidine derivatives and pharmaceutical compositions | |
DK52086A (da) | Farmaceutiske praeparater indeholdende ergotalkaloider | |
DK196885D0 (da) | Farmaceutiske praeparater indeholdende isoquinolinderivater og isoquinolinderivater indeholdende saadanne derivater | |
DK269289A (da) | Cyklopentanderivater og farmaceutiske praeparater indeholdende saadanne forbindelser | |
NZ215879A (en) | Quinolizine derivatives and pharmaceutical compositions | |
DK156771C (da) | Bis-dioxopiperazin-derivater med antitumor-aktivitet og laegemiddelformuleringer indeholdende saadanne forbindelser | |
NZ214815A (en) | 12-aminopyridazinopyrroloisoquinoline derivatives and pharmaceutical compositions | |
NZ216946A (en) | Penicillin derivatives and pharmaceutical compositions | |
DK35889D0 (da) | Vitamin d3 derivater og farmaceutiske praeparater indeholdende disse forbindelser |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
PBP | Patent lapsed |